Design, synthesis and biological evaluation of FLT3 covalent inhibitors with a resorcylic acid core von Xu, Jin, Ong, Esther H.Q., Hill, Jeffrey, Chen, Anqi, Chai, Christina L.L.

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Structure–Activity Relationship Studies of Mitogen Activated Protein Kinase Interacting Kinase (MNK) 1 and 2 and BCR-ABL1 Inhibitors Targeting Chronic Myeloid Leukemic Cells von Cherian, Joseph, Nacro, Kassoum, Poh, Zhi Ying, Guo, Samantha, Jeyaraj, Duraiswamy A, Wong, Yun Xuan, Ho, Melvyn, Yang, Hai Yan, Joy, Joma Kanikadu, Kwek, Zekui Perlyn, Liu, Boping, Wee, John Liang Kuan, Ong, Esther HQ, Choong, Meng Ling, Poulsen, Anders, Lee, May Ann, Pendharkar, Vishal, Ding, Li Jun, Manoharan, Vithya, Chew, Yun Shan, Sangthongpitag, Kanda, Lim, Sharon, Ong, S. Tiong, Hill, Jeffrey, Keller, Thomas H

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Deep learning for de-convolution of Smad2 versus Smad3 binding sites von Ng, Jeremy W.K, Ong, Esther H.Q, Tucker-Kellogg, Lisa, Tucker-Kellogg, Greg

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Designing a leucine‐rich antibacterial nonapeptide with potent activity against mupirocin‐resistant MRSA via a structure–activity relationship study von Ang, Qi An, Arfan, Giovinna, Ong, Chu Yang Fann, Ng, Fui Mee, Ong, Esther H. Q., Chia, Cheng San Brian

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An FDA-Drug Library Screen for Compounds with Bioactivities against Meticillin-Resistant Staphylococcus aureus (MRSA) von Lau, Qiu Ying, Tan, Yoke Yan Fion, Goh, Vanessa Chai Yin, Lee, David Jing Qin, Ng, Fui Mee, Ong, Esther H Q, Hill, Jeffrey, Chia, Cheng San Brian

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An industry perspective approach and control strategy for implementation of ready-to-use cells in bioassays: survey outcome and recommendations von White, John R, Ahmed, Sammina, Amstrup, Jan, Bennington, Petra, Cheng, Zhijie Jey, Day, Peter, Haenssen, Keneshia K, Kozminsky-Atias, Adi, Martinez, Eva, Ong, Esther Hq, Qahwash, Isam, Stokes, Elaine Se, Wang, Jenny

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Fragment-Based Drug Discovery of Potent Protein Kinase C Iota Inhibitors von Kwiatkowski, Jacek, Liu, Boping, Tee, Doris Hui Ying, Chen, Guoying, Ahmad, Nur Huda Binte, Wong, Yun Xuan, Poh, Zhi Ying, Ang, Shi Hua, Tan, Eldwin Sum Wai, Ong, Esther HQ, Nurul Dinie, Poulsen, Anders, Pendharkar, Vishal, Sangthongpitag, Kanda, Lee, May Ann, Sepramaniam, Sugunavathi, Ho, Soo Yei, Cherian, Joseph, Hill, Jeffrey, Keller, Thomas H, Hung, Alvin W

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Rational Design of Resorcylic Acid Lactone Analogues as Covalent MNK1/2 Kinase Inhibitors by Tuning the Reactivity of an Enamide Michael Acceptor von Xu, Jin, Chen, Anqi, Joy, Joma, Xavier, Vanessa Joanne, Ong, Esther H. Q., Hill, Jeffrey, Chai, Christina L. L.

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3-Deazaneplanocin A and Neplanocin A Analogues and Their Effects on Apoptotic Cell Death von Tam, Eric K. W., Nguyen, Tuan Minh, Lim, Cheryl Z. H., Lee, Puay Leng, Li, Zhimei, Jiang, Xia, Santhanakrishnan, Sridhar, Tan, Tiong Wei, Goh, Yi Ling, Wong, Sze Yue, Yang, Haiyan, Ong, Esther H. Q., Hill, Jeffrey, Yu, Qiang, Chai, Christina L. L.

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Fragment-based Discovery of a Small-Molecule Protein Kinase C‑iota Inhibitor Binding Post-kinase Domain Residues von Kwiatkowski, Jacek, Baburajendran, Nithya, Poulsen, Anders, Liu, Boping, Tee, Doris Hui Ying, Wong, Yun Xuan, Poh, Zhi Ying, Ong, Esther HQ, Dinie, Nurul, Cherian, Joseph, Jansson, Anna Elisabet, Hill, Jeffrey, Keller, Thomas H, Hung, Alvin W

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Screening for a Potent Antibacterial Peptide to Treat Mupirocin-Resistant MRSA Skin Infections von Ng, Siew Mei Samantha, Ching, Hui Si Vivian, Xu, GuiFang, Ng, Fui Mee, Ong, Esther H. Q., Lau, Qiu Ying, Jureen, Roland, Hill, Jeffrey, Chia, C. S. Brian

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3-DeazaneplanocinA and NeplanocinA Analogues and Their Effects on Apoptotic Cell Death von Tam, Eric K W, Nguyen, Tuan Minh, Lim, Cheryl Z H, Lee, Puay Leng, Li, Zhimei, Jiang, Xia, Santhanakrishnan, Sridhar, Tan, Tiong Wei, Goh, Yi Ling, Wong, Sze Yue, Yang, Haiyan, Ong, Esther H Q, Hill, Jeffrey, Yu, Qiang, Chai, Christina L L

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