Epi-Cyclophellitol Cyclosulfate, a Mechanism-Based Endoplasmic Reticulum α‑Glucosidase II Inhibitor, Blocks Replication of SARS-CoV‑2 and Other Coronaviruses von Thaler, Melissa, Ofman, Tim P., Kok, Ken, Heming, Jurriaan J. A., Moran, Elisha, Pickles, Isabelle, Leijs, Anouk A., van den Nieuwendijk, Adrianus M. C. H., van den Berg, Richard J. B. H. N., Ruijgrok, Gijs, Armstrong, Zachary, Salgado-Benvindo, Clarisse, Ninaber, Dennis K., Snijder, Eric J., van Boeckel, Constant A. A., Artola, Marta, Davies, Gideon J., Overkleeft, Herman S., van Hemert, Martijn J.

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Design and Synthesis of Exocyclic Cyclitol Aziridines as Potential Mechanism‐Based Glycosidase Inactivators von Ofman, Tim P., Marel, Gijsbert A., Codée, Jeroen D. C., Overkleeft, Hermen S.

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An Orthogonally Protected Cyclitol for the Construction of Nigerose- and Dextran-Mimetic Cyclophellitols von Ofman, Tim P, Küllmer, Florian, van der Marel, Gijsbert A, Codée, Jeroen D. C, Overkleeft, Herman S

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Structure–Activity Relationship Studies of α‑Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family von Zhou, Juan, Mock, Elliot D, Al Ayed, Karol, Di, Xinyu, Kantae, Vasudev, Burggraaff, Lindsey, Stevens, Anna F, Martella, Andrea, Mohr, Florian, Jiang, Ming, van der Wel, Tom, Wendel, Tiemen J, Ofman, Tim P, Tran, Yvonne, de Koster, Nicky, van Westen, Gerard J.P, Hankemeier, Thomas, van der Stelt, Mario

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Reactivity–Stereoselectivity Mapping for the Assembly of Mycobacterium marinum Lipooligosaccharides von Hansen, Thomas, Ofman, Tim P., Vlaming, Joey G. C., Gagarinov, Ivan A., Beek, Jessey, Goté, Tessa A., Tichem, Jacoba M., Ruijgrok, Gijs, Overkleeft, Herman S., Filippov, Dmitri V., Marel, Gijsbert A., Codée, Jeroen D. C.

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Conformational and Electronic Variations in 1,2‐ and 1,5a‐Cyclophellitols and their Impact on Retaining α‐Glucosidase Inhibition von Ofman, Tim P., Heming, Jurriaan J. A., Nin‐Hill, Alba, Küllmer, Florian, Moran, Elisha, Bennett, Megan, Steneker, Roy, Klein, Anne‐Mei, Ruijgrok, Gijs, Kok, Ken, Armstrong, Zach W. B., Aerts, Johannes M. F. G., Marel, Gijsbert A., Rovira, Carme, Davies, Gideon J., Artola, Marta, Codée, Jeroen D. C., Overkleeft, Herman S.

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Reactivity–Stereoselectivity Mapping for the Assembly of Mycobacterium marinum Lipooligosaccharides von Hansen, Thomas, Ofman, Tim P., Vlaming, Joey G. C., Gagarinov, Ivan A., Beek, Jessey, Goté, Tessa A., Tichem, Jacoba M., Ruijgrok, Gijs, Overkleeft, Herman S., Filippov, Dmitri V., Marel, Gijsbert A., Codée, Jeroen D. C.

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Epi-cyclophellitol cyclosulfate, a mechanism-based ER α-glucosidase II inhibitor, blocks replication of SARS-CoV-2 and other coronaviruses von Thaler, Melissa, Ofman, Tim P, Kok, Ken, Heming, Jurriaan J.A, Moran, Elisha, Pickles, Isabelle, Leijs, Anouk A, Nieuwendijk, Adrianus M. C. H. van den, Berg, Richard J. B. H. N van den, Ruijgrok, Gijs, Armstrong, Zach, Salgado-Benvindo, Clarisse, Ninaber, Dennis K, Snijder, Eric J, Boeckel, Constant A. A. van, Artola, Marta, Davies, Gideon J, Overkleeft, Herman S, Hemert, Martijn J. van

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Conformational and Electronic Variations in 1,2- and 1,6-Cyclophellitols and Their Impact on Retaining α-Glucosidase Inhibition von Ofman, Tim P, Heming, Jurriaan J. A, Nin-Hill, Alba, Küllmer, Florian, Moran, Elisha, Bennett, Megan, Steneker, Roy, Klein, Anne-Mei, Ruijgrok, Gijs, Kok, Ken, Armstrong, Zach W. B, Aerts, Johannes M. F. G, van der Marel, Gijsbert A, Rovira, Carme, Davies, Gideon J, Artola, Marta, Codée, Jeroen D. C, Overkleeft., Herman S

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