Discovery and mechanistic study of thiazole-4-acylsulfonamide derivatives as potent and orally active ChemR23 inhibitors with a long-acting effect in cynomolgus monkeys von Imaizumi, Takamichi, Otsubo, Shigeki, Maemoto, Michihiro, Kobayashi, Atsuko, Komai, Masato, Takada, Hidenori, Sakaida, Yumi, Otsubo, Nobumasa

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The design, synthesis and evaluation of 2-aminobenzoxazole analogues as potent and orally efficacious ChemR23 inhibitors von Imaizumi, Takamichi, Otsubo, Shigeki, Komai, Masato, Takada, Hidenori, Maemoto, Michihiro, Kobayashi, Atsuko, Otsubo, Nobumasa

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Corrigendum to “Discovery and mechanistic study of thiazole-4-acylsulfonamide derivatives as potent and orally active ChemR23 inhibitors with a long-acting effect in cynomolgus mon... von Imaizumi, Takamichi, Otsubo, Shigeki, Maemoto, Michihiro, Kobayashi, Atsuko, Komai, Masato, Takada, Hidenori, Sakaida, Yumi, Otsubo, Nobumasa

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The discovery and optimization of a series of 2-aminobenzoxazole derivatives as ChemR23 inhibitors von Imaizumi, Takamichi, Kobayashi, Atsuko, Otsubo, Shigeki, Komai, Masato, Magara, Megumiko, Otsubo, Nobumasa

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The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma von Kaneda, Ayumi, Seike, Toshihiro, Danjo, Tomohiro, Nakajima, Takahiro, Otsubo, Nobumasa, Yamaguchi, Daisuke, Tsuji, Yoshiro, Hamaguchi, Kaori, Yasunaga, Mai, Nishiya, Yoichi, Suzuki, Michihiko, Saito, Jun-Ichi, Yatsunami, Rie, Nakamura, Satoshi, Sekido, Yoshitaka, Mori, Kiyotoshi

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Abstract 3086: Discovery of a first-in-class TEAD inhibitor which directly inhibits YAP/TAZ-TEAD protein-protein interaction and shows a potent anti-tumor effect in malignant pleur... von Kaneda, Ayumi, Seike, Toshihiro, Uemori, Takeshi, Myojo, Kensuke, Aida, Kensuke, Danjo, Tomohiro, Nakajima, Takahiro, Yamaguchi, Daisuke, Hamada, Tomoko, Tsuji, Yoshiro, Hamaguchi, Kaori, Yasunaga, Mai, Otsubo, Nobumasa, Onodera, Hideyuki, Nishiya, Yoichi, Suzuki, Michihiko, Saito, Junichi, Ishii, Toshihiko, Nakai, Ryuichiro

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In vivo programming of endogenous antibodies via oral administration of adaptor ligands von Nagano, Masanobu, Carrillo, Nancy, Otsubo, Nobumasa, Hakamata, Wataru, Ban, Hitoshi, Fuller, Roberta P., Bashiruddin, Nasir K., Barbas, Carlos F.

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Chemically Programmed Antibodies As HIV‑1 Attachment Inhibitors von Sato, Shinichi, Inokuma, Tsubasa, Otsubo, Nobumasa, Burton, Dennis R, Barbas, Carlos F

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Potent Inhibition of HIV-1 Entry with a Chemically Programmed Antibody Aided by an Efficient Organocatalytic Synthesis von Gavrilyuk, Julia, Uehara, Hisatoshi, Otsubo, Nobumasa, Hessell, Ann, Burton, Dennis R, Barbas, Carlos F. III

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Chemoenzymatic synthesis of ganglioside GM4 analogs as potential immunosuppressive agents von Zhang, X, Kamiya, T, Otsubo, N, Ishida, H, Kiso, M

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Design and synthesis of a novel neo-glycolipid containing sialyl Lewis X determinant carried on the mucin GlcNAcβ1-6GalNAcα core structure von Otsubo, Nobumasa, Ishida, Hideharu, Kannagi, Reiji, Kiso, Makoto

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ALPHA.,.BETA.-UNSATURATED AMIDE COMPOUND von OTSUBO, NOBUMASA, FUJIWARA, KATSUAKI, SEIKE, TOSHIHIRO, NISHIKAWA, TOMOYUKI, NAKAJIMA, TAKAHIRO, DANJO, TOMOHIRO

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a, ß unsaturated amide compound von NAKAJIMA, Takahiro, NISHIKAWA, Tomoyuki, FUJIWARA, Katsuaki, DANJO, Tomohiro, SEIKE, Toshihiro, OTSUBO, Nobumasa

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a, ß unsaturated amide compound von NAKAJIMA, Takahiro, NISHIKAWA, Tomoyuki, FUJIWARA, Katsuaki, DANJO, Tomohiro, SEIKE, Toshihiro, OTSUBO, Nobumasa

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(),()-UNSATURATED AMIDE COMPOUND von NISHIKAWA TOMOYUKI, OTSUBO NOBUMASA, NAKAJIMA TAKAHIRO, FUJIWARA KATSUAKI, SEIKE TOSHIHIRO, DANJO TOMOHIRO

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Specific Detection of Sialyl Lewis X Determinant Carried on the Mucin GlcNAcβ1→6GalNAcα Core Structure as a Tumor-Associated Antigen von Kumamoto, Kensuke, Mitsuoka, Chikako, Izawa, Mineko, Kimura, Naoko, Otsubo, Nobumasa, Ishida, Hideharu, Kiso, Makoto, Yamada, Tesshi, Hirohashi, Setsuo, Kannagi, Reiji

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Synthesis of novel ganglioside GM4 analogues containing N-deacetylated and lactamized sialic acid: probes for searching new ligand structures for human L-selectin von Otsubo, Nobumasa, Ishida, Hideharu, Kiso, Makoto

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The first, highly efficient synthesis of spacer-armed O-glycans on GlyCAM-1 and PSGL-1: the counter-receptors for L- and P-selectin von Otsubo, Nobumasa, Ishida, Hideharu, Kiso, Makoto

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α,β-unsaturated amide compound von Nishikawa, Tomoyuki, Nakajima, Takahiro, Fujiwara, Katsuaki, Otsubo, Nobumasa, Danjo, Tomohiro, Seike, Toshihiro

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ALPHA,BETA-UNSATURATED AMIDE COMPOUND von NAKAJIMA, Takahiro, NISHIKAWA, Tomoyuki, FUJIWARA, Katsuaki, DANJO, Tomohiro, SEIKE, Toshihiro, OTSUBO, Nobumasa

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