Novel Vanilloid Receptor-1 Antagonists:  2. Structure−Activity Relationships of 4-Oxopyrimidines Leading to the Selection of a Clinical Candidate von Doherty, Elizabeth M, Fotsch, Christopher, Bannon, Anthony W, Bo, Yunxin, Chen, Ning, Dominguez, Celia, Falsey, James, Gavva, Narender R, Katon, Jodie, Nixey, Thomas, Ognyanov, Vassil I, Pettus, Liping, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Zhu, Jiawang, Treanor, James J. S, Norman, Mark H

Volltext

Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure−Activity Relationships of 2-Piperazin-1-yl-1H-benzimidazoles von Ognyanov, Vassil I, Balan, Chenera, Bannon, Anthony W, Bo, Yunxin, Dominguez, Celia, Fotsch, Christopher, Gore, Vijay K, Klionsky, Lana, Ma, Vu V, Qian, Yi-Xin, Tamir, Rami, Wang, Xianghong, Xi, Ning, Xu, Shimin, Zhu, Dawn, Gavva, Narender R, Treanor, James J. S, Norman, Mark H

Volltext

Discovery of Potent, Orally Available Vanilloid Receptor-1 Antagonists. Structure−Activity Relationship of N-Aryl Cinnamides von Doherty, Elizabeth M, Fotsch, Christopher, Bo, Yunxin, Chakrabarti, Partha P, Chen, Ning, Gavva, Narender, Han, Nianhe, Kelly, Michael G, Kincaid, John, Klionsky, Lana, Liu, Qingyian, Ognyanov, Vassil I, Tamir, Rami, Wang, Xianghong, Zhu, Jiawang, Norman, Mark H, Treanor, James J. S

Volltext

Novel Vanilloid Receptor-1 Antagonists:  1. Conformationally Restricted Analogues of trans-Cinnamides von Norman, Mark H, Zhu, Jiawang, Fotsch, Christopher, Bo, Yunxin, Chen, Ning, Chakrabarti, Partha, Doherty, Elizabeth M, Gavva, Narender R, Nishimura, Nobuko, Nixey, Thomas, Ognyanov, Vassil I, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Viswanadhan, Vellarkad N, Treanor, James J. S

Volltext

Trisubstituted pyrimidines as transient receptor potential vanilloid 1 (TRPV1) antagonists with improved solubility von Wang, Xianghong, Chakrabarti, Partha P., Ognyanov, Vassil I., Pettus, Liping H., Tamir, Rami, Tan, Helming, Tang, Phi, Treanor, James J.S., Gavva, Narender R., Norman, Mark H.

Volltext

Preparation of chiral cyanohydrins by an oxynitrilase-mediated transcyanation von Ognyanov, Vassil I, Datcheva, Violeta K, Kyler, Keith S

Volltext

Deoxygenated inositol 1,4,5-trisphosphate analogs and their interaction with metabolic enzymes. (1R,2R,4R)-Cyclohexane-1,2,4-tris(methylenesulfonate): a potent selective 5-phosphat... von Kozikowski, Alan P, Ognyanov, Vassil I, Chen, Chinpiao, Fauq, Abdul H, Safrany, Stephen T, Wilcox, Robert A, Nahorski, Stefan R

Volltext

Palladium-Catalyzed Synthesis of 2-Allyl-2-nitrocycloalkanones von Ognyanov, Vassil I., Hesse, Manfred

Volltext

Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure−Activity Relationships of 2-Piperazin-1-yl-1 H -benzimidazoles von Ognyanov, Vassil I., Balan, Chenera, Bannon, Anthony W., Bo, Yunxin, Dominguez, Celia, Fotsch, Christopher, Gore, Vijay K., Klionsky, Lana, Ma, Vu V., Qian, Yi-Xin, Tamir, Rami, Wang, Xianghong, Xi, Ning, Xu, Shimin, Zhu, Dawn, Gavva, Narender R., Treanor, James J. S., Norman, Mark H.

Volltext

Synthesis of 1H,2,3-Triazoles from 2-Substituted Cyclododecanones and Phenyl Azide von Ognyanov, Vassil I., Hesse, Manfred

Volltext

Synthesis of macrocyclic enaminolactams by ring expansion reaction of 2-oxocyclododecane-1-carbonitrile with diarylcarbodiimides von Ivancev, Wladislaw, Ognyanov, Vassil I., Hesse, Manfred

Volltext

1D-myo-inositol 1,4,5-trisphosphate and 1D-myo-inositol 1,3,4,5-tetrakisphosphate analogues modified at C-3; synthesis of 1D-3-C-(trifluoromethyl)-myo-inositol 1,4,5-trisphosphate... von Kozikowski, Alan P., Ognyanov, Vassil I., Fauq, Abdul H., Wilcox, Robert A., Nahorski, Stefan R.

Volltext

Synthesis of 1 H ,2,3‐Triazoles from 2‐Substituted Cyclododecanones and Phenyl Azide von Ognyanov, Vassil I., Hesse, Manfred

Volltext

Probing the D-1,4,5-IP3/D-1,3,4,5-IP4 functional interface. Synthesis and pharmacology of novel D-3-modified myo-inositol trisphosphate analogues von FAUQ, A. H, KOZIKOWSKI, A. P, OGNYANOV, V. I, WILCOX, R. A, NAHORSKI, S. R

Volltext

Synthese von Makrocyclen durch Ringerweiterung von 14gliedrigen cyclischen Imiden von Koch, Thomas, Ognyanov, Vassil I., Hesse, Manfred

Volltext

Glycine transport inhibitors: A new class of antipsychotics? von Borden, Laurence A., Bell, Stanley C., Ognyanov, Vassil I., Albert, Vivian R., Zhang, Jing, De Vivo, Michael, Yokoyama, Midori, Xie, Xiaping, Berger, Theodore, Gerhardt, Greg, McKelvy, Jeffrey F.

Volltext

Synthesis of macrocyclic imides by one-step ring enlargement von Ognyanov, Vassil I., Hesse, Manfred

Volltext

Cycloalkylations of N-(ω-Halogenoalkyl)-substituted Macrocyclic Imides von Ognyanov, Vassil I., Hesse, Manfred

Volltext

Vanilloid receptor ligands and their use in treatments von Chen, Ning, Nishimura, Nobuko, Norman, Mark H, Ognyanov, Vassil I

Volltext bestellen

Vanilloid receptor ligands and their use in treatments von NISHIMURA NOBUKO, OGNYANOV VASSIL I, CHEN NING, NORMAN MARK H

Volltext bestellen