Co-expression of GRK2 reveals a novel conformational state of the µ-opioid receptor von Nickolls, Sarah A, Humphreys, Sian, Clark, Mellissa, McMurray, Gordon

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Residues W320 and Y328 within the binding site of the μ-opioid receptor influence opiate ligand bias von Hothersall, J. Daniel, Torella, Rubben, Humphreys, Sian, Hooley, Monique, Brown, Alastair, McMurray, Gordon, Nickolls, Sarah A.

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Design and Identification of a Novel, Functionally Subtype Selective GABA A Positive Allosteric Modulator (PF-06372865) von Owen, Robert M, Blakemore, David, Cao, Lishuang, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R, Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A, Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C, Reynolds, David S, Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S, Watson, Christine

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Functional coupling of the human dopamine D 2 receptor with Gα i1 , Gα i2 , Gα i3 and Gα o G proteins: evidence for agonist regulation of G protein selectivity von Gazi, Lucien, Nickolls, Sarah A, Strange, Philip G

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Design and Identification of a Novel, Functionally Subtype Selective GABAA Positive Allosteric Modulator (PF-06372865) von Owen, Robert M, Blakemore, David, Cao, Lishuang, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R, Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A, Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C, Reynolds, David S, Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S, Watson, Christine

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Pharmacology in translation: the preclinical and early clinical profile of the novel α2/3 functionally selective GABAA receptor positive allosteric modulator PF‐06372865 von Nickolls, Sarah A, Gurrell, Rachel, Amerongen, Guido, Kammonen, Juha, Cao, Lishuang, Brown, Adam R, Stead, Clara, Mead, Andy, Watson, Christine, Hsu, Cathleen, Owen, Robert M, Pike, Andy, Fish, Rebecca L, Chen, Laigao, Qiu, Ruolun, Morris, Evan D, Feng, Gang, Whitlock, Mark, Gorman, Donal, Gerven, Joop, Reynolds, David S, Dua, Pinky, Butt, Richard P

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A potential role for cannabinoid receptors in the therapeutic action of fenofibrate von Priestley, Richard S., Nickolls, Sarah A., Alexander, Stephen P. H., Kendall, David A.

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Identification of CC Chemokine Receptor 7 Residues Important for Receptor Activation von Ott, Thomas R, Pahuja, Anil, Nickolls, Sarah A, Alleva, David G, Struthers, R Scott

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The influence of G protein subtype on agonist action at D2 dopamine receptors von Nickolls, Sarah A, Strange, Philip G

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Understanding the Effect of Different Assay Formats on Agonist Parameters: A Study Using the µ-Opioid Receptor von Nickolls, Sarah A., Waterfield, Alison, Williams, Rachael E., Kinloch, Ross A.

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Identification of a novel BODIPY minihepcidin tool for the high content analysis of ferroportin (SLC40A1) pharmacology von Skerratt, Sarah. E, Humphreys, Sian, Ferreira, Rita, Jorgensen, Csilla, Warmus, Joe, Zhao, Lei, Tong, Xiaohe, Nickolls, Sarah A

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The effect of assay formats on the estimation of melanocortin agonist affinity and efficacy using the operation model of agonism von Simon, Sylvie, Young, Tim J., Nickolls, Sarah A.

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Dimerization of the melanocortin 4 receptor: A study using bioluminescence resonance energy transfer von Nickolls, Sarah A., Maki, Rich A.

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Molecular Interactions of Nonpeptide Agonists and Antagonists with the Melanocortin-4 Receptor von Fleck, Beth A, Chen, Yang, Weidong, Huntley, Rajesh, Markison, Stacy, Nickolls, Sarah A, Foster, Alan C, Hoare, Sam R. J

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Interaction of the D2short dopamine receptor with G proteins: Analysis of receptor/G protein selectivity von NICKOLLS, Sarah A, STRANGE, Philip G

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Co-Expression of GRK2 Reveals a Novel Conformational State of the [micro]-Opioid Receptor von Nickolls, Sarah A, Humphreys, Sian, Clark, Mellissa, McMurray, Gordon

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Pharmacology in translation: the preclinical and early clinical profile of the novel α2/3 functionally selective GABA A receptor positive allosteric modulator PF-06372865 von Nickolls, Sarah A, Gurrell, Rachel, van Amerongen, Guido, Kammonen, Juha, Cao, Lishuang, Brown, Adam R, Stead, Clara, Mead, Andy, Watson, Christine, Hsu, Cathleen, Owen, Robert M, Pike, Andy, Fish, Rebecca L, Chen, Laigao, Qiu, Ruolun, Morris, Evan D, Feng, Gang, Whitlock, Mark, Gorman, Donal, van Gerven, Joop, Reynolds, David S, Dua, Pinky, Butt, Richard P

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Agonist Regulation of D2 Dopamine Receptor/G Protein Interaction von Cordeaux, Yolande, Nickolls, Sarah A., Flood, Lori A., Graber, Stephen G., Strange, Philip G.

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Dimerization of the melanocortin 4 receptor : A study using bioluminescence resonance energy transfer: The melanocortin pathway 2005. Part II von NICKOLLS, Sarah A, MAKI, Rich A

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The influence of G protein subtype on agonist action at D 2 dopamine receptors von Nickolls, Sarah A., Strange, Philip G.

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