Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors von Chino, Ayaka, Seo, Ryushi, Amano, Yasushi, Namatame, Ichiji, Hamaguchi, Wataru, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki, Masuda, Naoyuki

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Synthesis and in Vivo Evaluation of Novel Quinoline Derivatives as Phosphodiesterase 10A Inhibitors von Hamaguchi, Wataru, Masuda, Naoyuki, Samizu, Kiyohiro, Mihara, Takuma, Takama, Kaori, Watanabe, Toshihiro

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Stepwise Construction of Head-to-Tail-Type Oligothiophenes via Iterative Palladium-Catalyzed CH Arylation and Halogen Exchange von Masuda, Naoyuki, Tanba, Shunsuke, Sugie, Atsushi, Monguchi, Daiki, Koumura, Nagatoshi, Hara, Kohjiro, Mori, Atsunori

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Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436 von Hamaguchi, Wataru, Masuda, Naoyuki, Miyamoto, Satoshi, Kikuchi, Shigetoshi, Narazaki, Fumie, Shiina, Yasuhiro, Seo, Ryushi, Amano, Yasushi, Mihara, Takuma, Moriguchi, Hiroyuki, Hattori, Kouji

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Potent and orally bioavailable CCR4 antagonists: Synthesis and structure–activity relationship study of 2-aminoquinazolines von Yokoyama, Kazuhiro, Ishikawa, Noriko, Igarashi, Susumu, Kawano, Noriyuki, Masuda, Naoyuki, Hamaguchi, Wataru, Yamasaki, Shingo, Koganemaru, Yohei, Hattori, Kazuyuki, Miyazaki, Takahiro, Ogino, Shin-ichi, Matsumoto, Yuzo, Takeuchi, Makoto, Ohta, Mitsuaki

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Synthesis and Crystal Structure of N-Salicylidene-2-hydroxy-5-bromobenzylamine von MASUDA, Naoyuki, KAKUTA, Yoshihisa, YOSHIOKA, Daisuke, MIKURIYA, Masahiro

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Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability von Chino, Ayaka, Masuda, Naoyuki, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki

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Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors von Chino, Ayaka, Honda, Shugo, Morita, Masataka, Yonezawa, Koichi, Hamaguchi, Wataru, Amano, Yasushi, Moriguchi, Hiroyuki, Yamazaki, Mayako, Aota, Masaki, Tomishima, Masaki, Masuda, Naoyuki

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Design and synthesis of novel benzimidazole derivatives as phosphodiesterase 10A inhibitors with reduced CYP1A2 inhibition von Hamaguchi, Wataru, Masuda, Naoyuki, Isomura, Mai, Miyamoto, Satoshi, Kikuchi, Shigetoshi, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Watanabe, Toshihiro

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Synthesis, SAR study, and biological evaluation of novel quinoline derivatives as phosphodiesterase 10A inhibitors with reduced CYP3A4 inhibition von Hamaguchi, Wataru, Masuda, Naoyuki, Miyamoto, Satoshi, Shiina, Yasuhiro, Kikuchi, Shigetoshi, Mihara, Takuma, Moriguchi, Hiroyuki, Fushiki, Hiroshi, Murakami, Yoshihiro, Amano, Yasushi, Honbou, Kazuya, Hattori, Kouji

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Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors von Ayaka Chino, Ryushi Seo, Yasushi Amano, Ichiji Namatame, Wataru Hamaguchi, Kazuya Honbou, Takuma Mihara, Mayako Yamazaki, Masaki Tomishima, Naoyuki Masuda

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KDR-5169, a new gastrointestinal prokinetic agent, enhances gastric contractile and emptying activities in dogs and rats von Tazawa, Shigeki, Masuda, Naoyuki, Koizumi, Takashi, Kitazawa, Makio, Nakane, Tokio, Miyata, Hiroshi

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Bumper attachment device von Masuda, Naoyuki

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Binding Modes of Two Novel Non-Nucleoside Reverse Transcriptase Inhibitors, YM-215389 and YM-228855, to HIV Type-1 Reverse Transcriptase von Kodama, Eiichi, Orita, Masaya, Masuda, Naoyuki, Yamamoto, Osamu, Fujii, Masahiro, Ohgami, Tetsuro, Kageyama, Shunji, Ohta, Mitsuaki, Hatta, Toshifumi, Inoue, Hiroshi, Suzuki, Hiroshi, Sudo, Kenji, Shimizu, Yasuaki, Matsuoka, Masao

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The First Total Synthesis of (±)-Terpestacin, HIV Syncytium Formation Inhibitor von Tatsuta, Kuniaki, Masuda, Naoyuki, Nishida, Hidemitsu

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The First Total Synthesis of Natural (+)-Terpestacin, Syncytium Formation Inhibitor von TATSUTA, KUNIAKI, MASUDA, NAOYUKI

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Mononuclear cobalt (III) complexes with N-salicylidene-2-hydroxy-5-bromobenzylamine and N-salicylidene-2-hydroxy-5-chlorobenzylamine von Mikuriya, Masahiro, Masuda, Naoyuki, Kakuta, Yoshihisa, Minato, Shinya, Inui, Takaya, Yoshioka, Daisuke

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Dinuclear Copper(II) 3,4,5-Tri-O-benzylgallate von Mikuriya, Masahiro, Yamakawa, Chihiro, Masuda, Naoyuki, Yoshioka, Daisuke, Yamaguchi, Sayuri, Yamada, Hidetoshi, Mizuta, Tsutomu, Kawata, Naomi, Tanaka, Hidekazu, Handa, Makoto

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BUMPER ATTACHMENT DEVICE von MASUDA, Naoyuki

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Synthesis, crystal structures, spectral, electrochemical and magnetic properties of di-µ-phenoxido-bridged dinuclear copper(II) complexes with N-salicylidene-2-hydroxybenzylamine d... von Kakuta, Yoshihisa, Masuda, Naoyuki, Kurushima, Michihiro, Hashimoto, Takashi, Yoshioka, Daisuke, Sakiyama, Hiroshi, Hiraoka, Yuya, Handa, Makoto, Mikuriya, Masahiro

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