Discovery of AAT-008, a novel, potent, and selective prostaglandin EP4 receptor antagonist von Okumura, Yoshiyuki, Yamagishi, Tatsuya, Nukui, Seiji, Nakao, Kazunari

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Discovery and stereoselective synthesis of the novel isochroman neurokinin-1 receptor antagonist ‘CJ-17,493’ von Shishido, Yuji, Wakabayashi, Hiroaki, Koike, Hiroki, Ueno, Naomi, Nukui, Seiji, Yamagishi, Tatsuya, Murata, Yoshinori, Naganeo, Fumiharu, Mizutani, Mayumi, Shimada, Kaoru, Fujiwara, Yoshiko, Sakakibara, Ayano, Suga, Osamu, Kusano, Rinko, Ueda, Satoko, Kanai, Yoshihito, Tsuchiya, Megumi, Satake, Kunio

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3-Amino-5-bromo-2-iodopyridine von Bunker, Kevin D., Sach, Neal W., Nukui, Seiji, Rheingold, Arnold L., Yanovsky, Alex

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Palladium-Mediated Asymmetric Synthesis of Cis-3,6-Disubstituted Cyclohexenes. A Short Total Synthesis of Optically Active (+)-.gamma.-Lycorane von Yoshizaki, Hiroki, Satoh, Hisao, Sato, Yoshihiro, Nukui, Seiji, Shibasaki, Masakatsu, Mori, Miwako

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Catalytic asymmetric synthesis of a functionalized indolizidine derivative. A useful intermediate suitable for the synthesis of various glycosidase inhibitors von Nukui, Seiji, Sodeoka, Mikiko, Shibasaki, Masakatsu

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Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation von Vernier, William, Chong, Wesley, Rewolinski, David, Greasley, Samantha, Pauly, Thomas, Shaw, Morena, Dinh, Dac, Ferre, Rose Ann, Nukui, Seiji, Ornelas, Martha, Reyner, Eric

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Regio- and Stereoselective Functionalization of an Optically Active Tetrahydroindolizine Derivative. Catalytic Asymmetric Syntheses of Lentiginosine, 1,2-Diepilentiginosine, and Ge... von Nukui, Seiji, Sodeoka, Mikiko, Sasai, Hiroaki, Shibasaki, Masakatsu

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Discovery of a novel class of targeted kinase inhibitors that blocks protein kinase C signaling and ameliorates retinal vascular leakage in a diabetic rat model von Grant, Stephan, Tran, Phong, Zhang, Qin, Zou, Aihua, Dinh, Dac, Jensen, Jordan, Zhou, Sue, Kang, Xiaolin, Zachwieja, Joseph, Lippincott, John, Liu, Kevin, Johnson, Sarah Ludlum, Scales, Stephanie, Yin, Chunfeng, Nukui, Seiji, Stoner, Chad, Prasanna, Ganesh, Lafontaine, Jennifer, Wells, Peter, Li, Hui

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Discovery of novel and orally active NR2B-selective N-methyl- d-aspartate (NMDA) antagonists, pyridinol derivatives with reduced HERG binding affinity von Kawai, Makoto, Nakamura, Hiroshi, Sakurada, Isao, Shimokawa, Hirohisa, Tanaka, Hirotaka, Matsumizu, Miyako, Ando, Kazuo, Hattori, Kazunari, Ohta, Atsuko, Nukui, Seiji, Omura, Atsushi, Kawamura, Mitsuhiro

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Corrigendum to “Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation” [Bioorg. Med. Chem. 18... von Vernier, William F., Chong, Wesley K.M., Rewolinski, David A., Greasley, Samantha E., Pauly, Thomas A., Shaw, Morena N., Dinh, Dac M., Ferre, Rose Ann A., Meador, James W., Nukui, Seiji, Ornelas, Martha A., Paz, Robert L., Reyner, Eric L.

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4-Chloro-7-hydroxy-6-methyl-1,7-naphthyridin-8(7 H )-one von Bunker, Kevin D., Nukui, Seiji, Rheingold, Arnold L., DiPasquale, Antonio, Yanovsky, Alex

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Synthesis of the Vancomycin CD and DE Ring Systems von Boger, Dale L, Borzilleri, Robert M, Nukui, Seiji, Beresis, Richard T

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6-(2,6-Dimethyl-phen-yl)pyrido[2,3-d]pyrimidin-7-amine von Nukui, Seiji, Rheingold, Arnold L, Dipasquale, Antonio, Yanovsky, Alex

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ORAL GLP RECEPTOR AGONISTS von MUTO, Susumu, NUKUI, Seiji, SCULLY, Conor, BROWN, Giles Albert, PAUL, Rebecca, WADA, Hiroki, CONGREVE, Miles Stuart

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Substituted N-pyrimidin-4-yl-3-aminopyrrolo[3,4-C]pyrazoles as protein kinase C inhibitors von Scales, Stephanie Anne, Li, Hui, Yin, Chunfeng, Teng, Min, Nukui, Seiji

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Synthesis of (9R,12S)- and (9S,12S)-Cycloisodityrosine and Their N-Methyl Derivatives von Boger, Dale L, Zhou, Jiacheng, Borzilleri, Robert M, Nukui, Seiji, Castle, Steven L

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Synthesis of appropriately functionalized vancomycin CD and DE ring systems von Boger, Dale L., Borzilleri, Robert M., Nukui, Seiji

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Synthesis of (R)-(4-Methoxy-3,5-dihydroxyphenyl)glycine Derivatives:  The Central Amino Acid of Vancomycin and Related Agents von Boger, Dale L, Borzilleri, Robert M, Nukui, Seiji

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ORAL GLP RECEPTOR AGONISTS von MUTO, Susumu, NUKUI, Seiji, SCULLY, Conor, BROWN, Giles Albert, PAUL, Rebecca, WADA, Hiroki, CONGREVE, Miles Stuart

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Substituted n-pyrimidin-4-yl-3-amino-pyrrolo[3,4-c]pyrazoles as protein kinase C inhibitors von Scales, Stephanie Anne, Li, Hui, Yin, Chunfeng, Teng, Min, Nukui, Seiji

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