Orally available selective melanocortin-4 receptor antagonists stimulate food intake and reduce cancer-induced cachexia in mice von Weyermann, Philipp, Dallmann, Robert, Magyar, Josef, Anklin, Corinne, Hufschmid, Martina, Dubach-Powell, Judith, Courdier-Fruh, Isabelle, Henneböhle, Marco, Nordhoff, Sonja, Mondadori, Cesare

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Fragment-Based Discovery of Novel Potent Sepiapterin Reductase Inhibitors von Alen, Jo, Schade, Markus, Wagener, Markus, Christian, Frank, Nordhoff, Sonja, Merla, Beatrix, Dunkern, Torsten R, Bahrenberg, Gregor, Ratcliffe, Paul

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A Novel Biosynthetic Pathway Providing Precursors for Fatty Acid Biosynthesis and Secondary Metabolite Formation in Myxobacteria von Mahmud, Taifo, Bode, Helge Bjo¨rn, Silakowski, Barbara, Kroppenstedt, Reiner M., Xu, Mingjie, Nordhoff, Sonja, Ho¨fle, Gerhard, Mu¨ller, Rolf

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Inhibiting the immunoproteasome's β5i catalytic activity affects human peripheral blood‐derived immune cell viability von Pletinckx, Katrien, Vaßen, Silke, Schlusche, Ilka, Nordhoff, Sonja, Bahrenberg, Gregor, Dunkern, Torsten R.

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In silico fragment-based discovery of DPP-IV S1 pocket binders von Rummey, Christian, Nordhoff, Sonja, Thiemann, Meinolf, Metz, Günther

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The design of potent and selective inhibitors of DPP-4: Optimization of ADME properties by amide replacements von Nordhoff, Sonja, Bulat, Stephan, Cerezo-Gálvez, Silvia, Hill, Oliver, Hoffmann-Enger, Barbara, López-Canet, Meritxell, Rosenbaum, Claudia, Rummey, Christian, Thiemann, Meinolf, Matassa, Victor G., Edwards, Paul J., Feurer, Achim

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Discovery of β-homophenylalanine based pyrrolidin-2-ylmethyl amides and sulfonamides as highly potent and selective inhibitors of dipeptidyl peptidase IV von Nordhoff, Sonja, Cerezo-Gálvez, Silvia, Deppe, Holger, Hill, Oliver, López-Canet, Meritxell, Rummey, Christian, Thiemann, Meinolf, Matassa, Victor G., Edwards, Paul J., Feurer, Achim

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From lead to preclinical candidate: Optimization of β-homophenylalanine based inhibitors of dipeptidyl peptidase IV von Nordhoff, Sonja, López-Canet, Meritxell, Hoffmann-Enger, Barbara, Bulat, Stephan, Cerezo-Gálvez, Silvia, Hill, Oliver, Rosenbaum, Claudia, Rummey, Christian, Thiemann, Meinolf, Matassa, Victor G., Edwards, Paul J., Feurer, Achim

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The reversed binding of β-phenethylamine inhibitors of DPP-IV: X-ray structures and properties of novel fragment and elaborated inhibitors von Nordhoff, Sonja, Cerezo-Gálvez, Silvia, Feurer, Achim, Hill, Oliver, Matassa, Victor G., Metz, Günther, Rummey, Christian, Thiemann, Meinolf, Edwards, Paul J.

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6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL von RIDER, David, DUNKERN, Torsten, WAGENER, Markus, NORDHOFF, Sonja, BAHRENBERG, Gregor, JAKOB, Florian

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6-membered cyclic amines or lactames substituted with urea and phenyl von Nordhoff, Sonja, Wagener, Markus, Rider, David, Jakob, Florian, Bahrenberg, Gregor, Dunkern, Torsten

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6-membered cyclic amines or lactames substituted with urea and phenyl von Nordhoff, Sonja, Wagener, Markus, Rider, David, Jakob, Florian, Bahrenberg, Gregor, Dunkern, Torsten

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PYRAZOLYL-BASED CARBOXAMIDES II AS CRAC CHANNEL INHIBITORS von KLESS, Achim, WACHTEN, Sebastian, RITTER, Stefanie, VOSS, Felix, NORDHOFF, Sonja

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6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL von RIDER, DAVID, JAKOB, FLORIAN, WAGENER, MARKUS, BAHRENBERG, GREGOR, NORDHOFF, SONJA, DUNKERN, TORSTEN

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6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL von RIDER, David, DUNKERN, Torsten, WAGENER, Markus, NORDHOFF, Sonja, BAHRENBERG, Gregor, JAKOB, Florian

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6-MEMBERED CYCLIC AMINES OR LACTAMES SUBSTITUTED WITH UREA AND PHENYL von RIDER DAVID, JAKOB FLORIAN, WAGENER MARKUS, NORDHOFF SONJA, BAHRENBERG GREGOR, DUNKERN TORSTEN

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PYRAZOLYL-BASED CARBOXAMIDES V von KLESS, ACHIM, VOSS, FELIX, NORDHOFF, SONJA, WACHTEN, SEBASTIAN, RITTER, STEFANIE

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PYRAZOLYL-BASED CARBOXAMIDES AS CRAC INHIBITORS von VOSS, FELIX, OBERBÖRSCH, STEFAN, RITTER, STEFANIE, NORDHOFF, SONJA, WACHTEN, SEBASTIAN

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Pyrazolyl-based carboxamides I von KLESS ACHIM, VOSS FELIX, RITTER STEFANIE, WACHTEN SEBASTIAN, NORDHOFF SONJA

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PYRAZOLYL-BASED CARBOXAMIDES II AS CRAC CHANNEL INHIBITORS von KLESS, ACHIM, VOSS, FELIX, NORDHOFF, SONJA, WACHTEN, SEBASTIAN, RITTER, STEFANIE

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