Sperm Toolbox-A selection of small molecules to study human spermatozoa von Gruber, Franz S, Richardson, Anthony, Johnston, Zoe C, Myles, Rachel, Norcross, Neil R, Day, David P, Georgiou, Irene, Sesma-Sanz, Laura, Wilson, Caroline, Read, Kevin D, Martins da Silva, Sarah, Barratt, Christopher L R, Gilbert, Ian H, Swedlow, Jason R

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Exploring the Trypanosoma brucei Hsp83 potential as a target for structure guided drug design von Pizarro, Juan Carlos, Hills, Tanya, Senisterra, Guillermo, Wernimont, Amy K, Mackenzie, Claire, Norcross, Neil R, Ferguson, Michael A J, Wyatt, Paul G, Gilbert, Ian H, Hui, Raymond

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Compounds enhancing human sperm motility identified using a high-throughput phenotypic screening platform von Gruber, Franz S, Johnston, Zoe C, Norcross, Neil R, Georgiou, Irene, Wilson, Caroline, Read, Kevin D, Gilbert, Ian H, Swedlow, Jason R, Martins da Silva, Sarah, Barratt, Christopher L R

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Male contraceptive development: A medicinal chemistry perspective von Norcross, Neil R., Georgiou, Irene, Johnston, Zoe C., Gruber, Franz S., Swedlow, Jason R., Read, Kevin D., Barratt, Christopher LR, Gilbert, Ian H.

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Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity von Green, Simon R, Wilson, Caroline, Eadsforth, Thomas C, Punekar, Avinash S, Tamaki, Fabio K, Wood, Gavin, Caldwell, Nicola, Forte, Barbara, Norcross, Neil R, Kiczun, Michael, Post, John M, Lopez-Román, Eva Maria, Engelhart, Curtis A, Lukac, Iva, Zuccotto, Fabio, Epemolu, Ola, Boshoff, Helena I M, Schnappinger, Dirk, Walpole, Chris, Gilbert, Ian H, Read, Kevin D, Wyatt, Paul G, Baragaña, Beatriz

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Validation of N-myristoyltransferase as Potential Chemotherapeutic Target in Mammal-Dwelling Stages of Trypanosoma cruzi von Herrera, Linda J, Brand, Stephen, Santos, Andres, Nohara, Lilian L, Harrison, Justin, Norcross, Neil R, Thompson, Stephen, Smith, Victoria, Lema, Carolina, Varela-Ramirez, Armando, Gilbert, Ian H, Almeida, Igor C, Maldonado, Rosa A

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Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy von Baragaña, Beatriz, Norcross, Neil R, Wilson, Caroline, Porzelle, Achim, Hallyburton, Irene, Grimaldi, Raffaella, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Stojanovski, Laste, Simeons, Frederick R. C, Wyatt, Paul G, Delves, Michael J, Meister, Stephan, Duffy, Sandra, Avery, Vicky M, Winzeler, Elizabeth A, Sinden, Robert E, Wittlin, Sergio, Frearson, Julie A, Gray, David W, Fairlamb, Alan H, Waterson, David, Campbell, Simon F, Willis, Paul, Read, Kevin D, Gilbert, Ian H

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High-throughput phenotypic screening of the human spermatozoon von Johnston, Zoe C, Gruber, Franz S, Brown, Sean G, Norcross, Neil R, Swedlow, Jason, Gilbert, Ian H, Barratt, Christopher L R

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Substituted 2‑Phenylimidazopyridines: A New Class of Drug Leads for Human African Trypanosomiasis von Tatipaka, Hari Babu, Gillespie, J. Robert, Chatterjee, Arnab K, Norcross, Neil R, Hulverson, Matthew A, Ranade, Ranae M, Nagendar, Pendem, Creason, Sharon A, McQueen, Joshua, Duster, Nicole A, Nagle, Advait, Supek, Frantisek, Molteni, Valentina, Wenzler, Tanja, Brun, Reto, Glynne, Richard, Buckner, Frederick S, Gelb, Michael H

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Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma brucei N‑Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Tr... von Brand, Stephen, Norcross, Neil R, Thompson, Stephen, Harrison, Justin R, Smith, Victoria C, Robinson, David A, Torrie, Leah S, McElroy, Stuart P, Hallyburton, Irene, Norval, Suzanne, Scullion, Paul, Stojanovski, Laste, Simeons, Frederick R. C, van Aalten, Daan, Frearson, Julie A, Brenk, Ruth, Fairlamb, Alan H, Ferguson, Michael A. J, Wyatt, Paul G, Gilbert, Ian H, Read, Kevin D

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Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors von Brand, Stephen, Cleghorn, Laura A. T, McElroy, Stuart P, Robinson, David A, Smith, Victoria C, Hallyburton, Irene, Harrison, Justin R, Norcross, Neil R, Spinks, Daniel, Bayliss, Tracy, Norval, Suzanne, Stojanovski, Laste, Torrie, Leah S, Frearson, Julie A, Brenk, Ruth, Fairlamb, Alan H, Ferguson, Michael A. J, Read, Kevin D, Wyatt, Paul G, Gilbert, Ian H

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Trisubstituted Pyrimidines as Efficacious and Fast-Acting Antimalarials von Norcross, Neil R, Baragaña, Beatriz, Wilson, Caroline, Hallyburton, Irene, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Stojanovski, Laste, Simeons, Frederick R. C, Porzelle, Achim, Grimaldi, Raffaella, Wittlin, Sergio, Duffy, Sandra, Avery, Vicky M, Meister, Stephan, Sanz, Laura, Jiménez-Díaz, Belén, Angulo-Barturen, Iñigo, Ferrer, Santiago, Martínez, María Santos, Gamo, Francisco Javier, Frearson, Julie A, Gray, David W, Fairlamb, Alan H, Winzeler, Elizabeth A, Waterson, David, Campbell, Simon F, Willis, Paul, Read, Kevin D, Gilbert, Ian H

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Substituted Aminoacetamides as Novel Leads for Malaria Treatment von Norcross, Neil R., Wilson, Caroline, Baragaña, Beatriz, Hallyburton, Irene, Osuna‐Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Fletcher, Daniel, Sinden, Robert, Delves, Michael, Ruecker, Andrea, Duffy, Sandra, Meister, Stephan, Antonova‐Koch, Yevgeniya, Crespo, Benigno, de Cózar, Cristina, Sanz, Laura M., Gamo, Francisco Javier, Avery, Vicky M., Frearson, Julie A., Gray, David W., Fairlamb, Alan H., Winzeler, Elizabeth A., Waterson, David, Campbell, Simon F., Willis, Paul A., Read, Kevin D., Gilbert, Ian H.

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Dialkylimidazole inhibitors of Trypanosoma cruzi sterol 14α-demethylase as anti-Chagas disease agents von Suryadevara, Praveen Kumar, Racherla, Kishore Kumar, Olepu, Srinivas, Norcross, Neil R., Tatipaka, Hari Babu, Arif, Jennifer A., Planer, Joseph D., Lepesheva, Galina I., Verlinde, Christophe L.M.J., Buckner, Frederick S., Gelb, Michael H.

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Total Synthesis of (±)-α-Isosparteine, (±)-β-Isosparteine, and (±)-Sparteine from a Common Tetraoxobispidine Intermediate von Norcross, Neil R, Melbardis, John P, Solera, Margarita Ferris, Sephton, Mark A, Kilner, Colin, Zakharov, Lev N, Astles, Peter C, Warriner, Stuart L, Blakemore, Paul R

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Lead Optimization of a Pyrazole Sulfonamide Series of Trypanosoma bruceiN-Myristoyltransferase Inhibitors: Identification and Evaluation of CNS Penetrant Compounds as Potential Tre... von Brand, Stephen, Norcross, Neil R, Thompson, Stephen, Harrison, Justin R, Smith, Victoria C, Robinson, David A, Torrie, Leah S, McElroy, Stuart P, Hallyburton, Irene, Norval, Suzanne, Scullion, Paul, Stojanovski, Laste, Simeons, Frederick RC, van Aalten, Daan, Frearson, Julie A, Brenk, Ruth, Fairlamb, Alan H, Ferguson, Michael AJ, Wyatt, Paul G, Gilbert, Ian H, Read, Kevin D

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A Practical Synthesis of (±)-α-Isosparteine from a Tetraoxobispidine Core von Blakemore, Paul R, Kilner, Colin, Norcross, Neil R, Astles, Peter C

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Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis von Baragaña, Beatriz, Forte, Barbara, Choi, Ryan, Nakazawa Hewitt, Stephen, Bueren-Calabuig, Juan A, Pisco, João Pedro, Peet, Caroline, Dranow, David M, Robinson, David A, Jansen, Chimed, Norcross, Neil R, Vinayak, Sumiti, Anderson, Mark, Brooks, Carrie F, Cooper, Caitlin A, Damerow, Sebastian, Delves, Michael, Dowers, Karen, Duffy, James, Edwards, Thomas E, Hallyburton, Irene, Horst, Benjamin G, Hulverson, Matthew A, Ferguson, Liam, Jiménez-Díaz, María Belén, Jumani, Rajiv S, Lorimer, Donald D, Love, Melissa S, Maher, Steven, Matthews, Holly, McNamara, Case W, Miller, Peter, O'Neill, Sandra, Ojo, Kayode K, Osuna-Cabello, Maria, Pinto, Erika, Post, John, Riley, Jennifer, Rottmann, Matthias, Sanz, Laura M, Scullion, Paul, Sharma, Arvind, Shepherd, Sharon M, Shishikura, Yoko, Simeons, Frederick RC, Stebbins, Erin E, Stojanovski, Laste, Straschil, Ursula, Tamaki, Fabio K, Tamjar, Jevgenia, Torrie, Leah S, Vantaux, Amélie, Witkowski, Benoît, Wittlin, Sergio, Yogavel, Manickam, Zuccotto, Fabio, Angulo-Barturen, Iñigo, Sinden, Robert, Baum, Jake, Gamo, Francisco-Javier, Mäser, Pascal, Kyle, Dennis E, Winzeler, Elizabeth A, Myler, Peter J, Wyatt, Paul G, Floyd, David, Matthews, David, Sharma, Amit, Striepen, Boris, Huston, Christopher D, Gray, David W, Fairlamb, Alan H, Pisliakov, Andrei V, Walpole, Chris, Read, Kevin D, Van Voorhis, Wesley C, Gilbert, Ian H

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Substituted Aminoacetamides as Novel Leads for Malaria Treatment von Norcross, Neil R, Wilson, Caroline, Baragaña, Beatriz, Hallyburton, Irene, Osuna-Cabello, Maria, Norval, Suzanne, Riley, Jennifer, Fletcher, Daniel, Sinden, Robert, Delves, Michael, Ruecker, Andrea, Duffy, Sandra, Meister, Stephan, Antonova-Koch, Yevgeniya, Crespo, Benigno, de Cózar, Cristina, Sanz, Laura M, Gamo, Francisco Javier, Avery, Vicky M, Frearson, Julie A, Gray, David W, Fairlamb, Alan H, Winzeler, Elizabeth A, Waterson, David, Campbell, Simon F, Willis, Paul A, Read, Kevin D, Gilbert, Ian H

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Identification of Inhibitors of the Leishmania cdc2-Related Protein Kinase CRK3 von Cleghorn, Laura A. T., Woodland, Andrew, Collie, Iain T., Torrie, Leah S., Norcross, Neil, Luksch, Torsten, Mpamhanga, Chido, Walker, Roderick G., Mottram, Jeremy C., Brenk, Ruth, Frearson, Julie A., Gilbert, Ian H., Wyatt, Paul G.

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