Parallel Synthesis of Piperazine Tethered Thiazole Compounds with Antiplasmodial Activity von Rayala, Ramanjaneyulu, Chaudhari, Prakash, Bunnell, Ashley, Roberts, Bracken, Chakrabarti, Debopam, Nefzi, Adel

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1,5-Disubstituted Acylated 2-Amino-4,5-dihydroimidazoles as a New Class of Retinoic Acid Receptor-Related Orphan Receptor (ROR) Inhibitors von Ortiz, Maria A, Piedrafita, F Javier, Nefzi, Adel

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Solid phase synthesis of isoxazole and isoxazoline-carboxamides via [2+3]-dipolar cycloaddition using resin-bound alkynes or alkenes von Dadiboyena, Sureshbabu, Nefzi, Adel

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Small Molecule Compounds Identified from Mixture-Based Library Inhibit Binding between Plasmodium falciparum Infected Erythrocytes and Endothelial Receptor ICAM-1 von Chesnokov, Olga, Visitdesotrakul, Pimnitah, Kalani, Komal, Nefzi, Adel, Oleinikov, Andrew V

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Bis-Cyclic Guanidine Heterocyclic Peptidomimetics as Opioid Ligands with Mixed μ-, κ- and δ-Opioid Receptor Interactions: A Potential Approach to Novel Analgesics von McLaughlin, Jay P, Rayala, Ramanjaneyulu, Bunnell, Ashley J, Tantak, Mukund P, Eans, Shainnel O, Nefzi, Khadija, Ganno, Michelle L, Dooley, Colette T, Nefzi, Adel

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Evaluating the effect of dermaseptin S4 and its derivatives on multidrug-resistant bacterial strains and on the colon cancer cell line SW620 von Belaid, Afifa, Braiek, Afef, Alibi, Sana, Hassen, Wafa, Beltifa, Asma, Nefzi, Adel, Mansour, Hedi Ben

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Inhibition of methicillin-resistant Staphylococcus aureus (MRSA) by antimicrobial peptides (AMPs) and plant essential oils von Zouhir, Abdelmajid, Jridi, Taoufik, Nefzi, Adel, Ben Hamida, Jeannette, Sebei, Khaled

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Encoding mu-opioid receptor biased agonism with interaction fingerprints von Hernández-Alvarado, R. Bruno, Madariaga-Mazón, Abraham, Cosme-Vela, Fernando, Marmolejo-Valencia, Andrés F., Nefzi, Adel, Martinez-Mayorga, Karina

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Parallel solid-phase synthesis of disubstituted 3-(1H-benzo[d]imidazol-2-yl)imidazolidine-2,4-diones and 3-(1H-benzo[d]imidazol-2-yl)-2-thioxoimidazolidin-4-ones von Dadiboyena, Sureshbabu, Nefzi, Adel

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Identification of Bis-Cyclic Guanidines as Antiplasmodial Compounds from Positional Scanning Mixture-Based Libraries von Perry, Jr, David L, Roberts, Bracken F, Debevec, Ginamarie, Michaels, Heather A, Chakrabarti, Debopam, Nefzi, Adel

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Synthesis of functionalized tetrasubstituted pyrazolyl heterocycles – A review von Dadiboyena, Sureshbabu, Nefzi, Adel

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Small-molecule antagonists of apoptosis suppressor XIAP exhibit broad antitumor activity von Schimmer, Aaron D., Welsh, Kate, Pinilla, Clemencia, Wang, Zhiliang, Krajewska, Maryla, Bonneau, Marie-Josee, Pedersen, Irene M., Kitada, Shinichi, Scott, Fiona L., Bailly-Maitre, Beatrice, Glinsky, Gennadi, Scudiero, Dominick, Sausville, Edward, Salvesen, Guy, Nefzi, Adel, Ostresh, John M., Houghten, Richard A., Reed, John C.

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The Current Status of Heterocyclic Combinatorial Libraries von Nefzi, Adel, Ostresh, John M, Houghten, Richard A

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Combinatorial Chemistry:  Libraries from Libraries, the Art of the Diversity-Oriented Transformation of Resin-Bound Peptides and Chiral Polyamides to Low Molecular Weight Acyclic a... von Nefzi, Adel, Ostresh, John M, Yu, Jongping, Houghten, Richard A

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Combinatorial Synthesis of Oxazol-Thiazole Bis-Heterocyclic Compounds von Murru, Siva, Nefzi, Adel

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Small-molecule XIAP inhibitors derepress downstream effector caspases and induce apoptosis of acute myeloid leukemia cells von Carter, Bing Z., Gronda, Marcela, Wang, Zhiliang, Welsh, Kate, Pinilla, Clemencia, Andreeff, Michael, Schober, Wendy D., Nefzi, Adel, Pond, Gregory R., Mawji, Imtiaz A., Houghten, Richard A., Ostresh, John, Brandwein, Joseph, Minden, Mark D., Schuh, Andre C., Wells, Richard A., Messner, Hans, Chun, Kathy, Reed, John C., Schimmer, Aaron D.

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Recent methodologies toward the synthesis of valdecoxib: A potential 3,4-diarylisoxazolyl COX-II inhibitor von Dadiboyena, Sureshbabu, Nefzi, Adel

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Mixture-Based Synthetic Combinatorial Libraries von Houghten, Richard A, Pinilla, Clemencia, Appel, Jon R, Blondelle, Sylvie E, Dooley, Colette T, Eichler, Jutta, Nefzi, Adel, Ostresh, John M

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Potential therapeutic use of dermaseptin S4 from the frog Phyllomedusa sauvagii and its derivatives against bacterial pathogens in fish von Braik, Afef, Serna-Duque, John Alberto, Nefzi, Adel, Aroui, Sonia, Esteban, María Ángeles

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Polyheterocyclic peptidomimetics: Parallel solid phase synthesis of oligo cyclic guanidines and their inhibition activity against Mycobacterium tuberculosis DNA gyrase von Tantak, Mukund, Rayala, Ramanjaneyulu, Deng, Zifang, Bunnell, Ashley, Wang, Ting, Chaudhari, Prakash, Leng, Fenfei, Nefzi, Adel

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