Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoro- methyl)phenyl]ethyl]-... von Tagat, Jayaram R, Steensma, Ruo W, McCombie, Stuart W, Nazareno, Dennis V, Lin, Sue-Ing, Neustadt, Bernard R, Cox, Kathleen, Xu, Serena, Wojcik, Lisa, Murray, Michael G, Vantuno, Nicole, Baroudy, Bahige M, Strizki, Julie M

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Synthesis of Mono- and Difluoronaphthoic Acids von Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis V, Boyle, Craig D, Kozlowski, Joseph A, Chackalamannil, Samuel, Josien, Hubert, Wang, Yuguang, Zhou, Guowei

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Piperazine-Based CCR5 antagonists as HIV-1 inhibitors. I: 2( S)-methyl piperazine as a key pharmacophore element von Tagat, Jayaram R., McCombie, Stuart W., Steensma, Ruo W., Lin, Sue-Ing, Nazareno, Dennis V., Baroudy, Bahige, Vantuno, Nicole, Xu, Serena, Liu, Jia

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Metabolic stabilization of benzylidene ketal M2 muscarinic receptor antagonists via halonaphthoic acid substitution von BOYLE, Craig D, CHACKALAMANNIL, Samuel, YUGUANG WANG, GUOWEI ZHOU, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, COHEN-WILLIAMS, Mary, COFFIN, Vicki L, COX, Kathleen A, GROTZ, Diane E, DUFFY, Ruth A, CLADER, John W, RUPERTO, Vilma, LACHOWICZ, Jean E, GREENLEE, William J, JOSIEN, Hubert B, KAMINSKI, James J, KOZLOWSKI, Joseph A, MCCOMBIE, Stuart W, NAZARENO, Dennis V, TAGAT, Jayaram R

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Metabolic stabilization of benzylidene ketal M 2 muscarinic receptor antagonists via halonaphthoic acid substitution von Boyle, Craig D., Chackalamannil, Samuel, Clader, John W., Greenlee, William J., Josien, Hubert B., Kaminski, James J., Kozlowski, Joseph A., McCombie, Stuart W., Nazareno, Dennis V., Tagat, Jayaram R., Wang, Yuguang, Zhou, Guowei, Billard, William, Binch, Herbert, Crosby, Gordon, Cohen-Williams, Mary, Coffin, Vicki L., Cox, Kathleen A., Grotz, Diane E., Duffy, Ruth A., Ruperto, Vilma, Lachowicz, Jean E.

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Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3( S )-methyl-4-[1( S )-[4-(trifluoro- methyl)phenyl]eth... von Tagat, Jayaram R., Steensma, Ruo W., McCombie, Stuart W., Nazareno, Dennis V., Lin, Sue-Ing, Neustadt, Bernard R., Cox, Kathleen, Xu, Serena, Wojcik, Lisa, Murray, Michael G., Vantuno, Nicole, Baroudy, Bahige M., Strizki, Julie M.

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Synthetic inhibitors of interleukin-6 I: 2,3,7,8-tetrahydro-4-aryl-1H-cyclopent [e] imidazo [1,2-a]- pyridin-5(6H)-one and related compounds von Tagat, Jayaram R., Nazareno, Dennis V., McCombie, Stuart W., Barton, Beverly E., Shortall, Jennifer, Jackson, James

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Synthesis and anti-herpes activity of some a-ring functionalized dehydroabietane derivatives von Tagat, Jayaram R., Nazareno, Dennis V., Puar, Mohindar S., McCombie, Stuart W., Ganguly, Ashit K.

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ChemInform Abstract: Synthesis of Mono- and Difluoronaphthoic Acids von Tagat, Jayaram R., McCombie, Stuart W., Nazareno, Dennis V., Boyle, Craig D., Kozlowski, Joseph A., Chackalamannil, Samuel, Josien, Hubert, Wang, Yuguang, Zhou, Guowei

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ChemInform Abstract: Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. Part 1. 2(S)-Methyl Piperazine as a Key Pharmacophore Element von Tagat, Jayaram R., McCombie, Stuart W., Steensma, Ruo W., Lin, Sue-Ing, Nazareno, Dennis V., Baroudy, Bahige, Vantuno, Nicole, Xu, Serena, Liu, Jia

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Synthesis and structure–Activity relationships of M 2-Selective muscarinic receptor ligands in the 1-[4-(4-Arylsulfonyl)-phenylmethyl]-4-(4-piperidinyl)-piperazine family von McCombie, Stuart W, Lin, Sue-Ing, Tagat, Jayaram R, Nazareno, Dennis, Vice, Susan, Ford, Jennifer, Asberom, Theodros, Leone, Daria, Kozlowski, Joseph A, Zhou, Guowei, Ruperto, Vilma B, Duffy, Ruth A, Lachowicz, Jean E

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