Drug discovery for Duchenne muscular dystrophy via utrophin promoter activation screening von Moorwood, Catherine, Lozynska, Olga, Suri, Neha, Napper, Andrew D, Diamond, Scott L, Khurana, Tejvir S

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Identification of Specific Inhibitors of Human RAD51 Recombinase Using High-Throughput Screening von Huang, Fei, Motlekar, Nuzhat A, Burgwin, Chelsea M, Napper, Andrew D, Diamond, Scott L, Mazin, Alexander V

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Discovery of Indoles as Potent and Selective Inhibitors of the Deacetylase SIRT1 von Napper, Andrew D, Hixon, Jeffrey, McDonagh, Thomas, Keavey, Kenneth, Pons, Jean-Francois, Barker, Jonathan, Yau, Wei Tsung, Amouzegh, Patricia, Flegg, Adam, Hamelin, Estelle, Thomas, Russell J, Kates, Michael, Jones, Stephen, Navia, Manuel A, Saunders, Jeffrey O, DiStefano, Peter S, Curtis, Rory

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Perspectives on phenotypic screening−Screen Design and Assay Technology Special Interest Group von Pak, Chorom, Simpson, Kaylene J., Weston, Andrea D., Cvijic, Mary Ellen, Evans, Kenda, Napper, Andrew D.

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Discovery of Potent Small-Molecule Inhibitors of Multidrug-Resistant Plasmodium falciparum Using a Novel Miniaturized High-Throughput Luciferase-Based Assay von Lucumi, Edinson, Darling, Claire, Jo, Hyunil, Napper, Andrew D, Chandramohanadas, Rajesh, Fisher, Nicholas, Shone, Alison E, Jing, Huiyan, Ward, Stephen A, Biagini, Giancarlo A, DeGrado, William F, Diamond, Scott L, Greenbaum, Doron C

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Targeted drug discovery for pediatric leukemia von Napper, Andrew D, Watson, Venita G

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Beta-hairpin hydrogels as scaffolds for high-throughput drug discovery in three-dimensional cell culture von Worthington, Peter, Drake, Katherine M., Li, Zhiqin, Napper, Andrew D., Pochan, Darrin J., Langhans, Sigrid A.

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Kinetic Characterization and Molecular Docking of a Novel, Potent, and Selective Slow-Binding Inhibitor of Human Cathepsin L von Shah, Parag P, Myers, Michael C, Beavers, Mary Pat, Purvis, Jeremy E, Jing, Huiyan, Grieser, Heather J, Sharlow, Elizabeth R, Napper, Andrew D, Huryn, Donna M, Cooperman, Barry S, Smith, 3rd, Amos B, Diamond, Scott L

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Discriminating High-Value Hits from PAINS von Napper, Andrew D

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Perspectives in ASSAY and Drug Development Technologies von Napper, Andrew D

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A new chapter for ASSAY and drug development technologies von Napper, Andrew D

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Novel high-throughput screen against Candida albicans identifies antifungal potentiators and agents effective against biofilms von LAFLEUR, Michael D, LUCUMI, Edinson, NAPPER, Andrew D, DIAMOND, Scott L, LEWIS, Kim

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Interview with Jonathan Baell, PhD von Napper, Andrew D

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Implementation of a High-Throughput Pilot Screen in Peptide Hydrogel-Based Three-Dimensional Cell Cultures von Worthington, Peter, Drake, Katherine M., Li, Zhiqin, Napper, Andrew D., Pochan, Darrin J., Langhans, Sigrid A.

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Interview with Haian Fu, PhD von Fu, Haian, Napper, Andrew D

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Identification and characterization of 3-substituted pyrazolyl esters as alternate substrates for cathepsin B: The confounding effects of DTT and cysteine in biological assays von Myers, Michael C., Napper, Andrew D., Motlekar, Nuzhat, Shah, Parag P., Chiu, Chun-Hao, Beavers, Mary Pat, Diamond, Scott L., Huryn, Donna M., Smith, Amos B.

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A sensitive luminescent assay for the histone methyltransferase NSD1 and other SAM-dependent enzymes von Drake, Katherine M, Watson, Venita G, Kisielewski, Anne, Glynn, Rebecca, Napper, Andrew D

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Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy- d- xylo-4-hexopyranosid-4-ulose 3,5-epimerase (RmlC) von Sivendran, Sharmila, Jones, Victoria, Sun, Dianqing, Wang, Yi, Grzegorzewicz, Anna E., Scherman, Michael S., Napper, Andrew D., McCammon, J. Andrew, Lee, Richard E., Diamond, Scott L., McNeil, Michael

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A Special Focus on Drug Repurposing, Rescue, and Repositioning von Napper, Andrew D, Mucke, Hermann A M

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Discovery of chemical modulators of a conserved translational control pathway by parallel screening in yeast von Motlekar, Nuzhat, de Almeida, Rogerio Alves, Pavitt, Graham D, Diamond, Scott L, Napper, Andrew D

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