Synthesis and in vitro characterization of cinnoline and benzimidazole analogues as phosphodiesterase 10A inhibitors von Yang, Hao, Murigi, Francis N., Wang, Zhijian, Li, Junfeng, Jin, Hongjun, Tu, Zhude

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Galeterone and VNPT55 disrupt Mnk‐eIF4E to inhibit prostate cancer cell migration and invasion von Kwegyir‐Afful, Andrew K., Bruno, Robert D., Purushottamachar, Puranik, Murigi, Francis N., Njar, Vincent C.O.

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Improved Procedures for Gram-Scale Synthesis of Galeterone 3β-Imidazole and Galeterone 3β-Pyridine Methoxylate, Potent Androgen Receptor/Mnk Degrading Agents von Purushottamachar, Puranik, Murigi, Francis N, Njar, Vincent C. O

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The Novel Mnk1/2 Degrader and Apoptosis Inducer VNLG-152 Potently Inhibits TNBC Tumor Growth and Metastasis von Ramalingam, Senthilmurugan, Ramamurthy, Vidya P, Gediya, Lalji K, Murigi, Francis N, Purushottamachar, Puranik, Huang, Weiliang, Choi, Eun Yong, Zhang, Yuji, Vasaitis, Tadas S, Kane, Maureen A, Lapidus, Rena G, Njar, Vincent C O

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Galeterone and its analogs inhibit Mnk-eIF4E axis, synergize with gemcitabine, impede pancreatic cancer cell migration, invasion and proliferation and inhibit tumor growth in mice von Kwegyir-Afful, Andrew K, Murigi, Francis N, Purushottamachar, Puranik, Ramamurthy, Vidya P, Martin, Marlena S, Njar, Vincent C O

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Dose Optimization Study of AEOL 10150 as a Mitigator of Radiation-Induced Lung Injury in CBA/J Mice von Murigi, Francis N., Mohindra, Pranshu, Hung, Chiwei, Salimi, Shabnam, Goetz, Wilfried, Pavlovic, Radmila, Jackson, Isabel L., Vujaskovic, Zeljko

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Galeterone and The Next Generation Galeterone Analogs, VNPP414 and VNPP433-3β Exert Potent Therapeutic Effects in Castration-/Drug-Resistant Prostate Cancer Preclinical Models In V... von Kwegyir-Afful, Andrew K, Ramalingam, Senthilmurugan, Ramamurthy, Vidya P, Purushottamachar, Puranik, Murigi, Francis N, Vasaitis, Tadas S, Huang, Weiliang, Kane, Maureen A, Zhang, Yuji, Ambulos, Nicholas, Tiwari, Sudhir, Srivastava, Pratima, Nnane, Ivo P, Hussain, Arif, Qiu, Yun, Weber, David J, Njar, Vincent C O

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Synthesis of the Conformationally Constrained Tyrosine Analogues, (R)- and (S)-5-Hydroxy-2-aminoindan-2-carboxylic Acids von Murigi, Francis N, Nichol, Gary S, Mash, Eugene A

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Organic Crystal Engineering with 1,4-Piperazine-2,5-diones. 8. Synthesis, Crystal Packing, and Thermochemistry of Piperazinediones Derived from 2‑Amino-4,7-dialkoxyindan-2-carboxyl... von Wells, Kirk E, Weatherhead, Robin A, Murigi, Francis N, Nichol, Gary S, Carducci, Michael D, Selby, Hugh D, Mash, Eugene A

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A synchrotron study of (2R,5′S)-5′-benzyl-5-bromo-6-methoxyspiro[indane-2,2′-piperazine]-3′,6′-dione dimethylformamide solvate von Nichol, Gary S., Murigi, Francis N., Mash, Eugene A.

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Galeterone and VNPT 55 disrupt Mnk‐ eIF 4E to inhibit prostate cancer cell migration and invasion von Kwegyir‐Afful, Andrew K., Bruno, Robert D., Purushottamachar, Puranik, Murigi, Francis N., Njar, Vincent C.O.

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