Total Synthesis of (+)-Azaspiracid-1. An Exhibition of the Intricacies of Complex Molecule Synthesis von Evans, David A, Kværnø, Lisbet, Dunn, Travis B, Beauchemin, André, Raymer, Brian, Mulder, Jason A, Olhava, Edward J, Juhl, Martin, Kagechika, Katsuji, Favor, David A

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A Copper-Catalyzed C−N Bond Formation Involving sp-Hybridized Carbons. A Direct Entry to Chiral Ynamides via N-Alkynylation of Amides von Frederick, Michael O, Mulder, Jason A, Tracey, Michael R, Hsung, Richard P, Huang, Jian, Kurtz, Kimberly C. M, Shen, Lichun, Douglas, Christopher J

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The First Successful Base-Promoted Isomerization of Propargyl Amides to Chiral Ynamides. Applications in Ring-Closing Metathesis of Ene−Ynamides and Tandem RCM of Diene−Ynamides... von Huang, Jian, Xiong, Hui, Hsung, Richard P, Rameshkumar, C, Mulder, Jason A, Grebe, Tyler P

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Total Synthesis of (+)-Azaspiracid-1. Part II: Synthesis of the EFGHI Sulfone and Completion of the Synthesis von Evans, David A., Dunn, Travis B., Kværnø, Lisbet, Beauchemin, André, Raymer, Brian, Olhava, Edward J., Mulder, Jason A., Juhl, Martin, Kagechika, Katsuji, Favor, David A.

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Development of an Efficient Synthesis of (2-Aminopyrimidin-5-yl) Boronic Acid von Patel, Nitinchandra D, Zhang, Yongda, Gao, Joe, Sidhu, Kanwar, Lorenz, Jon C, Fandrick, Keith R, Mulder, Jason A, Herbage, Melissa A, Li, Zhibin, Ma, Shengli, Lee, Heewon, Grinberg, Nelu, Song, Jinhua J, Busacca, Carl A, Yee, Nathan K, Senanayake, Chris H

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Total Synthesis of (+)-Azaspiracid-1. Part I: Synthesis of the Fully Elaborated ABCD Aldehyde von Evans, David A., Kværnø, Lisbet, Mulder, Jason A., Raymer, Brian, Dunn, Travis B., Beauchemin, André, Olhava, Edward J., Juhl, Martin, Kagechika, Katsuji

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The First Stereoselective Ficini−Claisen Rearrangement Using Chiral Ynamides von Mulder, Jason A, Hsung, Richard P, Frederick, Michael O, Tracey, Michael R, Zificsak, Craig A

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Highly Stereoselective Saucy−Marbet Rearrangement Using Chiral Ynamides. Synthesis of Highly Substituted Chiral Homoallenyl Alcohols von Frederick, Michael O, Hsung, Richard P, Lambeth, Robert H, Mulder, Jason A, Tracey, Michael R

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A Michael Equilibration Model To Control Site Selectivity in the Condensation toward Aminopyrazoles von Fandrick, Daniel R, Sanyal, Sanjit, Kaloko, Joseph, Mulder, Jason A, Wang, Yuwen, Wu, Ling, Lee, Heewon, Roschangar, Frank, Hoffmann, Matthias, Senanayake, Chris H

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One-Pot Synthesis of 2,5-Disubstituted Pyrimidines from Nitriles von Frutos, Rogelio P, Wei, Xudong, Patel, Nitinchandra D, Tampone, Thomas G, Mulder, Jason A, Busacca, Carl A, Senanayake, Chris H

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Development of a Practical Process for the Synthesis of PDE4 Inhibitors von Frutos, Rogelio P, Tampone, Thomas G, Mulder, Jason A, Rodriguez, Sonia, Yee, Nathan K, Yang, Bing-Shiou, Senanayake, Chris H

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Remarkable Enhancement of Enantioselectivity in the Asymmetric Conjugate Addition of Dimethylzinc to (Z)-Nitroalkenes with a Catalytic [(MeCN)4Cu]PF6-Hoveyda Ligand Complex von Zeng, Xingzhong, Gao, Joe J., Song, Jinhua J., Ma, Shengli, Desrosiers, Jean-Nicolas, Mulder, Jason A., Rodriguez, Sonia, Herbage, Melissa A., Haddad, Nizar, Qu, Bo, Fandrick, Keith R., Grinberg, Nelu, Lee, Heewon, Wei, Xudong, Yee, Nathan K., Senanayake, Chris H.

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Development of an Asymmetric Synthesis of a Chiral Quaternary FLAP Inhibitor von Fandrick, Keith R, Mulder, Jason A, Patel, Nitinchandra D, Gao, Joe, Konrad, Michael, Archer, Elizabeth, Buono, Frederic G, Duran, Adil, Schmid, Rolf, Daeubler, Juergen, Desrosiers, Jean-Nicolas, Zeng, Xingzhong, Rodriguez, Sonia, Ma, Shengli, Qu, Bo, Li, Zhibin, Fandrick, Daniel R, Grinberg, Nelu, Lee, Heewon, Bosanac, Todd, Takahashi, Hidenori, Chen, Zhidong, Bartolozzi, Alessandra, Nemoto, Peter, Busacca, Carl A, Song, Jinhua J, Yee, Nathan K, Mahaney, Paige E, Senanayake, Chris H

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Addressing the Configuration Stability of Lithiated Secondary Benzylic Carbamates for the Development of a Noncryogenic Stereospecific Boronate Rearrangement von Fandrick, Keith R, Patel, Nitinchandra D, Mulder, Jason A, Gao, Joe, Konrad, Michael, Archer, Elizabeth, Buono, Frederic G, Duran, Adil, Schmid, Rolf, Daeubler, Juergen, Fandrick, Daniel R, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Busacca, Carl A, Song, Jinhua J, Yee, Nathan K, Senanayake, Chris H

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Development of a Safe and Economical Synthesis of Methyl 6‑Chloro-5-(trifluoromethyl)nicotinate: Trifluoromethylation on Kilogram Scale von Mulder, Jason A, Frutos, Rogelio P, Patel, Nitinchandra D, Qu, Bo, Sun, Xiufeng, Tampone, Thomas G, Gao, Joe, Sarvestani, Max, Eriksson, Magnus C, Haddad, Nizar, Shen, Sherry, Song, Jinhua J, Senanayake, Chris H

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Early Development Scale-Up of a Structurally-Challenging 5‑Lipoxygenase Activating Protein (FLAP) Inhibitor von Mulder, Jason A, Gao, Joe, Fandrick, Keith R, Zeng, Xingzhong, Desrosiers, Jean-Nicolas, Patel, Nitinchandra D, Li, Zhibin, Rodriguez, Sonia, Lorenz, Jon C, Wang, Jun, Ma, Shengli, Fandrick, Daniel R, Grinberg, Nelu, Lee, Heewon, Bosanac, Todd, Takahashi, Hidenori, Chen, Zhidong, Bartolozzi, Alessandra, Nemoto, Peter, Busacca, Carl A, Song, Jinhua J, Yee, Nathan K, Mahaney, Paige E, Senanayake, Chris H

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Highly Stereoselective Synthesis of Novel α-Haloenamides via a Mild and Efficient Hydrohalogenation of Ynamides von Mulder, Jason A, Kurtz, Kimberly C. M, Hsung, Richard P, Coverdale, Heather, Frederick, Michael O, Shen, Lichun, Zificsak, Craig A

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Sonogashira Cross-Couplings of Ynamides. Syntheses of Urethane- and Sulfonamide-Terminated Conjugated Phenylacetylenic Systems von Tracey, Michael R, Zhang, Yanshi, Frederick, Michael O, Mulder, Jason A, Hsung, Richard P

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Synthesis of chiral allenes from ynamides through a highly stereoselective Saucy–Marbet rearrangement von Kurtz, Kimberly C.M., Frederick, Michael O., Lambeth, Robert H., Mulder, Jason A., Tracey, Michael R., Hsung, Richard P.

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A new and practical boronic acid catalyzed intramolecular cyclodehydration of ureas for the synthesis of LFA-1 antagonists von Frutos, Rogelio P., Tampone, Thomas, Mulder, Jason A., Xu, Yibo, Reeves, Diana, Wang, Xiao-Jun, Zhang, Li, Krishnamurthy, Dhileepkumar, Senanayake, Chris H.

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