Immune Checkpoint PD‐1/PD‐L1: Is There Life Beyond Antibodies? von Konstantinidou, Markella, Zarganes‐Tzitzikas, Tryfon, Magiera‐Mularz, Katarzyna, Holak, Tad A., Dömling, Alexander

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Bioactive Macrocyclic Inhibitors of the PD‐1/PD‐L1 Immune Checkpoint von Magiera‐Mularz, Katarzyna, Skalniak, Lukasz, Zak, Krzysztof M., Musielak, Bogdan, Rudzinska‐Szostak, Ewa, Berlicki, Łukasz, Kocik, Justyna, Grudnik, Przemyslaw, Sala, Dominik, Zarganes‐Tzitzikas, Tryfon, Shaabani, Shabnam, Dömling, Alexander, Dubin, Grzegorz, Holak, Tad A.

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Nutlin‐3a‐aa: Improving the Bioactivity of a p53/MDM2 Interaction Inhibitor by Introducing a Solvent‐Exposed Methylene Group von Nietzold, Florian, Rubner, Stefan, Labuzek, Beata, Golik, Przemysław, Surmiak, Ewa, Corte, Xabier, Kitel, Radoslaw, Protzel, Christoph, Reppich‐Sacher, Regina, Stichel, Jan, Magiera‐Mularz, Katarzyna, Holak, Tad A., Berg, Thorsten

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A combined approach of structure‐based virtual screening and NMR to interrupt the PD‐1/PD‐L1 axis: Biphenyl‐benzimidazole containing compounds as novel PD‐L1 inhibitors von Donati, Greta, Viviano, Monica, D'Amore, Vincenzo Maria, Cipriano, Alessandra, Diakogiannaki, Isidora, Amato, Jussara, Tomassi, Stefano, Brancaccio, Diego, Russomanno, Pasquale, Di Leva, Francesco Saverio, Arosio, Daniela, Seneci, Pierfausto, Taliani, Sabrina, Magiera‐Mularz, Katarzyna, Musielak, Bogdan, Skalniak, Lukasz, Holak, Tad A., Castellano, Sabrina, La Pietra, Valeria, Marinelli, Luciana

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CA-170 - A Potent Small-Molecule PD-L1 Inhibitor or Not? von Musielak, Bogdan, Kocik, Justyna, Skalniak, Lukasz, Magiera-Mularz, Katarzyna, Sala, Dominik, Czub, Miroslawa, Stec, Malgorzata, Siedlar, Maciej, Holak, Tad A, Plewka, Jacek

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Design, Synthesis, Evaluation, and Structural Studies of C2-Symmetric Small Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction von Basu, Subhadwip, Yang, Jeffrey, Xu, Bin, Magiera-Mularz, Katarzyna, Skalniak, Lukasz, Musielak, Bogdan, Kholodovych, Vladyslav, Holak, Tad A, Hu, Longqin

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Correction: Reyes Romero et al. Computer- and NMR-Aided Design of Small-Molecule Inhibitors of the Hub1 Protein. Molecules 2022, 27 , 8282 von Reyes Romero, Atilio, Kubica, Katarzyna, Kitel, Radoslaw, Rodríguez, Ismael, Magiera-Mularz, Katarzyna, Dömling, Alexander, Holak, Tad A, Surmiak, Ewa

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PD-L1 Inhibitors: Different Classes, Activities, and Mechanisms of Action von Surmiak, Ewa, Magiera-Mularz, Katarzyna, Musielak, Bogdan, Muszak, Damian, Kocik-Krol, Justyna, Kitel, Radoslaw, Plewka, Jacek, Holak, Tad A, Skalniak, Lukasz

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Development of selective ssDNA micro-probe for PD1 detection as a novel strategy for cancer imaging von Malicki, Stanisław, Czarna, Anna, Żyła, Edyta, Pucelik, Barbara, Gałan, Wojciech, Chruścicka, Barbara, Kamińska, Marta, Sochaj-Gregorczyk, Alicja, Magiera-Mularz, Katarzyna, Wang, Jun, Winiarski, Marek, Benedyk-Machaczka, Małgorzata, Kozieł, Joanna, Dubin, Grzegorz, Mydel, Piotr

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Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions von Musielak, Bogdan, Janczyk, Weronika, Rodriguez, Ismael, Plewka, Jacek, Sala, Dominik, Magiera-Mularz, Katarzyna, Holak, Tad

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Computer- and NMR-Aided Design of Small-Molecule Inhibitors of the Hub1 Protein von Reyes Romero, Atilio, Kubica, Katarzyna, Kitel, Radoslaw, Rodríguez, Ismael, Magiera-Mularz, Katarzyna, Dömling, Alexander, Holak, Tad A, Surmiak, Ewa

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Quiz WHAT IS YOUR DIAGNOSIS? von Püsküllüoglu, Mirosława, Kruczak, Anna, Mularz, Katarzyna, Rozmus, Magdalena, Grela-Wojewoda, Aleksandra, Ryś, Janusz

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Identification of small-molecule inhibitors of USP2a von Tomala, Marcin D., Magiera-Mularz, Katarzyna, Kubica, Katarzyna, Krzanik, Sylwia, Zieba, Bartosz, Musielak, Bogdan, Pustula, Marcin, Popowicz, Grzegorz M., Sattler, Michael, Dubin, Grzegorz, Skalniak, Lukasz, Holak, Tad A.

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Macrocyclic Peptide Inhibitor of PD‐1/PD‐L1 Immune Checkpoint von Magiera‐Mularz, Katarzyna, Kuska, Katarzyna, Skalniak, Lukasz, Grudnik, Przemyslaw, Musielak, Bogdan, Plewka, Jacek, Kocik, Justyna, Stec, Malgorzata, Weglarczyk, Kazimierz, Sala, Dominik, Wladyka, Benedykt, Siedlar, Maciej, Holak, Tad A., Dubin, Grzegorz

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Peptide-based inhibitors targeting the PD-1/PD-L1 axis: potential immunotherapeutics for cancer von Bojko, Magdalena, Węgrzyn, Katarzyna, Sikorska, Emilia, Ciura, Piotr, Battin, Claire, Steinberger, Peter, Magiera-Mularz, Katarzyna, Dubin, Grzegorz, Kulesza, Adam, Sieradzan, Adam K., Spodzieja, Marta, Rodziewicz-Motowidło, Sylwia

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Structural and biological characterization of pAC65, a macrocyclic peptide that blocks PD-L1 with equivalent potency to the FDA-approved antibodies von Rodriguez, Ismael, Kocik-Krol, Justyna, Skalniak, Lukasz, Musielak, Bogdan, Wisniewska, Aneta, CiesioÅkiewicz, Agnieszka, Berlicki, Åukasz, Plewka, Jacek, Grudnik, Przemyslaw, Stec, Malgorzata, Siedlar, Maciej, Holak, Tad A, Magiera-Mularz, Katarzyna

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Human and mouse PD-L1: similar molecular structure, but different druggability profiles von Magiera-Mularz, Katarzyna, Kocik, Justyna, Musielak, Bogdan, Plewka, Jacek, Sala, Dominik, Machula, Monika, Grudnik, Przemyslaw, Hajduk, Malgorzata, Czepiel, Marcin, Siedlar, Maciej, Holak, Tad A., Skalniak, Lukasz

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Biphenyl Ether Analogs Containing Pomalidomide as Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed Cell Death-Ligand 1 Interaction von Shaabani, Shabnam, Gadina, Louis, Surmiak, Ewa, Wang, Zefeng, Zhang, Bidong, Butera, Roberto, Zarganes-Tzitzikas, Tryfon, Rodriguez, Ismael, Kocik-Krol, Justyna, Magiera-Mularz, Katarzyna, Skalniak, Lukasz, Dömling, Alexander, Holak, Tad A

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Quiz. What is your diagnosis? von Krupińska, Martyna, Kaznowska, Ewa, Kruczak, Anna, Mularz, Katarzyna, Długosz, Jarosław, Gancarz, Józef, Ryś, Janusz

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Primary cardiac atrial sarcomas. Report of two histologically different cases and review of the literature von Püsküllüoglu, Mirosława, Kruczak, Anna, Mularz, Katarzyna, Rozmus, Magdalena, Harazin-Lechowska, Agnieszka, Pietruszka, Agnieszka, Jaworska, Justyna, Ziobro, Marek, Grela-Wojewoda, Aleksandra, Ryś, Janusz

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