Synthesis of sp-rich scaffolds for molecular libraries through complexity-generating cascade reactions von Flagstad, T, Min, G, Bonnet, K, Morgentin, R, Roche, D, Clausen, M. H, Nielsen, T. E

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272 8-(1-Anilino)ethyl)-2-morpholino-4-oxo-4H-chromene-6-carboxamides as PI3Kbeta/delta inhibitors: structure–activity relationships and identification of AZD8186, a clinical candi... von Barlaam, B, Cosulich, S, Degorce, S, Fitzek, M, Green, S, Hancox, U, Lambert-van der Brempt, C, Lohmann, J.J, Maudet, M, Morgentin, R, Pasquest, M.J, Peru, A, Ple, P, Saleh, T, Vautier, M, Walker, M, Ward, L, Warin, N

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Synthesis of sp 3 -rich scaffolds for molecular libraries through complexity-generating cascade reactions von Flagstad, T., Min, G., Bonnet, K., Morgentin, R., Roche, D., Clausen, M. H., Nielsen, T. E.

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Trichloroacetylhydrazones: new highly reactive alkylating agents von Atlan, V., El Kaim, L., Lacroix, S., Morgentin, R.

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5-Substituted 4-anilinoquinazolines as potent, selective and orally active inhibitors of erbB2 receptor tyrosine kinase von Ballard, Peter, Bradbury, Robert H., Hennequin, Laurent F.A., Hickinson, D. Mark, Johnson, Paul D., Kettle, Jason G., Klinowska, Teresa, Morgentin, Remy, Ogilvie, Donald J., Olivier, Annie

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Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket von Ballard, Peter, Bradbury, Robert H., Harris, Craig S., Hennequin, Laurent F.A., Hickinson, Mark, Johnson, Paul D., Kettle, Jason G., Klinowska, Teresa, Leach, Andrew G., Morgentin, Remy, Pass, Martin, Ogilvie, Donald J., Olivier, Annie, Warin, Nicolas, Williams, Emma J.

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New heterocyclic analogues of 4-(2-chloro-5-methoxyanilino)quinazolines as potent and selective c-Src kinase inhibitors von Barlaam, Bernard, Fennell, Mike, Germain, Hervé, Green, Tim, Hennequin, Laurent, Morgentin, Rémy, Olivier, Annie, Plé, Patrick, Vautier, Michel, Costello, Gerard

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Trichloroacetic acid hydrazones I: New formation of 1,3,4-oxadiazoles from aldehydes von El Kaim, Laurent, Le Menestrel, Isabelle, Morgentin, Remy

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Asymmetric Syntheses of Enantiopure 4-Substituted Pipecolic Acid Derivatives von Agami, Claude, Bisaro, Fabrice, Comesse, Sébastien, Guesné, Sébastien, Kadouri-Puchot, Catherine, Morgentin, Rémy

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Asymmetric Synthesis of Unsaturated Pipecolic Acid Derivatives von Agami, Claude, Bihan, Dominique, Morgentin, Rémy, Puchot-Kadouri, Cathy

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Translation of Innovative Chemistry into Screening Libraries: An Exemplar Partnership from the European Lead Factory von Morgentin, R, Dow, M, Aimon, A, Karageorgis, G, Kalliokoski, T, Roche, D, Marsden, S, Nelson, AS

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Realisation of small molecule libraries based on frameworks distantly related to natural products von Aimon, A, Karageorgis, G, Masters, J, Dow, M, Craven, PGE, Ohsten, M, Willaume, A, Morgentin, R, Ruiz-Llamas, N, Lemoine, H, Kalliokoski, T, Eatherton, AJ, Foley, DJ, Marsden, SP, Nelson, A

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Expansion of chemical space for collaborative lead generation and drug discovery: the European Lead Factory Perspective von Karawajczyk, A, Giordanetto, F, Benningshof, J, Hamza, D, Kalliokoski, T, Pouwer, K, Morgentin, R, Nelson, A, Muller, G, Piechot, A, Tzalis, D

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Exploitation of the Ugi-Joullie Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins von Firth, JD, Zhang, R, Morgentin, R, Guilleux, R, Kalliokoski, T, Warriner, S, Foster, R, Marsden, SP, Nelson, A

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ChemInform Abstract: Trichloroacetylhydrazones: New Highly Reactive Alkylating Agents von Atlan, V., El Kaim, L., Lacroix, S., Morgentin, R.

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ChemInform Abstract: Trichloroacetic Acid Hydrazones. Part 1: New Formation of 1,3,4-Oxadiazoles from Aldehydes von EL KAIM, L., LE MENESTREL, I., MORGENTIN, R.

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ChemInform Abstract: Asymmetric Synthesis of Unsaturated Pipecolic Acid Derivatives von AGAMI, C., BIHAN, D., MORGENTIN, R., PUCHOT-KADOURI, C.

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