Efficient Azacycle Formations Developed in Japanese Pharmaceutical Industries: Elegancy, Logistics, and Training (ELT) “Sandwich” for Process Chemists von Mizufune, Hideya

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A Nitrogen-Assisted One-Pot Heteroaryl Ketone Synthesis from Carboxylic Acids and Heteroaryl Halides von Demkiw, Krystyna, Araki, Hirofumi, Elliott, Eric L, Franklin, Christopher L, Fukuzumi, Yoonjoo, Hicks, Frederick, Hosoi, Kazushi, Hukui, Tadashi, Ishimaru, Yoichiro, O’Brien, Erin, Omori, Yoshimasa, Mineno, Masahiro, Mizufune, Hideya, Sawada, Naotaka, Sawai, Yasuhiro, Zhu, Lei

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Integrated Pd-catalyzed cross-coupling strategies for furnishing α-carbolines von Sera, Misayo, Mizufune, Hideya, Ueda, Tsuyoshi, Mineno, Masahiro, Zanka, Atsuhiko

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Ligand-free Heck–Mizoroki reaction for 1,3,5-Trisubstituted Pyrazoles von Sera, Misayo, Mizufune, Hideya, Tawada, Hiroyuki

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Double Reformatsky Reaction: Divergent Synthesis of δ‑Hydroxy-β-ketoesters von Mineno, Masahiro, Sawai, Yasuhiro, Kanno, Kazuaki, Sawada, Naotaka, Mizufune, Hideya

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Expedient Pd‐Catalyzed α‐Arylation towards Dibenzoxepinones: Pivotal Manske's Ketone for the Formal Synthesis of Cularine Alkaloids von Deichert, Julie A., Mizufune, Hideya, Patel, Jignesh J., Hurst, Timothy E., Maheta, Ashish, Kitching, Matthew O., Ross, Avena C., Snieckus, Victor

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A rapid and diverse construction of 6-substituted-5,6-dihydro-4-hydroxy-2-pyrones through double Reformatsky reaction von Mineno, Masahiro, Sawai, Yasuhiro, Kanno, Kazuaki, Sawada, Naotaka, Mizufune, Hideya

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Integrated Cross-Coupling Strategy for an α‑Carboline-Based Aurora B Kinase Inhibitor von Mineno, Masahiro, Sera, Misayo, Ueda, Tsuyoshi, Mizufune, Hideya, Zanka, Atsuhiko, O’Bryan, Colin, Brown, Jason, Scorah, Nick

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Rapid access to diverse α-carbolines through sequential transition metal catalyzed amination and direct C–H arylation von Mineno, Masahiro, Sera, Misayo, Ueda, Tsuyoshi, Mizuno, Masahiro, Yamano, Mitsuhisa, Mizufune, Hideya, Zanka, Atsuhiko

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Process research on arylnaphthalene lignan aza-analogues: a new palladium-catalyzed benzannulation of α,β-bisbenzylidenesuccinic acid derivatives von Mizufune, Hideya, Nakamura, Minoru, Mitsudera, Hiroyuki

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A new efficient synthetic strategy for N-(dialkylamino)azacycle as a tetrasubstituted hydrazine derivative using sodium triacyloxyborohydride von Mizufune, Hideya, Yamamoto, Hiroaki, Nakamura, Minoru, Miki, Shokyo

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Effects of α-Substituents on Ion Selectivity of Bis(12-crown-4-methyl) Malonates as Neutral Carriers for Sodium Ion-Selective Electrodes von KIMURA, Keiichi, YOSHINAGA, Masanobu, FUNAKI, Kaoru, SHIBUTANI, Yasuhiko, YAKABE, Kenji, SHONO, Toshiyuki, KASAI, Mitsuhiro, MIZUFUNE, Hideya, TANAKA, Minoru

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The first regiospecific synthesis of helioxanthin by novel palladium-catalyzed benzannulation reaction of α,β-bisbenzylidene-γ-lactone von Mizufune, Hideya, Nakamura, Minoru, Mitsudera, Hiroyuki

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Process for producing pyrrole compound von Yamasaki, Takeshi, Mizufune, Hideya, Nagata, Toshiaki, Ikemoto, Tomomi

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INTERMEDIATES FOR USE IN A PROCESS OF PRODUCING PYRROLE COMPOUNDS von SERA, MISAYO, MIZUFUNE, HIDEYA, YAMASAKI, TAKESHI, IKEMOTO, TOMOMI, NAGATA, TOSHIAKI, FUKUDA, NAOHIRO

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Process development of potassium channel opener, TCV-295, based on convenient ring formation of 2H-1,3-benzoxazine and selective N-oxidation of the pyridyl moiety von Mizufune, Hideya, Irie, Hiroyuki, Katsube, Susumu, Okada, Tadataka, Mizuno, Yukio, Arita, Miichiro

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PROCESS FOR PRODUCING PYRROLE COMPOUND von Fukuda, Naohiro, Yamasaki, Takeshi, Mizufune, Hideya, Nagata, Toshiaki, Sera, Misayo, Ikemoto, Tomomi

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ChemInform Abstract: Ligand-free Heck-Mizoroki Reaction for 1,3,5-Trisubstituted Pyrazoles von Sera, Misayo, Mizufune, Hideya, Tawada, Hiroyuki

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PROCESS FOR PRODUCING PYRROLE COMPOUND von FUKUDA, Naohiro, MIZUFUNE, Hideya, SERA, Misayo, NAGATA, Toshiaki, YAMASAKI, Takeshi, IKEMOTO, Tomomi

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PROCESS FOR PRODUCING PYRROLE COMPOUND von FUKUDA, Naohiro, MIZUFUNE, Hideya, SERA, Misayo, NAGATA, Toshiaki, YAMASAKI, Takeshi, IKEMOTO, Tomomi

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