Ligands of the neuropeptide Y Y2 receptor von Mittapalli, Gopi Kumar, Roberts, Edward

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Mapping the Landscape of Potentially Primordial Informational Oligomers: Oligodipeptides and Oligodipeptoids Tagged with Triazines as Recognition Elements von Mittapalli, Gopi Kumar, Reddy, Kondreddi Ravinder, Xiong, Hui, Munoz, Omar, Han, Bo, De Riccardis, Francesco, Krishnamurthy, Ramanarayanan, Eschenmoser, Albert

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A Deep Hydrophobic Binding Cavity is the Main Interaction for Different Y2R Antagonists von Burkert, Kerstin, Zellmann, Tristan, Meier, René, Kaiser, Anette, Stichel, Jan, Meiler, Jens, Mittapalli, Gopi K., Roberts, Edward, Beck‐Sickinger, Annette G.

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A Deep Hydrophobic Binding Cavity is the Main Interaction for Different Y 2 R Antagonists von Burkert, Kerstin, Zellmann, Tristan, Meier, René, Kaiser, Anette, Stichel, Jan, Meiler, Jens, Mittapalli, Gopi K, Roberts, Edward, Beck-Sickinger, Annette G

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Mapping the Landscape of Potentially Primordial Informational Oligomers: Oligodipeptides Tagged with 2,4-Disubstituted 5-Aminopyrimidines as Recognition Elements von Mittapalli, Gopi Kumar, Osornio, Yazmin M., Guerrero, Miguel A., Reddy, Kondreddi Ravinder, Krishnamurthy, Ramanarayanan, Eschenmoser, Albert

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Discovery of ITX 4520: A highly potent orally bioavailable hepatitis C virus entry inhibitor von Mittapalli, Gopi Kumar, Zhao, Fang, Jackson, Andrew, Gao, Hongfeng, Lee, Haekyung, Chow, Stephine, Kaur, Maninder Pal, Nguyen, Natalie, Zamboni, Robert, McKelvy, Jeffrey, Wong-Staal, Flossie, Macdonald, James E.

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Synthesis and SAR of selective small molecule neuropeptide Y Y2 receptor antagonists von Mittapalli, Gopi Kumar, Vellucci, Danielle, Yang, Jun, Toussaint, Marion, Brothers, Shaun P., Wahlestedt, Claes, Roberts, Edward

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890-P: Ultraselective DYRK1A/B Inhibitors Mediated ß-Cell Proliferation and Insulin Production In Vitro and In Vivo von Mittapalli, Gopi Kumar, Mak, Chi-Ching, Bossard, Carine, Vakiti, Ramkrishna Reddy, Creger, Emily, Gutierrez, Erik, Horsley, Erich A, Swearingen, Christopher, Hill, John S

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Tau pathology reduction with SM07883, a novel, potent, and selective oral DYRK1A inhibitor: A potential therapeutic for Alzheimer's disease von Melchior, Benoît, Mittapalli, Gopi Kumar, Lai, Carolyn, Duong‐Polk, Karen, Stewart, Joshua, Güner, Bora, Hofilena, Brian, Tjitro, Amanda, Anderson, Scott D., Herman, David S., Dellamary, Luis, Swearingen, Christopher J., Sunil, K.C., Yazici, Yusuf

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O4‐05‐03: TAU PATHOLOGY REDUCTION WITH SM07883, A NOVEL, POTENT, AND SELECTIVE ORAL DYRK1A INHIBITOR: A POTENTIAL THERAPEUTIC FOR ALZHEIMER'S DISEASE von Melchior, Ben, Lai, Carolyn, Duong-Polk, Karen, Tjitro, Amanda, Ince, Deniz C., Stewart, Joshua, Dellamary, Luis, Hofilena, Brian, Mittapalli, Gopi, KC, Sunil, Yazici, Yusuf

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TAU PATHOLOGY REDUCTION WITH SM07883, A NOVEL, POTENT, AND SELECTIVE ORAL DYRK1A INHIBITOR: A POTENTIAL THERAPEUTIC FOR ALZHEIMER’S DISEASE von Melchior, Ben, Lai, Carolyn, Duong-Polk, Karen, Tjitro, Amanda, Ince, Deniz C., Stewart, Joshua, Dellamary, Luis, Hofilena, Brian, Mittapalli, Gopi, KC, Sunil, Yazici, Yusuf

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Abstract 5019: Next-generation DYRK1A inhibitors as a new therapeutic approach for the treatment of hematological malignancies von Jarvis, Matthew C., Mittapalli, Gopi, Creger, Emily, Nora, Chelsea, Ibanez, Maureen, Bhat, Deepti, Hofilena, Brian, Stewart, Josh, McMillan, Elizabeth A., Falahatpisheh, Hadi, Mak, Chi-Ching, White, Michael, Hill, John S., Bossard, Carine

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A Deep Hydrophobic Binding Cavity is the Main Interaction for Different Y sub(2)R Antagonists von Burkert, Kerstin, Zellmann, Tristan, Meier, Rene, Kaiser, Anette, Stichel, Jan, Meiler, Jens, Mittapalli, Gopi K, Roberts, Edward, Beck-Sickinger, Annette G

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Different Y2 receptor antagonists share the same deep, hydrophobic binding pocket von Burkert, Kerstin, Zellmann, Tristan, Mittapalli, Gopi Kumar, Roberts, Edward, Beck-Sickinger, Annette G

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Discovery of highly potent small molecule Hepatitis C Virus entry inhibitors von Mittapalli, Gopi Kumar, Jackson, Andrew, Zhao, Fang, Lee, Haekyung, Chow, Stephine, McKelvy, Jeffrey, Wong-Staal, Flossie, Macdonald, James E.

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A Deep Hydrophobic Binding Cavity is the Main Interaction for Different Y2 R Antagonists von Burkert, Kerstin, Zellmann, Tristan, Meier, René, Kaiser, Anette, Stichel, Jan, Meiler, Jens, Mittapalli, Gopi K, Roberts, Edward, Beck-Sickinger, Annette G

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Design, synthesis, conformational and membrane ion transport studies of proline-adamantane hybrid cyclic depsipeptides von Karle, Isabella L., Ranganathan, Darshan, Kumar, Mittapalli Gopi, Nagaraj, Ramakrishnan

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Cover Picture: Mapping the Landscape of Potentially Primordial Informational Oligomers: Oligodipeptides and Oligodipeptoids Tagged with Triazines as Recognition Elements / Mapping... von Mittapalli, Gopi Kumar, Reddy, Kondreddi Ravinder, Xiong, Hui, Munoz, Omar, Han, Bo, De Riccardis, Francesco, Krishnamurthy, Ramanarayanan, Eschenmoser, Albert, Osornio, Yazmin M., Guerrero, Miguel A.

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4-AMINOPYRROLO[2,1-F][1,2,4]TRIAZINES AND PREPARATION AND USES THEREOF von HOFILENA, Brian, VAKITI, Ramkrishna, TURNER, Lewis, MAK, Chi, MITTAPALLI, Gopi, EASTMAN, Brian

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PYRROLO[2,1-F][1,2,4]TRIAZINES AND PREPARATION AND USES THEREOF von MAK, Chi Ching, TURNER, Lewis Daniel, HOFILENA, Brian Joseph, VAKITI, Ramkrishna Reddy, MITTAPALLI, Gopi Kumar, EASTMAN, Brian Walter

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