Synthesis, X-Ray Crystal Structure, Hirshfeld Surface Analysis, and Molecular Docking Study of Novel Hepatitis B (HBV) Inhibitor: 8-Fluoro-5-(4-fluorobenzyl)-3-(2-methoxybenzyl)-3,... von Ivashchenko, Aleksandr V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kuznetsova, Irina V., Kovalenko, Sergiy M., Bunyatyan, Natalya D., Langer, Thierry

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Synthesis, X-ray crystal structure, Hirshfeld surface analysis, and molecular docking study of novel inhibitor of hepatitis B: methyl 4-fluoro-3-(morpholinosulfonyl)benzo[b]thiophe... von Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Dmitrieva, Irina G., Ivanov, Vladimir V., Langer, Thierry

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Novel One-Pot Synthesis of Methyl 4-Hydroxy-2-thioxo-1,2-dihydroquinoline-3-carboxylate: Synthetic and Crystallographic Studies von Kovalenko, Sergiy M., Drushlyak, Oleksandr G., Konovalova, Irina S., Mariutsa, Illia O., Kravchenko, Dmitry V., Ivachtchenko, Alexandre V., Mitkin, Oleg D.

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Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses von Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Ryakhovskiy, Alexey, Karapetian, Ruben N, Kravchenko, Dmitry V, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V

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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) A... von Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M

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Synthesis, inhibitory activity and oral dosing formulation of AV5124, the structural analogue of influenza virus endonuclease inhibitor baloxavir von Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Karapetian, Ruben N, Kravchenko, Dmitry V, Mochalov, Stephan V, Ryakhovskiy, Alexey A, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V

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Synthesis, biological evaluation and in silico modeling of novel integrase strand transfer inhibitors (INSTIs) von Ivashchenko, Andrey A., Ivanenkov, Yan A., Koryakova, Angela G., Karapetian, Ruben N., Mitkin, Oleg D., Aladinskiy, Vladimir A., Kravchenko, Dmitry V., Savchuk, Nikolai P., Ivashchenko, Alexander V.

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Synthesis, biological evaluation and in silico modeling of novel pan-genotypic NS5A inhibitors von Ivashchenko, Andrey A., Ivanenkov, Yan A., Aladinskiy, Vladimir A., Karapetian, Ruben N., Koryakova, Angela G., Ryakhovskiy, Alexey A., Mitkin, Oleg D., Kravchenko, Dmitry V., Savchuk, Nikolai P., Zagribelnyy, Bogdan A., Ivashchenko, Alexander V.

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Photoactive Barbiturate Receptors:  An Ultimate Lock-and-Key System in Which the Key Unlocks the Lock von Lakkakula, Suman, Mitkin, Oleg D, Valiulin, Roman A, Kutateladze, Andrei G

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Safety and efficacy of aviandr in patients with generalized anxiety disorder: A multicenter, randomized, double-blind, placebo-controlled, dose-finding, pilot study von Ivashchenko, Andrey A., Morozova, Margarita A., Vostokova, Natalia V., Beniashvily, Allan G., Bukhanovskaya, Olga A., Burminskiy, Denis S., Egorova, Alina N., Gluskina, Lubov Y., Gorchakov, Dmitriy S., Karapetian, Ruben N., Kasimova, Lala N., Kravchenko, Dmitry V., Lepilkina, Taissia A., Merkulova, Elena A., Mitkin, Oleg D., Penchul, Nataliya A., Potanin, Sergey S., Rupchev, George E., Ivachtchenko, Alexandre V.

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(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor von Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Okun, Ilya M, Tkachenko, Sergey E, Vorobiev, Anton A

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Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists von Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Vorobiev, Anton A., Kuznetsova, Irina V., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Trifelenkov, Andrey S., Kravchenko, Dmitry V., Veselov, Mark S., Chufarova, Nina V.

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Novel oral anti-influenza drug candidate AV5080 von Ivachtchenko, Alexandre V, Ivanenkov, Yan A, Mitkin, Oleg D, Yamanushkin, Pavel M, Bichko, Vadim V, Shevkun, Natalia A, Karapetian, Ruben N, Leneva, Irina A, Borisova, Olga V, Veselov, Mark S

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Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya

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Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines—Synthesis and ‘s... von Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Vorobiev, Anton A., Okun, Ilya

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Discovery of Novel Highly Potent Hepatitis C Virus NS5A Inhibitor (AV4025) von Ivachtchenko, Alexandre V, Mitkin, Oleg D, Yamanushkin, Pavel M, Kuznetsova, Irina V, Bulanova, Elena A, Shevkun, Natalia A, Koryakova, Angela G, Karapetian, Ruben N, Bichko, Vadim V, Trifelenkov, Andrey S, Kravchenko, Dmitry V, Vostokova, Natalia V, Veselov, Mark S, Chufarova, Nina V, Ivanenkov, Yan A

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Crystal structure, Hirshfeld analysis and a molecular docking study of a new inhibitor of the Hepatitis B virus (HBV): ethyl 5-methyl-1,1-dioxo-2-{[5-(pentan-3-yl)-1,2,4-oxadiazol-... von Alexandre V. Ivachtchenko, Sergiy M. Kovalenko, Dmitry V. Kravchenko, Oleg D. Mitkin, Vladimir V. Ivanov, Thierry Langer

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2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: new series of highly potent and specific serotonin 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Mitkin, Oleg D, Tkachenko, Sergey E, Kysil, Volodymyr M, Okun, Ilya

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Crystal structure, Hirshfeld analysis and a mol-ecular docking study of a new inhibitor of the Hepatitis B virus (HBV): ethyl 5-methyl-1,1-dioxo-2-{[5-(pentan-3-yl)-1,2,4-oxa-diazo... von Ivachtchenko, Alexandre V, Kovalenko, Sergiy M, Kravchenko, Dmitry V, Mitkin, Oleg D, Ivanov, Vladimir V, Langer, Thierry

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Synthesis, Single Crystal X-Ray Analysis, Prediction and Study of Pharmacological Activity of 4-(1H-Benzo[d]imidazol-2-yl)-1-Phenyl-1H-1,2,3-triazol-5-Amine and Its Solvates von Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Ivanov, Vladimir V., Konovalova, Olena D., Langer, Thierry

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