Discovery of GSK2795039, a Novel Small Molecule NADPH Oxidase 2 Inhibitor von Hirano, Kazufumi, Chen, Woei Shin, Chueng, Adeline L W, Dunne, Angela A, Seredenina, Tamara, Filippova, Aleksandra, Ramachandran, Sumitra, Bridges, Angela, Chaudry, Laiq, Pettman, Gary, Allan, Craig, Duncan, Sarah, Lee, Kiew Ching, Lim, Jean, Ma, May Thu, Ong, Agnes B, Ye, Nicole Y, Nasir, Shabina, Mulyanidewi, Sri, Aw, Chiu Cheong, Oon, Pamela P, Liao, Shihua, Li, Dizheng, Johns, Douglas G, Miller, Neil D, Davies, Ceri H, Browne, Edward R, Matsuoka, Yasuji, Chen, Deborah W, Jaquet, Vincent, Rutter, A Richard

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Synthesis and Pharmacological Evaluation of Dual Acting Ligands Targeting the Adenosine A2A and Dopamine D2 Receptors for the Potential Treatment of Parkinson’s Disease von Jörg, Manuela, May, Lauren T, Mak, Frankie S, Lee, Kiew Ching K, Miller, Neil D, Scammells, Peter J, Capuano, Ben

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Novel adenosine A2A receptor ligands: A synthetic, functional and computational investigation of selected literature adenosine A2A receptor antagonists for extending into extracell... von Jörg, Manuela, Shonberg, Jeremy, Mak, Frankie S., Miller, Neil D., Yuriev, Elizabeth, Scammells, Peter J., Capuano, Ben

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Novel adenosine A(2A) receptor ligands: a synthetic, functional and computational investigation of selected literature adenosine A(2A) receptor antagonists for extending into extra... von Jörg, Manuela, Shonberg, Jeremy, Mak, Frankie S, Miller, Neil D, Yuriev, Elizabeth, Scammells, Peter J, Capuano, Ben

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Procognitive 5-HT6 antagonists in the rat forced swimming test: potential therapeutic utility in mood disorders associated with Alzheimer's disease von Hirano, Kazufumi, Piers, Thomas M, Searle, Kirsten L, Miller, Neil D, Rutter, A Richard, Chapman, Paul F

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Intramolecular Palladium-Catalyzed Direct Arylation of Alkenyl Triflates von Cruz, Ana C. F, Miller, Neil D, Willis, Michael C

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A novel series of benzimidazole NR2B-selective NMDA receptor antagonists von Davies, David J., Crowe, Matthew, Lucas, Nolwenn, Quinn, Joanna, Miller, David D., Pritchard, Sara, Grose, David, Bettini, Ezio, Calcinaghi, Novella, Virginio, Caterina, Abberley, Lee, Goldsmith, Paul, Michel, Anton D., Chessell, Iain P., Kew, James N.C., Miller, Neil D., Gunthorpe, Martin J.

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2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: identification, stereochemistry and initial SAR von Wyatt, Paul G., Allen, Michael J., Borthwick, Alan D., Davies, Dave E., Exall, Anne M., Hatley, Richard J.D., Irving, Wendy R., Livermore, David G., Miller, Neil D., Nerozzi, Fabrizio, Sollis, Steve L., Szardenings, Anna Katrin

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P4-319: 5-HT6 receptor antagonists modulate brain monoaminergic neurotransmission: Different mode of action from acetylcholinesterase (AchE) inhibitors von Hirano, Kazufumi, Rutter, Richard A, Miller, Neil D, Chapman, Paul F

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Structure–activity relationship investigations of a potent and selective benzodiazepine oxytocin antagonist von Wyatt, Paul G, Allen, Michael J, Chilcott, Josie, Hickin, Gwen, Miller, Neil D, Woollard, Patrick M

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Development of a Co-Mediated Rearrangement Reaction von Carbery, David R., Reignier, Serge, Myatt, James W., Miller, Neil D., Harrity, Joseph P. A.

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Investigation of a Stereoselective Co-Mediated Rearrangement Reaction von Carbery, David R, Reignier, Serge, Miller, Neil D, Adams, Harry, Harrity, Joseph P. A

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A Novel Approach to the CP-225,917 and CP-263,114 Core von Nicolaou, K. C., Postema, Maarten H. D., Miller, Neil D., Yang, Guang

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Tandem cobalt mediated rearrangement and Pauson–Khand reaction for the synthesis of functionalised polycyclic systemsElectronic supplementary information (ESI) available: experimen... von Carbery, David R., Miller, Neil D., Harrity, Joseph P. A.

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Synthesis and Pharmacological Evaluation of Dual Acting Ligands Targeting the Adenosine A 2A and Dopamine D 2 Receptors for the Potential Treatment of Parkinson’s Disease von Jörg, Manuela, May, Lauren T., Mak, Frankie S., Lee, Kiew Ching K., Miller, Neil D., Scammells, Peter J., Capuano, Ben

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Synthesis, molecular structure, NMR spectroscopic and computational analysis of a selective adenosine A2A antagonist, ZM 241385 von Jörg, Manuela, Agostino, Mark, Yuriev, Elizabeth, Mak, Frankie S., Miller, Neil D., White, Jonathan M., Scammells, Peter J., Capuano, Ben

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The Synthesis of Proline Derived Homochiral Amine Oxides von O’Neil, Ian A., Miller, Neil D., Barkley, Jim V., Low, Caroline M. R., Kalindjian, S. Barret

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Post-Cataract Surgery Optic Neuropathy (PCSON): Prevalence, Incidence, Temporal Relationship and Fellow Eye Involvement von Moradi, Ahmadreza, MD, Kanagalingam, Sivashakthi, MD, Diener-West, Marie, PhD, Miller, Neil R., MD

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Investigation of novel ropinirole analogues: synthesis, pharmacological evaluation and computational analysis of dopamine D2 receptor functionalized congeners and homobivalent liga... von Jörg, Manuela, Kaczor, Agnieszka A, Mak, Frankie S, Lee, Kiew Ching K, Poso, Antti, Miller, Neil D, Scammells, Peter J, Capuano, Ben

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Investigation of novel ropinirole analogues: synthesis, pharmacological evaluation and computational analysis of dopamine D 2 receptor functionalized congeners and homobivalent lig... von Jörg, Manuela, Kaczor, Agnieszka A., Mak, Frankie S., Lee, Kiew Ching K., Poso, Antti, Miller, Neil D., Scammells, Peter J., Capuano, Ben

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