The hepatitis B virus ribonuclease H is sensitive to inhibitors of the human immunodeficiency virus ribonuclease H and integrase enzymes von Tavis, John E, Cheng, Xiaohong, Hu, Yuan, Totten, Michael, Cao, Feng, Michailidis, Eleftherios, Aurora, Rajeev, Meyers, Marvin J, Jacobsen, E Jon, Parniak, Michael A, Sarafianos, Stefan G

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Identification of potent and orally efficacious phosphodiesterase inhibitors in Cryptosporidium parvum-infected immunocompromised male mice von Ajiboye, Jubilee, Teixeira, José E., Gasonoo, Makafui, Mattice, Ethan B., Korwin-Mihavics, Bethany, Miller, Peter, Cameron, Alexandra C., Stebbins, Erin, Campbell, Scott D., Griggs, David W., Spangenberg, Thomas, Meyers, Marvin J., Huston, Christopher D.

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Clinical and microbiologic efficacy of the piperazine-based drug lead MMV665917 in the dairy calf cryptosporidiosis model von Stebbins, Erin, Jumani, Rajiv S, Klopfer, Connor, Barlow, John, Miller, Peter, Campbell, Mary A, Meyers, Marvin J, Griggs, David W, Huston, Christopher D

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Hydroxylated tropolones inhibit hepatitis B virus replication by blocking viral ribonuclease H activity von Lu, Gaofeng, Lomonosova, Elena, Cheng, Xiaohong, Moran, Eileen A, Meyers, Marvin J, Le Grice, Stuart F J, Thomas, Craig J, Jiang, Jian-kang, Meck, Christine, Hirsch, Danielle R, D'Erasmo, Michael P, Suyabatmaz, Duygu M, Murelli, Ryan P, Tavis, John E

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The therapeutic efficacy of azithromycin and nitazoxanide in the acute pig model of Cryptosporidium hominis von Lee, Sangun, Harwood, Melanie, Girouard, Don, Meyers, Marvin J, Campbell, Mary A, Beamer, Gillian, Tzipori, Saul

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Hepatitis B virus replication is blocked by a 2-hydroxyisoquinoline-1,3(2H,4H)-dione (HID) inhibitor of the viral ribonuclease H activity von Cai, Catherine W., Lomonosova, Elena, Moran, Eileen A., Cheng, Xiaohong, Patel, Kunjan B., Bailly, Fabrice, Cotelle, Philippe, Meyers, Marvin J., Tavis, John E.

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The anti-cancer efficacy of a novel phenothiazine derivative is independent of dopamine and serotonin receptor inhibition von Vanneste, Marion, Venzke, Anita, Guin, Soumitra, Fuller, Andrew J, Jezewski, Andrew J, Beattie, Sarah R, Krysan, Damian J, Meyers, Marvin J, Henry, Michael D

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Chemical Approaches to Inhibiting the Hepatitis B Virus Ribonuclease H von Tavis, John E, Zoidis, Grigoris, Meyers, Marvin J, Murelli, Ryan P

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Repurposing and optimization of drugs for discovery of novel antifungals von Donlin, Maureen J., Meyers, Marvin J.

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Pyrrolopyridine Inhibitors of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MK-2) von Anderson, David R, Meyers, Marvin J, Vernier, William F, Mahoney, Matthew W, Kurumbail, Ravi G, Caspers, Nicole, Poda, Gennadiy I, Schindler, John F, Reitz, David B, Mourey, Robert J

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Discovery of (3S,3aR)-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Recep... von Meyers, Marvin J, Arhancet, Graciela B, Hockerman, Susan L, Chen, Xiangyang, Long, Scott A, Mahoney, Matthew W, Rico, Joseph R, Garland, Danny J, Blinn, James. R, Collins, Joe T, Yang, Shengtian, Huang, Horng-Chih, McGee, Kevin F, Wendling, Jay M, Dietz, Jessica D, Payne, Maria A, Homer, Bruce L, Heron, Marcia I, Reitz, David B, Hu, Xiao

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Synthesis and Evaluation of Troponoids as a New Class of Antibiotics von Cao, Feng, Orth, Cari, Donlin, Maureen J, Adegboyega, Patrick, Meyers, Marvin J, Murelli, Ryan P, Elagawany, Mohamed, Elgendy, Bahaa, Tavis, John E

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Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism von Shiau, Andrew K., Barstad, Danielle, Radek, James T., Meyers, Marvin J., Nettles, Kendall W., Katzenellenbogen, Benita S., Katzenellenbogen, John A., Agard, David A., Greene, Geoffrey L.

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Rev-Erb co-regulates muscle regeneration via tethered interaction with the NF-Y cistrome von Welch, Ryan D, Guo, Chun, Sengupta, Monideepa, Carpenter, Katherine J, Stephens, Natalie A, Arnett, Stacy A, Meyers, Marvin J, Sparks, Lauren M, Smith, Steven R, Zhang, Jinsong, Burris, Thomas P, Flaveny, Colin A

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Mechanism of Action of N -Acyl and N -Alkoxy Fosmidomycin Analogs: Mono- and Bisubstrate Inhibition of IspC from Plasmodium falciparum , a Causative Agent of Malaria von Girma, Misgina B, Ball, Haley S, Wang, Xu, Brothers, Robert C, Jackson, Emily R, Meyers, Marvin J, Dowd, Cynthia S, Couch, Robin D

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Synthetic Derivatives of Ciclopirox are Effective Inhibitors of Cryptococcus neoformans von Lin, Jeffrey, Zangi, Maryam, Kumar, Tanguturi Venkata Narayana Hajay, Shakar Reddy, Makala, Reddy, Lingala Vijaya Raghava, Sadhukhan, Subir Kumar, Bradley, Daniel P, Moreira-Walsh, Brenda, Edwards, Tiffany C, O’Dea, Austin T, Tavis, John E, Meyers, Marvin J, Donlin, Maureen J

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Clinically Advanced p38 Inhibitors Suppress DUX4 Expression in Cellular and Animal Models of Facioscapulohumeral Muscular Dystrophy von Oliva, Jonathan, Galasinski, Scott, Richey, Amelia, Campbell, Amy E, Meyers, Marvin J, Modi, Neal, Zhong, Jun Wen, Tawil, Rabi, Tapscott, Stephen J, Sverdrup, Francis M

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Plasmepsins IX and X are essential and druggable mediators of malaria parasite egress and invasion von Nasamu, Armiyaw S., Glushakova, Svetlana, Russo, Ilaria, Vaupel, Barbara, Oksman, Anna, Kim, Arthur S., Fremont, Daved H., Tolia, Niraj, Beck, Josh R., Meyers, Marvin J., Niles, Jacquin C., Zimmerberg, Joshua, Goldberg, Daniel E.

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Efficient Inhibition of Hepatitis B Virus (HBV) Replication and cccDNA Formation by HBV Ribonuclease H Inhibitors during Infection von Chauhan, Ranjit, Li, Qilan, Woodson, Molly E, Gasonoo, Makafui, Meyers, Marvin J, Tavis, John E

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Identification of 4-Amino-Thieno[2,3- d ]Pyrimidines as QcrB Inhibitors in Mycobacterium tuberculosis von Harrison, Gregory A, Mayer Bridwell, Anne E, Singh, Megh, Jayaraman, Keshav, Weiss, Leslie A, Kinsella, Rachel L, Aneke, Janessa S, Flentie, Kelly, Schene, Miranda E, Gaggioli, Margaret, Solomon, Samantha D, Wildman, Scott A, Meyers, Marvin J, Stallings, Christina L

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