Discovery of SYD5115, a novel orally active small molecule TSH-R antagonist von Karstens, Willem F.J., M.B.P. Menge, Wiro, Martens, Gijs, op het Veld, Sanne J.N., Th.H. van Eupen, Jacobus, Demon, Marco, van Achterberg, Tanja A.E., Arisse-Thijssen, Monica J., Santegoeds-Lenssen, Ellen W.H., van der Lee, Miranda M.C., Ubink, Ruud, Arends, Roel J., Sesink, Aloys, Blomenröhr, Marion, Marco Timmers, C.

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Pharmacological characterization of the human histamine H2 receptor stably expressed in Chinese hamster ovary cells von Leurs, Rob, Smit, Martine J., Menge, Wiro M.B.P., Timmerman, Hendrik

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Clobenpropit analogs as dual activity ligands for the histamine H 3 and H 4 receptors: Synthesis, pharmacological evaluation, and cross-target QSAR studies von Lim, Herman D., Istyastono, Enade P., van de Stolpe, Andrea, Romeo, Giuseppe, Gobbi, Silvia, Schepers, Marjo, Lahaye, Roger, Menge, Wiro M.B.P., Zuiderveld, Obbe P., Jongejan, Aldo, Smits, Rogier A., Bakker, Remko A., Haaksma, Eric E.J., Leurs, Rob, de Esch, Iwan J.P.

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Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: Synthesis, pharmacological evaluation, and cross-target QSAR studies von LIM, Herman D, ISTYASTONO, Enade P, SMITS, Rogier A, BAKKER, Remko A, HAAKSMA, Eric E. J, LEURS, Rob, DE ESCH, Iwan J. P, VAN DE STOLPE, Andrea, ROMEO, Giuseppe, GOBBI, Silvia, SCHEPERS, Marjo, LAHAYE, Roger, MENGE, Wiro M. B. P, ZUIDERVELD, Obbe P, JONGEJAN, Aldo

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Synthesis and Pharmacological Identification of Neutral Histamine H 1 -Receptor Antagonists von Govoni, Marinella, Bakker, Remko A., van de Wetering, Ineke, Smit, Martine J., Menge, Wiro M. B. P., Timmerman, Henk, Elz, Sigurd, Schunack, Walter, Leurs, Rob

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Pharmacological characterization of the human histamine H 2 receptor stably expressed in Chinese hamster ovary cells von Leurs, Rob, Smit, Martine J., Menge, Wiro M.B.P., Timmerman, Hendrik

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Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5‐HT3 receptor revealed von Leurs, Rob, Tulp, Martin Th.M., Menge, Wiro M.B.P., Adolfs, Martin J.P., Zuiderveld, Obbe P., Timmerman, Hendrik

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Evaluation of the receptor selectivity of the H 3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5‐HT 3 receptor revealed von Leurs, Rob, Tulp, Martin Th.M., Menge, Wiro M.B.P., Adolfs, Martin J.P., Zuiderveld, Obbe P., Timmerman, Hendrik

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