Assessment of Mycobacterium tuberculosis Pantothenate Kinase Vulnerability through Target Knockdown and Mechanistically Diverse Inhibitors von KISHORE REDDY, B. K, LANDGE, Sudhir, AMBADY, Anisha, GHOSH, Anirban, TUNDUGURU, Ragadeepthi, KAUR, Parvinder, SINGH, Ragini, KUMAR, Naveen, BHARATH, Sowmya, SUNDARAM, Aishwarya, BHAT, Jyothi, SAMBANDAMURTHY, Vasan K, RAVISHANKAR, Sudha, BJÖRKELID, Christofer, ALWYN JONES, T, DAS, Kaveri, BANDODKAR, Balachandra, MALOLANARASIMHAN, Krishnan, MUKHERJEE, Kakoli, RAMACHANDRAN, Vasanthi, PATIL, Vikas, SHINDE, Vikas, TANTRY, Subramanyam, KALE, Manoj, RAICHURKAR, Anandkumar, MENASINAKAI, Sreenivasaiah, NAINA VINAY MUDUGAL

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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate von Hameed P., Shahul, Solapure, Suresh, Patil, Vikas, Henrich, Philipp P., Magistrado, Pamela A., Bharath, Sowmya, Murugan, Kannan, Viswanath, Pavithra, Puttur, Jayashree, Srivastava, Abhishek, Bellale, Eknath, Panduga, Vijender, Shanbag, Gajanan, Awasthy, Disha, Landge, Sudhir, Morayya, Sapna, Koushik, Krishna, Saralaya, Ramanatha, Raichurkar, Anandkumar, Rautela, Nikhil, Roy Choudhury, Nilanjana, Ambady, Anisha, Nandishaiah, Radha, Reddy, Jitendar, Prabhakar, K. R., Menasinakai, Sreenivasaiah, Rudrapatna, Suresh, Chatterji, Monalisa, Jiménez-Díaz, María Belén, Martínez, María Santos, Sanz, Laura María, Coburn-Flynn, Olivia, Fidock, David A., Lukens, Amanda K., Wirth, Dyann F., Bandodkar, Balachandra, Mukherjee, Kakoli, McLaughlin, Robert E., Waterson, David, Rosenbrier-Ribeiro, Lyn, Hickling, Kevin, Balasubramanian, V., Warner, Peter, Hosagrahara, Vinayak, Dudley, Adam, Iyer, Pravin S., Narayanan, Shridhar, Kavanagh, Stefan, Sambandamurthy, Vasan K.

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Novel N‑Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis von Hameed P, Shahul, Patil, Vikas, Solapure, Suresh, Sharma, Umender, Madhavapeddi, Prashanti, Raichurkar, Anandkumar, Chinnapattu, Murugan, Manjrekar, Praveena, Shanbhag, Gajanan, Puttur, Jayashree, Shinde, Vikas, Menasinakai, Sreenivasaiah, Rudrapatana, Suresh, Achar, Vijayashree, Awasthy, Disha, Nandishaiah, Radha, Humnabadkar, Vaishali, Ghosh, Anirban, Narayan, Chandan, Ramya, V. K, Kaur, Parvinder, Sharma, Sreevalli, Werngren, Jim, Hoffner, Sven, Panduga, Vijender, Kumar, C. N. Naveen, Reddy, Jitendar, Kumar KN, Mahesh, Ganguly, Samit, Bharath, Sowmya, Bheemarao, Ugarkar, Mukherjee, Kakoli, Arora, Uma, Gaonkar, Sheshagiri, Coulson, Michelle, Waterson, David, Sambandamurthy, Vasan K, de Sousa, Sunita M

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Genetic and chemical validation identifies Mycobacterium tuberculosis topoisomerase I as an attractive anti-tubercular target von Ravishankar, Sudha, Ambady, Anisha, Awasthy, Disha, Mudugal, Naina Vinay, Menasinakai, Sreenivasaiah, Jatheendranath, Sandesh, Guptha, Supreeth, Sharma, Sreevalli, Balakrishnan, Gayathri, Nandishaiah, Radha, Ramachandran, Vasanthi, Eyermann, Charles J, Reck, Folkert, Rudrapatna, Suresh, Sambandamurthy, Vasan K, Sharma, Umender K

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Benzimidazoles: Novel Mycobacterial Gyrase Inhibitors from Scaffold Morphing von Hameed P, Shahul, Raichurkar, Anandkumar, Madhavapeddi, Prashanti, Menasinakai, Sreenivasaiah, Sharma, Sreevalli, Kaur, Parvinder, Nandishaiah, Radha, Panduga, Vijender, Reddy, Jitendar, Sambandamurthy, Vasan K, Sriram, D

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Whole cell screen based identification of spiropiperidines with potent antitubercular properties von Tantry, Subramanyam J., Degiacomi, Giulia, Sharma, Sreevalli, Jena, Lalit kumar, Narayan, Ashwini, Guptha, Supreeth, Shanbhag, Gajanan, Menasinakai, Sreenivasaiah, Mallya, Meenakshi, Awasthy, Disha, Balakrishnan, Gayathri, Kaur, Parvinder, Bhattacharjee, Deepa, Narayan, Chandan, Reddy, Jitendar, Naveen Kumar, C.N., Shandil, Radha, Boldrin, Francesca, Ventura, Marcello, Manganelli, Riccardo, Hartkoorn, Ruben C., Cole, Stewart T., Panda, Manoranjan, Markad, Shankar D., Ramachandran, Vasanthi, Ghorpade, Sandeep R., Dinesh, Neela

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N‑Aryl-2-aminobenzimidazoles: Novel, Efficacious, Antimalarial Lead Compounds von Ramachandran, Sreekanth, Hameed P, Shahul, Srivastava, Abhishek, Shanbhag, Gajanan, Morayya, Sapna, Rautela, Nikhil, Awasthy, Disha, Kavanagh, Stefan, Bharath, Sowmya, Reddy, Jitendar, Panduga, Vijender, Prabhakar, K. R, Saralaya, Ramanatha, Nanduri, Robert, Raichurkar, Anandkumar, Menasinakai, Sreenivasaiah, Achar, Vijayashree, Jiménez-Díaz, María Belén, Martínez, María Santos, Angulo-Barturen, Iñigo, Ferrer, Santiago, Sanz, Laura María, Gamo, Francisco Javier, Duffy, Sandra, Avery, Vicky M, Waterson, David, Lee, Marcus C. S, Coburn-Flynn, Olivia, Fidock, David A, Iyer, Pravin S, Narayanan, Shridhar, Hosagrahara, Vinayak, Sambandamurthy, Vasan K

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Thiazolopyridone ureas as DNA gyrase B inhibitors: Optimization of antitubercular activity and efficacy von Kale, Ramesh R., Kale, Manoj G., Waterson, David, Raichurkar, Anandkumar, Hameed, Shahul P., Manjunatha, M.R., Kishore Reddy, B.K., Malolanarasimhan, Krishnan, Shinde, Vikas, Koushik, Krishna, Jena, Lalit Kumar, Menasinakai, Sreenivasaiah, Humnabadkar, Vaishali, Madhavapeddi, Prashanti, Basavarajappa, Halesha, Sharma, Sreevalli, Nandishaiah, Radha, Mahesh Kumar, K.N., Ganguly, Samit, Ahuja, Vijaykamal, Gaonkar, Sheshagiri, Naveen Kumar, C.N., Ogg, Derek, Boriack-Sjodin, P. Ann, Sambandamurthy, Vasan K., de Sousa, Sunita M., Ghorpade, Sandeep R.

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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate von Hameed P., Shahul, Solapure, Suresh, Patil, Vikas, Henrich, Philipp P, Magistrado, Pamela A, Bharath, Sowmya, Murugan, Kannan, Viswanath, Pavithra, Puttur, Jayashree, Srivastava, Abhishek, Bellale, Eknath, Panduga, Vijender, Shanbag, Gajanan, Awasthy, Disha, Landge, Sudhir, Morayya, Sapna, Koushik, Krishna, Saralaya, Ramanatha, Raichurkar, Anandkumar, Rautela, Nikhil, Roy Choudhury, Nilanjana, Ambady, Anisha, Nandishaiah, Radha, Reddy, Jitendar, Prabhakar, K. R, Menasinakai, Sreenivasaiah, Rudrapatna, Suresh, Chatterji, Monalisa, Jiménez-Díaz, María Belén, Martínez, María Santos, Sanz, Laura María, Coburn-Flynn, Olivia, Fidock, David A, Lukens, Amanda K, Wirth, Dyann F, Bandodkar, Balachandra, Mukherjee, Kakoli, McLaughlin, Robert E, Waterson, David, Rosenbrier-Ribeiro, Lyn, Hickling, Kevin, Balasubramanian, V, Warner, Peter, Hosagrahara, Vinayak, Dudley, Adam, Iyer, Pravin S, Narayanan, Shridhar, Kavanagh, Stefan, Sambandamurthy, Vasan K

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