mGluR5 metabotropic glutamate receptors and dyskinesias in MPTP monkeys von Samadi, Pershia, Grégoire, Laurent, Morissette, Marc, Calon, Fréderic, Hadj Tahar, Abdallah, Dridi, Mehdi, Belanger, Nancy, Meltzer, Leonard T, Bédard, Paul J, Di Paolo, Thérèse

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Normalization of GABAA receptor specific binding in the substantia nigra reticulata and the prevention of L-dopa-induced dyskinesias in MPTP parkinsonian monkeys von Samadi, Pershia, Morissette, Marc, Calon, Fréderic, Tahar, Abdallah Hadj, Dridi, Mehdi, Belanger, Nancy, Meltzer, Leonard T., Bédard, Paul J., Di Paolo, Thérèse

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Structure−Activity Relationships of Pregabalin and Analogues That Target the α2-δ Protein von Belliotti, Thomas R, Capiris, Thomas, Ekhato, I. Victor, Kinsora, Jack J, Field, Mark J, Heffner, Thomas G, Meltzer, Leonard T, Schwarz, Jacob B, Taylor, Charles P, Thorpe, Andrew J, Vartanian, Mark G, Wise, Lawrence D, Zhi-Su, Ti, Weber, Mark L, Wustrow, David J

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Implication of NMDA Receptors in the Antidyskinetic Activity of Cabergoline, CI-1041, and Ro 61-8048 in MPTP Monkeys with Levodopa-induced Dyskinesias von Ouattara, Bazoumana, Belkhir, Samah, Morissette, Marc, Dridi, Mehdi, Samadi, Pershia, Grégoire, Laurent, Meltzer, Leonard T., Di Paolo, Thérèse

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Subtype-Selective N-Methyl-d-aspartate Receptor Antagonists:  Benzimidazalone and Hydantoin as Phenol Replacements von Schelkun, Robert M, Yuen, Po-wai, Serpa, Kevin, Meltzer, Leonard T, Wise, Lawrence D, Whittemore, Edward R, Woodward, Richard M

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Asenapine effects in animal models of psychosis and cognitive function von Marston, Hugh M., Young, Jared W., Martin, Frederic D. C., Serpa, Kevin A., Moore, Christopher L., Wong, Erik H. F., Gold, Lisa, Meltzer, Leonard T., Azar, Marc R., Geyer, Mark A., Shahid, Mohammed

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Prevention of levodopa-induced dyskinesias by a selective NR1A/2B N-methyl-D-aspartate receptor antagonist in parkinsonian monkeys: Implication of preproenkephalin von Morissette, Marc, Dridi, Mehdi, Calon, Frédéric, Tahar, Abdallah Hadj, Meltzer, Leonard T., Bédard, Paul J., Di Paolo, Thérèse

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APN1125: A NOVEL A7 NICOTINIC ACETYLCHOLINE RECEPTOR PARTIAL AGONIST von Koelsch, Gerald, Meltzer, Leonard T, Yoshimura, Ryan F, Terry, Alvin V, Callahan, Patrick M, Bilcer, Geoffrey, Ng, John, Ng, Raymond, Gee, Kelvin W, Kelly, Terence A

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Prevention of dyskinesia by an NMDA receptor antagonist in MPTP monkeys: Effect on adenosine A2A receptors von Morissette, Marc, Dridi, Mehdi, Calon, Frédéric, Tahar, Abdallah Hadj, Meltzer, Leonard T., Bédard, Paul J., Di Paolo, Thérèse

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Synthesis and SAR of tolylamine 5-HT6 antagonists von SINGER, Jamie M, WILSON, Michael W, ROUSH, Nicole, CAMPBELL, Jeffrey E, SU, Ti-Zhi, HURST, Susan I, STONER, Chad L, SCHWARZ, Jacob B, JOHNSON, Paul D, GRAHAM, Shelley R, COOKE, Leonard W, ROOF, Robin L, BOXER, Peter A, GOLD, Lisa H, MELTZER, Leonard T, JANSSEN, Ann

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Synthesis and Pharmacological Evaluation of Thiopyran Analogues of the Dopamine D3 Receptor-Selective Agonist (4aR,10bR)-(+)-trans-3,4,4a,10b- Tetrahydro-4-n-propyl-2H,5H-[1]benzop... von van Vliet, L. Alexander, Rodenhuis, Nienke, Dijkstra, Durk, Wikström, Håkan, Pugsley, Thomas A, Serpa, Kevin A, Meltzer, Leonard T, Heffner, Thomas G, Wise, Lawrence D, Lajiness, Mary E, Huff, Rita M, Svensson, Kjell, Sundell, Staffan, Lundmark, Max

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Subtype-Selective N-Methyl-d-Aspartate Receptor Antagonists:  Synthesis and Biological Evaluation of 1-(Heteroarylalkynyl)-4-benzylpiperidines von Wright, Jon L, Gregory, Tracy F, Kesten, Suzanne R, Boxer, Peter A, Serpa, Kevin A, Meltzer, Leonard T, Wise, Lawrence D, Espitia, Stephen A, Konkoy, Christopher S, Whittemore, Edward R, Woodward, Richard M

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Synthesis and in vivo evaluation of 3,4-disubstituted gababutins von Blakemore, David C., Bryans, Justin S., Carnell, Pauline, Field, Mark J., Kinsella, Natasha, Kinsora, Jack K., Meltzer, Leonard T., Osborne, Simon A., Thompson, Lisa R., Williams, Sophie C.

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Synthesis and dopamine agonist properties of (+)-trans-3,4,4a,10b-tetrahydro-4-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol and its enantiomers von DeWald, Horace A, Heffner, Thomas G, Jaen, Juan C, Lustgarten, David M, McPhail, Andrew T, Meltzer, Leonard T, Pugsley, Thomas A, Wise, Lawrence D

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4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties von Jaen, Juan C, Wise, Lawrence D, Caprathe, Bradley W, Tecle, Haile, Bergmeier, Stephen, Humblet, Christine C, Heffner, Thomas G, Meltzer, Leonard T, Pugsley, Thomas A

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Orally Active Analogues of the Dopaminergic Prodrug 6-(N,N-Di-n-propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one:  Synthesis and Pharmacological Activity von Venhuis, Bastiaan J, Dijkstra, Durk, Wustrow, David J, Meltzer, Leonard T, Wise, Lawrence D, Johnson, Stephen J, Heffner, Thomas G, Wikström, Håkan V

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Subtype selective NMDA receptor antagonists: evaluation of some novel alkynyl analogues von KORNBERG, Brian E, NIKAM, Sham S, WRIGHT, Jon L, KESTEN, Suzanne R, MELTZER, Leonard T, COUGHENOUR, Linda, BARR, Bridget, SERPA, Kevin A, MCCORMICK, Julie

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Reversal of Haloperidol-Induced Extrapyramidal Side Effects in Cebus Monkeys by 8-Hydroxy-2-(di-n-propylamino)tetralin and Its Enantiomers von Christoffersen, B.A, Curt L, Meltzer, Ph.D, Leonard T

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Thiazoloindans and Thiazolobenzopyrans:  A Novel Class of Orally Active Central Dopamine (Partial) Agonists von van Vliet, L. Alexander, Rodenhuis, Nienke, Wikström, Håkan, Pugsley, Thomas A, Serpa, Kevin A, Meltzer, Leonard T, Heffner, Thomas G, Wise, Lawrence D, Lajiness, Mary E, Huff, Rita M, Svensson, Kjell, Haenen, Guido R. M. M, Bast, Aalt

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Structure-activity relationships of pregabalin and analogues that target the alpha(2)-delta protein von Belliotti, Thomas R, Capiris, Thomas, Ekhato, I Victor, Kinsora, Jack J, Field, Mark J, Heffner, Thomas G, Meltzer, Leonard T, Schwarz, Jacob B, Taylor, Charles P, Thorpe, Andrew J, Vartanian, Mark G, Wise, Lawrence D, Zhi-Su, Ti, Weber, Mark L, Wustrow, David J

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