Fluorinated Cycloalkyl Building Blocks for Drug Discovery von Grygorenko, Oleksandr O., Melnykov, Kostiantyn P., Holovach, Serhii, Demchuk, Oleksandr

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Parallel Minisci Reaction of gem-Difluorocycloalkyl Building Blocks von Holovach, Serhii, Poroshyn, Illia, Melnykov, Kostiantyn P., Liashuk, Oleksandr S., Pariiska, Olena O., Kolotilov, Sergey V., Rozhenko, Alexander B., Volochnyuk, Dmytro M., Grygorenko, Oleksandr O.

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Scalable Synthesis of Biologically Relevant Spirocyclic Pyrrolidines von Melnykov, Kostiantyn P, Artemenko, Artem N, Ivanenko, Bohdan O, Sokolenko, Yevhenii M, Nosik, Pavel S, Ostapchuk, Eugeniy N, Grygorenko, Oleksandr O, Volochnyuk, Dmitriy M, Ryabukhin, Sergey V

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Effect of gem‐Difluorination on the Key Physicochemical Properties Relevant to Medicinal Chemistry: The Case of Functionalized Cycloalkanes von Holovach, Sergey, Melnykov, Kostiantyn P., Skreminskiy, Artem, Herasymchuk, Maksym, Tavlui, Olha, Aloshyn, Danylo, Borysko, Petro, Rozhenko, Alexander B., Ryabukhin, Sergey V., Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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Impact of Fluoroalkyl Substituents on the Physicochemical Properties of Saturated Heterocyclic Amines von Melnykov, Kostiantyn P., Tavlui, Olha, Skreminskiy, Artem, Kuchkovska, Yuliya O., Grygorenko, Oleksandr O.

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Stellane at the Forefront: Derivatization and Reactivity Studies of a Promising Saturated Bioisostere of ortho-Substituted Benzenes von Smyrnov, Oleh K., Melnykov, Kostiantyn P., Pashenko, Olexandr Ye, Volochnyuk, Dmytro M., Ryabukhin, Serhiy V.

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α‐CF3‐Substituted Saturated Bicyclic Amines: Advanced Building Blocks for Medicinal Chemistry von Smyrnov, Oleh, Melnykov, Kostiantyn P., Semeno, Volodymyr, Liashuk, Oleksandr S., Grygorenko, Oleksandr O.

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Mono‐ and Difluorinated Saturated Heterocyclic Amines for Drug Discovery: Systematic Study of Their Physicochemical Properties von Melnykov, Kostiantyn P., Nazar, Kostiantyn, Smyrnov, Oleh, Skreminskyi, Artem, Pavlenko, Serhii, Klymenko‐Ulianov, Oleksii, Shishkina, Svitlana, Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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C−C Coupling through Nitrogen Deletion: Application to Library Synthesis von Holovach, Serhii, Melnykov, Kostiantyn P., Poroshyn, Illia, Iminov, Rustam T., Dudenko, Dmytro, Kondratov, Ivan, Levin, Mark, Grygorenko, Oleksandr O.

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C−C Coupling through Nitrogen Deletion: Application to Library Synthesis von Holovach, Serhii, Melnykov, Kostiantyn P., Poroshyn, Illia, Iminov, Rustam T., Dudenko, Dmytro, Kondratov, Ivan, Levin, Mark, Grygorenko, Oleksandr O.

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Bicyclo[m.n.k]alkane Building Blocks as Promising Benzene and Cycloalkane Isosteres: Multigram Synthesis, Physicochemical and Structural Characterization von Semeno, Volodymyr V., Vasylchenko, Vadym O., Fesun, Ihor M., Ruzhylo, Liudmyla Yu, Kipriianov, Mykhailo O., Melnykov, Kostiantyn P., Skreminskyi, Artem, Iminov, Rustam, Mykhailiuk, Pavel, Vashchenko, Bohdan V., Grygorenko, Oleksandr O.

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3,3-Difluorooxetane - A Versatile Functional Group for Bioisosteric Replacements in Drug Discovery von Liashuk, Oleksandr S, Fedinchyk, Anastasiya, Melnykov, Kostiantyn P, Herasymchuk, Maksym, Alieksieieva, Diana, Lesyk, Dmytro, Bas, Yuliia P, Keda, Tetiana Ye, Yatsymyrskiy, Andriy V, Holota, Yuliia, Borysko, Petro, Yarmolchuk, Volodymyr S, Grygorenko, Oleksandr O

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Multigram Synthesis of Dimethyl Stellane‐1,5‐Dicarboxylate as a Key Precursor for ortho‐Benzene Mimics von Smyrnov, Oleh K., Melnykov, Kostiantyn P., Rusanov, Eduard B., Suikov, Sergey Yu, Pashenko, Olexandr E., Fokin, Andrey A., Volochnyuk, Dmytro M., Ryabukhin, Serhiy V.

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Last of the gem-Difluorocycloalkanes: Synthesis and Characterization of 2,2-Difluorocyclobutyl-Substituted Building Blocks von Chernykh, Anton V, Melnykov, Kostiantyn P, Tolmacheva, Nataliya A, Kondratov, Ivan S, Radchenko, Dmytro S, Daniliuc, Constantin G, Volochnyuk, Dmitriy M, Ryabukhin, Sergey V, Kuchkovska, Yuliya O, Grygorenko, Oleksandr O

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Cover Feature: Multigram Synthesis of Dimethyl Stellane‐1,5‐Dicarboxylate as a Key Precursor for ortho‐Benzene Mimics (Chem. Eur. J. 70/2023) von Smyrnov, Oleh K., Melnykov, Kostiantyn P., Rusanov, Eduard B., Suikov, Sergey Yu, Pashenko, Olexandr E., Fokin, Andrey A., Volochnyuk, Dmytro M., Ryabukhin, Serhiy V.

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Fluorine‐Containing sp3‐Enriched Building Blocks for the Multigram Synthesis of Fluorinated Pyrazoles and Pyrimidines with (Hetero)aliphatic Substituents von Fedinchyk, Anastasiya, Herasymchuk, Maksym, Smirnov, Vladyslav O., Melnykov, Kostiantyn P., Yarmoliuk, Dmytro V., Kyrylchuk, Andrii A., Grygorenko, Oleksandr O.

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Last of the gem‐Difluorocycloalkanes 2: Synthesis of Fluorinated Cycloheptane Building Blocks von Herasymchuk, Maksym, Melnykov, Kostiantyn P., Yarmoliuk, Dmytro V., Serhiichuk, Dmytro, Rotar, Valeriia, Pukhovoi, Timur, Kuchkovska, Yuliya O., Holovach, Sergey, Volochnyuk, Dmitriy M., Ryabukhin, Sergey V., Grygorenko, Oleksandr O.

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Fluoroalkyl‐Containing 1,2‐Disubstituted Cyclobutanes: Advanced Building Blocks for Medicinal Chemistry von Demchuk, Oleksandr P., Hryshchuk, Oleksandr V., Vashchenko, Bohdan V., Trofymchuk, Serhii A., Melnykov, Kostiantyn P., Skreminskiy, Artem, Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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N‐Difluorocyclopropyl‐Substituted Pyrazoles: Synthesis and Reactivity von Nosik, Pavel S., Poturai, Andrii S., Pashko, Mykola O., Melnykov, Kostiantyn P., Ryabukhin, Sergey V., Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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A conformationally restricted GABA analogue based on octahydro-1H-cyclopenta[b]pyridine scaffold von Melnykov, Kostiantyn P., Volochnyuk, Dmitriy M., Ryabukhin, Sergey V., Rusanov, Eduard B., Grygorenko, Oleksandr O.

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