MRK-409 (MK-0343), a GABAA receptor subtype-selective partial agonist, is a non-sedating anxiolytic in preclinical species but causes sedation in humans von Atack, JR, Wafford, KA, Street, LJ, Dawson, GR, Tye, S, Van Laere, K, Bormans, G, Sanabria-Bohórquez, SM, De Lepeleire, I, de Hoon, JN, Van Hecken, A, Burns, HD, McKernan, RM, Murphy, MG, Hargreaves, RJ

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Preclinical and clinical pharmacology of TPA023B, a GABAA receptor α2/α3 subtype-selective partial agonist von Atack, JR, Hallett, DJ, Tye, S, Wafford, KA, Ryan, C, Sanabria-Bohórquez, SM, Eng, Wai-si, Gibson, RE, Burns, HD, Dawson, GR, Carling, RW, Street, LJ, Pike, A, De Lepeleire, I, Van Laere, K, Bormans, G, de Hoon, JN, Van Hecken, A, McKernan, RM, Murphy, MG, Hargreaves, RJ

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Characterization of [ 35 S] t ‐butylbicyclophosphorothionate ([ 35 S]TBPS) binding to GABA A receptors in postmortem human brain von Atack, J R, Ohashi, Y, McKernan, R M

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θ , a Novel γ -Aminobutyric Acid Type A Receptor Subunit von Bonnert, Timothy P., McKernan, Ruth M., Farrar, Sophie, le Bourdellès, Béatrice, Heavens, Robert P., Smith, David W., Hewson, Louise, Rigby, Michael R., Dalip J. S. Sirinathsinghji, Brown, Nicola, Wafford, Keith A., Whiting, Paul J.

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Age-related changes in GABA A receptor subunit composition and function in rat auditory system von Caspary, D.M, Holder, T.M, Hughes, L.F, Milbrandt, J.C, McKernan, R.M, Naritoku, D.K

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Stoichiometry of a Ligand-gated Ion Channel Determined by Fluorescence Energy Transfer von Farrar, S J, Whiting, P J, Bonnert, T P, McKernan, R M

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Gamma-aminobutyric acid type B receptors with specific heterodimer composition and postsynaptic actions in hippocampal neurons are targets of anticonvulsant gabapentin action von Ng, G Y, Bertrand, S, Sullivan, R, Ethier, N, Wang, J, Yergey, J, Belley, M, Trimble, L, Bateman, K, Alder, L, Smith, A, McKernan, R, Metters, K, O'Neill, G P, Lacaille, J C, Hébert, T E

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Loss of the major GABA(A) receptor subtype in the brain is not lethal in mice von Sur, C, Wafford, K A, Reynolds, D S, Hadingham, K L, Bromidge, F, Macaulay, A, Collinson, N, O'Meara, G, Howell, O, Newman, R, Myers, J, Atack, J R, Dawson, G R, McKernan, R M, Whiting, P J, Rosahl, T W

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Which GABA A-receptor subtypes really occur in the brain? von McKernan, Ruth M., Whiting, Paul J.

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Model of subunit composition of gamma-aminobutyric acid A receptor subtypes expressed in rat cerebellum with respect to their alpha and gamma/delta subunits von QUIRK, K, GILLARD, N. P, RAGAN, C. I, WHITING, P. J, MCKERNAN, R. M

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Retinoic Acid-Evoked Differentiation of Neuroblastoma Cells Predominates over Growth Factor Stimulation: An Automated Image Capture and Quantitation Approach to Neuritogenesis von Simpson, Peter B., Bacha, Jamil I., Palfreyman, Emma L., Woollacott, Anthony J., McKernan, Ruth M., Kerby, Julie

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Localization of 5-HT3 receptors in the rat spinal cord: immunohistochemistry and in situ hybridization von Kia, Hossein K, Miquel, Marie-Christine, McKernan, Ruth M, Laporte, Anne-Marie, Lombard, Marie-Christine, Bourgoin, Sylvie, Hamon, Michel, Vergé, Daniel

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Biology and migration of Eared Grebes at the Salton Sea von JEHL, Joseph R, MCKERNAN, Robert L

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CSF neuron-specific enolase as a quantitative marker of neuronal damage in a rat stroke model von Hatfield, Richard H., McKernan, Ruth M.

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Anxiolytic-like action of diazepam: which GABA A receptor subtype is involved? von Reynolds, David S., McKernan, Ruth M., Dawson, Gerard R.

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Generation and Characterisation of Stable Cell Lines Expressing Recombinant Human N‐Methyl‐d‐Aspartate Receptor Subtypes von Grimwood, Sarah, Le Bourdellès, Béatrice, Atack, John R., Barton, Cheryl, Cockett, Wendy, Cook, Susan M., Gilbert, Elizabeth, Hutson, Peter H., McKernan, Ruth M., Myers, Jan, Ragan, C. Ian, Wingrove, Peter B., Whiting, Paul J.

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Anxiogenic properties of an inverse agonist selective for α 3 subunit‐containing GABA A receptors von Atack, John R, Hutson, Peter H, Collinson, Neil, Marshall, George, Bentley, Graham, Moyes, Christopher, Cook, Susan M, Collins, Ian, Wafford, Keith, McKernan, Ruth M, Dawson, Gerard R

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Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach von Huang, Q, He, X, Ma, C, Liu, R, Yu, S, Dayer, C A, Wenger, G R, McKernan, R, Cook, J M

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Differential expression of GABAA receptor α-subunits in rat brain during development von McKernan, R.M., Cox, P., Gillard, N.P., Whiting, P.

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Association of Within-Territory Vegetation Characteristics and Fitness Components of California Gnatcatchers von Braden, Gerald T., McKernan, Robert L., Powell, Shawn M.

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