Blockade of mGluR1 receptor results in analgesia and disruption of motor and cognitive performances: effects of A‐841720, a novel non‐competitive mGluR1 receptor antagonist von El‐Kouhen, O, Lehto, S G, Pan, J B, Chang, R, Baker, S J, Zhong, C, Hollingsworth, P R, Mikusa, J P, Cronin, E A, Chu, K L, McGaraughty, S P, Uchic, M E, Miller, L N, Rodell, N M, Patel, M, Bhatia, P, Mezler, M, Kolasa, T, Zheng, G Z, Fox, G B, Stewart, A O, Decker, M W, Moreland, R B, Brioni, J D, Honore, P

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Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists von Gomtsyan, Arthur, Schmidt, Robert G, Bayburt, Erol K, Gfesser, Gregory A, Voight, Eric A, Daanen, Jerome F, Schmidt, Diana L, Cowart, Marlon D, Liu, Huaqing, Altenbach, Robert J, Kort, Michael E, Clapham, Bruce, Cox, Phil B, Shrestha, Anurupa, Henry, Rodger, Whittern, David N, Reilly, Regina M, Puttfarcken, Pamela S, Brederson, Jill-Desiree, Song, Ping, Li, Bin, Huang, Susan M, McDonald, Heath A, Neelands, Torben R, McGaraughty, Steve P, Gauvin, Donna M, Joshi, Shailen K, Banfor, Patricia N, Segreti, Jason A, Shebley, Mohamad, Faltynek, Connie R, Dart, Michael J, Kym, Philip R

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Blockade of mGluRI receptor results in analgesia and disruption of motor and cognitive performances: effects of A-841720, a novel non-competitive mGluR1 receptor antagonist von El-Kouhen, O, Lehto, S G, Pan, J B, Chang, R, Baker, S J, Zhong, C, Hollingsworth, PR, Mikusa, J P, Cronin, E A, Chu, K L, McGaraughty, S P, Uchic, ME, Miller, L N, Honore, P

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Chronic Pelvic Pain: Assessment, Evaluation, and Objectivation von Passavanti, Maria Beatrice, Pota, Vincenzo, Sansone, Pasquale, Aurilio, Caterina, De Nardis, Lorenzo, Pace, Maria Caterina

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Vulnerability and Resilience in Patients with Chronic Pain in Occupational Healthcare: A Pilot Study with a Patient-Centered Approach von Peilot, Birgitta, Andréll, Paulin, Gottfries, Johan, Sundler, Annelie J., Mannheimer, Clas

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Selective blockade of TRPA1 channel attenuates pathological pain without altering noxious cold sensation or body temperature regulation von Chen, Jun, Joshi, Shailen K., DiDomenico, Stanley, Perner, Richard J., Mikusa, Joe P., Gauvin, Donna M., Segreti, Jason A., Han, Ping, Zhang, Xu-Feng, Niforatos, Wende, Bianchi, Bruce R., Baker, Scott J., Zhong, Chengmin, Simler, Gricelda H., McDonald, Heath A., Schmidt, Robert G., McGaraughty, Steve P., Chu, Katharine L., Faltynek, Connie R., Kort, Michael E., Reilly, Regina M., Kym, Philip R.

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IL-23 induces regulatory T cell plasticity with implications for inflammatory skin diseases von Kannan, Arun K., Su, Zhi, Gauvin, Donna M., Paulsboe, Stephanie E., Duggan, Ryan, Lasko, Loren M., Honore, Prisca, Kort, Michael E., McGaraughty, Steve P., Scott, Victoria E., Gauld, Stephen B.

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Pharmacologic characterization of atogepant: A potent and selective calcitonin gene–related peptide receptor antagonist von Moore, Eric, Bell, Ian M, Fraley, Mark E, Burgey, Christopher S, White, Rebecca B, Li, Chi-Chung, Regan, Christopher P, Danziger, Andrew, McGaraughty, Steve P, Naseri Kouzehgarani, Ghazal, Salvatore, Christopher, Banerjee, Pradeep

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Oral and cutaneous thermosensory profile of selective TRPV1 inhibition by ABT-102 in a randomized healthy volunteer trial von Rowbotham, Michael C., Nothaft, Wolfram, Duan, W. Rachel, Wang, Yi, Faltynek, Connie, McGaraughty, Steve, Chu, Katharine L., Svensson, Peter

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Small Molecule IL-36γ Antagonist as a Novel Therapeutic Approach for Plaque Psoriasis von Todorović, Viktor, Su, Zhi, Putman, C. Brent, Kakavas, Stevan J., Salte, Katherine M., McDonald, Heath A., Wetter, Joseph B., Paulsboe, Stephanie E., Sun, Qi, Gerstein, Clare E., Medina, Limary, Sielaff, Bernhard, Sadhukhan, Ramkrishna, Stockmann, Henning, Richardson, Paul L., Qiu, Wei, Argiriadi, Maria A., Henry, Rodger F., Herold, J. Martin, Shotwell, J. Brad, McGaraughty, Steve P., Honore, Prisca, Gopalakrishnan, Sujatha M., Sun, Chaohong C., Scott, Victoria E.

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A-803467, a potent and selective Nav1.8 sodium channel blocker, attenuates neuropathic and inflammatory pain in the rat von Jarvis, Michael F, Honore, Prisca, Shieh, Char-Chang, Chapman, Mark, Joshi, Shailen, Zhang, Xu-Feng, Kort, Michael, Carroll, William, Marron, Brian, Atkinson, Robert, Thomas, James, Liu, Dong, Krambis, Michael, Liu, Yi, McGaraughty, Steve, Chu, Katharine, Roeloffs, Rosemarie, Zhong, Chengmin, Mikusa, Joseph P, Hernandez, Gricelda, Gauvin, Donna, Wade, Carrie, Zhu, Chang, Pai, Madhavi, Scanio, Marc, Shi, Lei, Drizin, Irene, Gregg, Robert, Matulenko, Mark, Hakeem, Ahmed, Gross, Michael, Johnson, Matthew, Marsh, Kennan, Wagoner, P. Kay, Sullivan, James P, Faltynek, Connie R, Krafte, Douglas S

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Inhibition of Interleukin-23–Mediated Inflammation with a Novel Small Molecule Inverse Agonist of RORγt von Gauld, Stephen B., Jacquet, Sebastien, Gauvin, Donna, Wallace, Craig, Wang, Yibing, McCarthy, Richard, Goess, Christian, Leys, Laura, Huang, Susan, Su, Zhi, Edelmayer, Rebecca, Wetter, Joseph, Salte, Katherine, McGaraughty, Steven P., Argiriadi, Maria A., Honore, Prisca, Luccarini, Jean-Michel, Bressac, Didier, Desino, Kelly, Breinlinger, Eric, Cusack, Kevin, Potin, Dominique, Kort, Michael E., Masson, Philippe J

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716 TSLP induced atopic dermatitis-like skin inflammation in mice von Paulsboe, S.E., Su, Z., Salte, K., Wetter, J., Honore, P., McGaraughty, S.

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474 IL-25 induces skin inflammation in mice: Effects of a selective JAK inhibitor von Su, Z., McDonald, H., Todorovic, V., Wetter, J., Paulsboe, S., Chu, K., Leys, L., Namovic, M., Donnelly-Roberts, D., Scott, V., Honore, P., McGaraughty, S.

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P2X7 -related modulation of pathological nociception in rats von McGaraughty, S, Chu, K.L, Namovic, M.T, Donnelly-Roberts, D.L, Harris, R.R, Zhang, X.-F, Shieh, C.-C, Wismer, C.T, Zhu, C.Z, Gauvin, D.M, Fabiyi, A.C, Honore, P, Gregg, R.J, Kort, M.E, Nelson, D.W, Carroll, W.A, Marsh, K, Faltynek, C.R, Jarvis, M.F

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A-306989, an inhibitor of adenosine kinase, is renoprotective in rodent models of podocyte, basement membrane, and obstructive injury von Zhu, Chang Z., Gopalakrishnan, Sujatha, Doyle, Kelly, Nikkel, Arthur L., Olson, Lauren, Abraham, Vivek C., Leys, Laura, Widomski, Deborah, Salte, Katherine, Putman, Brent, Pratt, Steve, Ma, Ji, Su, Zhi, Gopalakrishnan, Murali, Lee, Chih-Hung, McGaraughty, Steve P.

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Sedation and Analgesia in Intensive Care: A Comparison of Fentanyl and Remifentanil von Cevik, F., Celik, M., Clark, P. M., Macit, C.

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015 The adaptor protein Act1 plays a key role in psoriatic inflammation mediated by IL23 von Lipovsky, A., Slivka, P., Su, Z., Wang, Y., Paulsboe, S.E., Gauvin, D., Wetter, J., Namovic, M., Gauld, S., McGaraughty, S., Goedken, E.

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712 Comparing RNAseq analysis of the mouse IL-23 minicircle model to human psoriasis and other preclinical models of skin inflammation von Leys, L., Bi, Y., Paulsboe, S.E., Su, Z., Olson, L., Wetter, J., Salte, K., Honore, P., Scott, V.E., Wang, Y., McGaraughty, S., Smith, K.

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Pharmacological MRI in awake rats reveals neural activity in area postrema and nucleus tractus solitarius: Relevance as a potential biomarker for detecting drug-induced emesis von Chin, Chih-Liang, Fox, Gerard B., Hradil, Vincent P., Osinski, Mark A., McGaraughty, Steve P., Skoubis, Pamela D., Cox, Bryan F., Luo, Yanping

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