Allosteric Modulators of Steroid Hormone Receptors: Structural Dynamics and Gene Regulation von Kumar, Raj, McEwan, Iain J

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Mechanistic insights into steroid hormone-mediated regulation of the androgen receptor gene von Gillen, Andrew D, Hunter, Irene, Ullner, Ekkehard, McEwan, Iain J

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An androgen receptor N-terminal domain antagonist for treating prostate cancer von Myung, Jae-Kyung, Banuelos, Carmen A, Fernandez, Javier Garcia, Mawji, Nasrin R, Wang, Jun, Tien, Amy H, Yang, Yu Chi, Tavakoli, Iran, Haile, Simon, Watt, Kate, McEwan, Iain J, Plymate, Stephen, Andersen, Raymond J, Sadar, Marianne D

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Regression of Castrate-Recurrent Prostate Cancer by a Small-Molecule Inhibitor of the Amino-Terminus Domain of the Androgen Receptor von Andersen, Raymond J., Mawji, Nasrin R., Wang, Jun, Wang, Gang, Haile, Simon, Myung, Jae-Kyung, Watt, Kate, Tam, Teresa, Yang, Yu Chi, Bañuelos, Carmen A., Williams, David E., McEwan, Iain J., Wang, Yuzhou, Sadar, Marianne D.

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A sting in the tail： the N-terminal domain of the androgen receptor as a drug target von Monaghan, Amy, McEwan, Iain

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Tissue control of androgen action: The ups and downs of androgen receptor expression von Hunter, Irene, Hay, Colin W., Esswein, Bianca, Watt, Kate, McEwan, Iain J.

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Novel Selective Agents for the Degradation of Androgen Receptor Variants to Treat Castration-Resistant Prostate Cancer von Ponnusamy, Suriyan, Coss, Christopher C, Thiyagarajan, Thirumagal, Watts, Kate, Hwang, Dong-Jin, He, Yali, Selth, Luke A, McEwan, Iain J, Duke, Charles B, Pagadala, Jayaprakash, Singh, Geetika, Wake, Robert W, Ledbetter, Christopher, Tilley, Wayne D, Moldoveanu, Tudor, Dalton, James T, Miller, Duane D, Narayanan, Ramesh

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The impact of point mutations in the human androgen receptor: classification of mutations on the basis of transcriptional activity von Hay, Colin W, McEwan, Iain J

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Structure and function of steroid receptor AF1 transactivation domains: induction of active conformations von Lavery, Derek N, McEwan, Iain J

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Breaking apart condensates von McEwan, Iain J.

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Regulation of the androgen receptor by SET9-mediated methylation von Gaughan, Luke, Stockley, Jacqueline, Wang, Nan, McCracken, Stuart R.C, Treumann, Achim, Armstrong, Kelly, Shaheen, Fadhel, Watt, Kate, McEwan, Iain J, Wang, Chenguang, Pestell, Richard G, Robson, Craig N

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An Sp1 Modulated Regulatory Region Unique to Higher Primates Regulates Human Androgen Receptor Promoter Activity in Prostate Cancer Cells von Hay, Colin W, Hunter, Irene, MacKenzie, Alasdair, McEwan, Iain J

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What lies beneath: natural products from marine organisms as nuclear receptor modulators von McEwan, Iain J

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Conformation of the Mineralocorticoid Receptor N-terminal Domain: Evidence for Induced and Stable Structure von Fischer, Katharina, Kelly, Sharon M, Watt, Kate, Price, Nicholas C, McEwan, Iain J

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Mutation of Histidine 874 in the Androgen Receptor Ligand-Binding Domain Leads to Promiscuous Ligand Activation and Altered p160 Coactivator Interactions von Duff, Jennifer, McEwan, Iain J

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The Nuclear Receptor Superfamily at Thirty von McEwan, Iain J.

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Intrinsic disorder in the androgen receptor: identification, characterisation and drugability von McEwan, Iain J

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Nuclear Receptors: One Big Family von McEwan, Iain J.

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New Generation of Selective Androgen Receptor Degraders: Our Initial Design, Synthesis, and Biological Evaluation of New Compounds with Enzalutamide-Resistant Prostate Cancer Activ... von Hwang, Dong-Jin, He, Yali, Ponnusamy, Suriyan, Mohler, Michael L, Thiyagarajan, Thirumagal, McEwan, Iain J, Narayanan, Ramesh, Miller, Duane D

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Ion mobility mass spectrometry unveils conformational effects of drug lead EPI‐001 on the intrinsically disordered N‐terminal domain of the androgen receptor von Ahmed, Ikhlas M. M., Rofe, Adam, Henry, Martyn C., West, Eric, Jamieson, Craig, McEwan, Iain J., Beveridge, Rebecca

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