Peripheral Cannabinoid-1 Receptor Inverse Agonism Reduces Obesity by Reversing Leptin Resistance von Tam, Joseph, Cinar, Resat, Liu, Jie, Godlewski, Grzegorz, Wesley, Daniel, Jourdan, Tony, Szanda, Gergő, Mukhopadhyay, Bani, Chedester, Lee, Liow, Jeih-San, Innis, Robert B., Cheng, Kejun, Rice, Kenner C., Deschamps, Jeffrey R., Chorvat, Robert J., McElroy, John F., Kunos, George

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JD-5006 and JD-5037: Peripherally restricted (PR) cannabinoid-1 receptor blockers related to SLV-319 (Ibipinabant) as metabolic disorder therapeutics devoid of CNS liabilities von Chorvat, Robert J., Berbaum, Jennifer, Seriacki, Kristine, McElroy, John F.

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Behavioral and Pharmacological Validation of the Gerbil Forced-Swim Test: Effects of Neurokinin-1 Receptor Antagonists von Wallace-Boone, Tanya L, Newton, Amy E, Wright, Robert N, Lodge, Nicholas J, McElroy, John F

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Synthesis and Structure−Activity Relationships of 8-(Pyrid-3-yl)pyrazolo[1,5-a]-1,3,5-triazines: Potent, Orally Bioavailable Corticotropin Releasing Factor Receptor-1 (CRF1) Antago... von Gilligan, Paul J, Clarke, Todd, He, Liqi, Lelas, Snjezana, Li, Yu-Wen, Heman, Karen, Fitzgerald, Lawrence, Miller, Keith, Zhang, Ge, Marshall, Anne, Krause, Carol, McElroy, John F, Ward, Kathyrn, Zeller, Kim, Wong, Harvey, Bai, Steven, Saye, Joanne, Grossman, Scott, Zaczek, Robert, Arneric, Stephen P, Hartig, Paul, Robertson, David, Trainor, George

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The CRF1 receptor antagonist DMP696 produces anxiolytic effects and inhibits the stress-induced hypothalamic-pituitary-adrenal axis activation without sedation or ataxia in rats von MCELROY, John F, WARD, Kathryn A, ZELLER, Kim L, JONES, Keith W, GILLIGAN, Paul J, LIQI HE, LELAS, Sniezana

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Effects of CRF1 receptor antagonists and benzodiazepines in the Morris water maze and delayed non-matching to position tests von HOGAN, John B, HODGES, Donald B, LELAS, Snjezana, GILLIGAN, Paul J, MCELROY, John F, LINDNER, Mark D

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Adverse Effects of Gabapentin and Lack of Anti-Allodynic Efficacy of Amitriptyline in the Streptozotocin Model of Painful Diabetic Neuropathy von Lindner, Mark D, Bourin, Clotilde, Chen, Ping, McElroy, John F, Leet, John E, Hogan, John B, Stock, David A, Machet, Frederic

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The anxiolytic CRF1 antagonist DMP696 fails to function as a discriminative stimulus and does not substitute for chlordiazepoxide in rats von LELAS, Snjezana, ZELLER, Kim L, WARD, Kathryn A, MCELROY, John F

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Synthesis, Structure−Activity Relationships, and in Vivo Properties of 3,4-Dihydro-1H-pyrido[2,3-b]pyrazin-2-ones as Corticotropin-Releasing Factor-1 Receptor Antagonists von Dzierba, Carolyn D, Takvorian, Amy G, Rafalski, Maria, Kasireddy-Polam, Padmaja, Wong, Harvey, Molski, Thaddeus F, Zhang, Ge, Li, Yu-Wen, Lelas, Snjezana, Peng, Yong, McElroy, John F, Zaczek, Robert C, Taub, Rebecca A, Combs, Andrew P, Gilligan, Paul J, Trainor, George L

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Novel, highly potent, selective 5-HT2A/D2 receptor antagonists as potential atypical antipsychotics von TAEKYU LEE, ROBICHAUD, Albert J, BOYLE, Kristopher E, YIMIN LU, ROBERTSON, David W, MILLER, Keith J, FITZGERALD, Larry W, MCELROY, John F, LARGENT, Brian L

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Novel piperidine .sigma. receptor ligands as potential antipsychotic drugs von Gilligan, Paul J, Cain, Gary A, Christos, Thomas E, Cook, Leonard, Drummond, Spencer, Johnson, Alexander L, Kergaye, Ahmed A, McElroy, John F, Rohrbach, Kenneth W

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Short- and long-term effects of ovariectomy on food intake, body weight, carcass composition, and brown adipose tissue in rats von McElroy, John F., Wade, George N.

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Piperidinyltetralin .sigma. Ligands von Gilligan, Paul J, Kergaye, Ahmed A, Lewis, Bryan M, McElroy, John F

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Behavioral and Pharmacological Validation of the Gerbil Forced-Swim Test : Effects of Neurokinin-I Receptor Antagonists von WALLACE-BOONE, Tanya L, NEWTON, Amy E, WRIGHT, Robert N, LODGE, Nicholas J, MCELROY, John F

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Cannabinoid receptor antagonists/inverse agonists useful for treating disease conditions, including metabolic disorders and cancers von McElroy, John F, Chorvat, Robert J

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Repetition, Contrariety, and Individualization in Edward II von McElroy, John F.

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CANNABINOID RECEPTOR ANTAGONISTS/INVERSE AGONISTS USEFUL FOR TREATING DISEASE CONDITIONS, INCLUDING METABOLIC DISORDERS AND CANCERS von McElroy, John F, Chorvat, Robert J

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Effects of CRF sub(1) receptor antagonists and benzodiazepines in the Morris water maze and delayed non-matching to position tests von Hogan, John B, Hodges, Donald B, Lelas, Snjezana, Gilligan, Paul J, McElroy, John F, Lindner, Mark D

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Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes von McElroy, John F, Chorvat, Robert J

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The anxiolytic CRF(1) antagonist DMP696 fails to function as a discriminative stimulus and does not substitute for chlordiazepoxide in rats von Lelas, Snjezana, Zeller, Kim L, Ward, Kathryn A, McElroy, John F

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