Discovery of an In Vivo Chemical Probe for BCL6 Inhibition by Optimization of Tricyclic Quinolinones von Harnden, Alice C., Davis, Owen A., Box, Gary M., Hayes, Angela, Johnson, Louise D., Henley, Alan T., de Haven Brandon, Alexis K., Valenti, Melanie, Cheung, Kwai-Ming J., Brennan, Alfie, Huckvale, Rosemary, Pierrat, Olivier A., Talbot, Rachel, Bright, Michael D., Akpinar, Hafize Aysin, Miller, Daniel S. J., Tarantino, Dalia, Gowan, Sharon, de Klerk, Selby, McAndrew, Peter Craig, Le Bihan, Yann-Vaï, Meniconi, Mirco, Burke, Rosemary, Kirkin, Vladimir, van Montfort, Rob L. M., Raynaud, Florence I., Rossanese, Olivia W., Bellenie, Benjamin R., Hoelder, Swen

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Structure-Based Design of Orally Bioavailable 1H‑Pyrrolo[3,2‑c]pyridine Inhibitors of Mitotic Kinase Monopolar Spindle 1 (MPS1) von Naud, Sébastien, Westwood, Isaac M, Faisal, Amir, Sheldrake, Peter, Bavetsias, Vassilios, Atrash, Butrus, Cheung, Kwai-Ming J, Liu, Manjuan, Hayes, Angela, Schmitt, Jessica, Wood, Amy, Choi, Vanessa, Boxall, Kathy, Mak, Grace, Gurden, Mark, Valenti, Melanie, de Haven Brandon, Alexis, Henley, Alan, Baker, Ross, McAndrew, Craig, Matijssen, Berry, Burke, Rosemary, Hoelder, Swen, Eccles, Suzanne A, Raynaud, Florence I, Linardopoulos, Spiros, van Montfort, Rob L. M, Blagg, Julian

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Structure-Based Design of Orally Bioavailable 1 H -Pyrrolo[3,2- c ]pyridine Inhibitors of Mitotic Kinase Monopolar Spindle 1 (MPS1) von Naud, Sébastien, Westwood, Isaac M., Faisal, Amir, Sheldrake, Peter, Bavetsias, Vassilios, Atrash, Butrus, Cheung, Kwai-Ming J., Liu, Manjuan, Hayes, Angela, Schmitt, Jessica, Wood, Amy, Choi, Vanessa, Boxall, Kathy, Mak, Grace, Gurden, Mark, Valenti, Melanie, de Haven Brandon, Alexis, Henley, Alan, Baker, Ross, McAndrew, Craig, Matijssen, Berry, Burke, Rosemary, Hoelder, Swen, Eccles, Suzanne A., Raynaud, Florence I., Linardopoulos, Spiros, van Montfort, Rob L. M., Blagg, Julian

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Abstract 3242: CCT271850, a novel, selective, highly potent and orally bioavailable Mps1 kinase inhibitor von Faisal, Amir, Innocenti, Paolo, Westwood, Isaac, Naud, Sebastan, Schmitt, Jessica, Hayes, Angela, Mak, Grace, Gurden, Mark, Bavetsias, Vassilios, Cheung, Jack, Woodward, Hannah, Sheldrake, Peter, Atrash, Butrus, Burke, Rosemary, Baker, Ross, McAndrew, Craig, Rowlands, Martin, Valenti, Melanie, Workman, Paul, Eccles, Suzanne, Raynaud, Florence, vanMontfort, Rob, Hoelder, Swen, Blagg, Julian, Linardopoulos, Spiros

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Abstract 1817: Characterisation of CCT251455, a novel, selective and highly potent Mps1 kinase inhibitor von Faisal, Amir, Naud, Sebastian, Schmitt, Jessica, Westwood, Isaac, Hayes, Angela, Gurden, Mark, Bavetsias, Vassilios, Berry, Teeara, Mak, Grace, Innocenti, Paolo, Cheung, Jack, Sheldrake, Peter, Atrash, Butrus, Sun, Chongbo, Matijssen, Berry, Burke, Rosemary, Baker, Ross, McAndrew, Craig, Rowlands, Martin, Workman, Paul, Eccles, Suzanne A., Hoelder, Swen, Raynaud, Florence I., vanMontfort, Rob, Blagg, Julian, Linardopoulos, Spiros

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Versatile expression vectors for high-level synthesis of cloned gene products in Escherichia coli von Crowl, Robert, Seamans, Craig, Lomedico, Peter, McAndrew, Stephen

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Versatile expression vectors for high-level synthesis of cloned gene products in Escherichia coli von Crowl, Robert, Seamans, Craig, Lomedico, Peter, McAndrew, Stephen

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