Monoclonal Antibody Conjugates of Doxorubicin Prepared with Branched Peptide Linkers:  Inhibition of Aggregation by Methoxytriethyleneglycol Chains von King, H. Dalton, Dubowchik, Gene M, Mastalerz, Harold, Willner, David, Hofstead, Sandra J, Firestone, Raymond A, Lasch, Shirley J, Trail, Pamela A

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New dual inhibitors of EGFR and HER2 protein tyrosine kinases von Fink, Brian E., Vite, Gregory D., Mastalerz, Harold, Kadow, John F., Kim, Soong-Hoon, Leavitt, Kenneth J., Du, Karen, Crews, Donald, Mitt, Toomas, Wong, Tai W., Hunt, John T., Vyas, Dolatrai M., Tokarski, John S.

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The discovery of BMS-275183: an orally efficacious novel taxane von Mastalerz, Harold, Cook, Donald, Fairchild, Craig R, Hansel, Steven, Johnson, Walter, Kadow, John F, Long, Byron H, Rose, William C, Tarrant, James, Wu, Mu-Jen, Xue, May Quifen, Zhang, Guifen, Zoeckler, Mary, Vyas, Dolatrai M

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Doxorubicin immunoconjugates containing bivalent, lysosomally-Cleavable dipeptide linkages von Dubowchik, Gene M, Radia, Shilpa, Mastalerz, Harold, Walker, Michael A, Firestone, Raymond A, Dalton King, H, Hofstead, Sandra J, Willner, David, Lasch, Shirley J, Trail, Pamela A

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Synthesis of 7β-Sulfur Analogues of Paclitaxel Utilizing a Novel Epimerization of the 7α-Thiol Group von Mastalerz, Harold, Zhang, Guifen, Kadow, John, Fairchild, Craig, Long, Byron, Vyas, Dolatrai M

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Thiol esters from sulfoxides via rearrangement of sulfoxide phosphines to sulfide phosphine oxides von Vedejs, E, Meier, G. P, Powell, D. W, Mastalerz, H

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Stereocontrolled osmylation of medium-ring alkenes: synthesis of a C1-C9 erythronolide fragment von Vedejs, E, Dolphin, J. M, Mastalerz, H

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Synthesis of 7beta-sulfur analogues of paclitaxel utilizing a novel epimerization of the 7alpha-thiol group von Mastalerz, H, Zhang, G, Kadow, J, Fairchild, C, Long, B, Vyas, D M

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Synthesis of a 4β-(hydroxymethyl)carbapenem von MASTALERZ, H, MENARD, M

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Palladium-catalyzed conversion of esters of 4-(trimethylsilyl)-2-buten-1-ol to trimethylsilyl esters: a new carboxyl protecting group von Mastalerz, Harold

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Synthesis of a 4β-carboxyethyl derivative of thienamycin von Bouthillier, Gilles, Mastalerz, Harold, Menard, Marcel

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Synthesis of an esperamicin core analog with an epoxide trigger von Mastalerz, Harold, Doyle, Terrence W, Kadow, John F, Vyas, Dolatrai M

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Synthesis of a hybrid analog of the esperamicin and dynemicin cores von Mastalerz, Harold, Doyle, Terrence W, Kadow, John F, Vyas, Dolatrai M

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Synthesis of Intermediates for the Preparation of Core Analogs of Esperamicin von Mastalerz, H

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Synthesis and antibacterial activity of some novel 6-methyl- and 6-propenyl-substituted carbapenems von Mastalerz, Harold, Menard, Marcel, Ruediger, Edward, Fung-Tomc, Joan

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The synthesis of an asparenomycin analog von Bouthillier, Gilles, Mastalerz, Harold, Ménard, Marcel

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An examination of O-2-isocephems as orally absorbable antibiotics von Mastalerz, Harold, Menard, Marcel, Vinet, Vivianne, Desiderio, James, Fung-Tomc, Joan, Kessler, Robert, Tsai, Yuan

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An alternative approach to the synthesis of the carbapenam ring system. Allenes as acceptor-donor reagents in 3 + 2 annelations von Mastalerz, Harold, Vinet, Vivianne

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THE SYNTHESIS, ANTIBACTERIAL, AND β-LACTAMASE INHIBITORY ACTIVITY OF A NOVEL ASPARENOMYCIN ANALOG von BOUTHILLIER, GILLES, MASTALERZ, HAROLD, MENARD, MARCEL, FUNG-TOMC, JOAN, GRADELSKI, ELIZABETH

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A 2-methylthio-3,5-diaryl-1,3,4-thiadiazolium cation; its reactions, and further exploration of the chemistry of 2-alkyl-3,5-diaryl-1,3,4-thiadiazolium cations von Mastalerz, Harold, Mohammad, Taj, Gibson, Martin S

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