CDK1 structures reveal conserved and unique features of the essential cell cycle CDK von Brown, Nicholas R., Korolchuk, Svitlana, Martin, Mathew P., Stanley, Will A., Moukhametzianov, Rouslan, Noble, Martin E. M., Endicott, Jane A.

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Roger Courtney Martin von Martin, Mathew, Carr, Tom

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FragLitesMinimal, Halogenated Fragments Displaying Pharmacophore Doublets. An Efficient Approach to Druggability Assessment and Hit Generation von Wood, Daniel J, Lopez-Fernandez, J. Daniel, Knight, Leanne E, Al-Khawaldeh, Islam, Gai, Conghao, Lin, Shengying, Martin, Mathew P, Miller, Duncan C, Cano, Céline, Endicott, Jane A, Hardcastle, Ian R, Noble, Martin E. M, Waring, Michael J

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Exiting the tunnel of uncertainty: crystal soak to validated hit von Martin, Mathew P., Noble, Martin E. M.

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Differences in the Conformational Energy Landscape of CDK1 and CDK2 Suggest a Mechanism for Achieving Selective CDK Inhibition von Wood, Daniel J., Korolchuk, Svitlana, Tatum, Natalie J., Wang, Lan-Zhen, Endicott, Jane A., Noble, Martin E.M., Martin, Mathew P.

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Multi-modal and bi-directional effects of a synthetic Δ9-Tetrahydrocannabinol (THC) analogue, Nabilone, on spatio-temporal binding windows: Evidence from the projected hand illusio... von Lim, Mark J H, Iyyalol, Rajan, Lee, Joseph W Y, Martin-Iverson, Mathew T

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Recent Advances in Kinase Drug Discovery Part I: The Editors' Take von Tucker, Julie A., Martin, Mathew P.

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Dexamphetamine influences funneling illusion based on psychometric score von Kassim, Faiz M., Mark Lim, J. H., Albrecht, Matthew A., Martin‐Iverson, Mathew T.

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Bi‐directional and multi‐modal effects of dexamphetamine on spatial binding windows in healthy individuals von Lim, Mark J. H., Loffman, Sean J., Gaus, Katharina, Slawik, Sophie V., Iyyalol, Rajan, Lee, Joseph W. Y., Hepple, Emily K., Martin‐Iverson, Mathew T.

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Dexamphetamine increased speech and visual unimodal illusions in healthy participants without affecting temporal binding window von Voon, Fui‐Ling, Loffman, Sean J., Lim, Mark J. H., Lee, Joseph W. Y., Iyyalol, Rajan, Martin‐Iverson, Mathew T.

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The effects of caffeine and d-amphetamine on spatial span task in healthy participants von Kassim, Faiz M, Lim, J H Mark, Slawik, Sophie V, Gaus, Katharina, Peters, Benjamin, Lee, Joseph W Y, Hepple, Emily K, Rodger, Jennifer, Albrecht, Matthew A, Martin-Iverson, Mathew T

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Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease von Douangamath, Alice, Fearon, Daren, Gehrtz, Paul, Krojer, Tobias, Lukacik, Petra, Owen, C. David, Resnick, Efrat, Strain-Damerell, Claire, Aimon, Anthony, Ábrányi-Balogh, Péter, Brandão-Neto, José, Carbery, Anna, Davison, Gemma, Dias, Alexandre, Downes, Thomas D., Dunnett, Louise, Fairhead, Michael, Firth, James D., Jones, S. Paul, Keeley, Aaron, Keserü, György M., Klein, Hanna F., Martin, Mathew P., Noble, Martin E. M., O’Brien, Peter, Powell, Ailsa, Reddi, Rambabu N., Skyner, Rachael, Snee, Matthew, Waring, Michael J., Wild, Conor, London, Nir, von Delft, Frank, Walsh, Martin A.

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Cyclin-Dependent Kinase Inhibitor Dinaciclib Interacts with the Acetyl-Lysine Recognition Site of Bromodomains von Martin, Mathew P, Olesen, Sanne H, Georg, Gunda I, Schönbrunn, Ernst

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Modulation of ERK5 Activity as a Therapeutic Anti-Cancer Strategy von Miller, Duncan C., Harnor, Suzannah J., Martin, Mathew P., Noble, Richard A., Wedge, Stephen R., Cano, Celine

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Cyclin-Dependent Kinase (CDK) Inhibitors: Structure–Activity Relationships and Insights into the CDK‑2 Selectivity of 6‑Substituted 2‑Arylaminopurines von Coxon, Christopher R, Anscombe, Elizabeth, Harnor, Suzannah J, Martin, Mathew P, Carbain, Benoit, Golding, Bernard T, Hardcastle, Ian R, Harlow, Lisa K, Korolchuk, Svitlana, Matheson, Christopher J, Newell, David R, Noble, Martin E. M, Sivaprakasam, Mangaleswaran, Tudhope, Susan J, Turner, David M, Wang, Lan Z, Wedge, Stephen R, Wong, Christopher, Griffin, Roger J, Endicott, Jane A, Cano, Céline

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Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors von Zhu, Jin-Yi, Cuellar, Rebecca A, Berndt, Norbert, Lee, Hee Eun, Olesen, Sanne H, Martin, Mathew P, Jensen, Jeffrey T, Georg, Gunda I, Schönbrunn, Ernst

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Is there a role for REBOA? A system assessment von Karmy-Jones, Riyad, Friend, Allen, Collins, David, Martin, Mathew J., Long, William

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Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors von Ember, Stuart W. J, Zhu, Jin-Yi, Olesen, Sanne H, Martin, Mathew P, Becker, Andreas, Berndt, Norbert, Georg, Gunda I, Schönbrunn, Ernst

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Comparison of Quantitative Mass Spectrometric Methods for Drug Target Identification by Thermal Proteome Profiling von George, Amy L., Sidgwick, Frances R., Watt, Jessica E., Martin, Mathew P., Trost, Matthias, Marín-Rubio, José Luis, Dueñas, Maria Emilia

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What is the optimal frequency of sink drain decontamination with a foam disinfectant? von Varghese, Martin Mathew, Torres-Teran, Maria M., Greentree, David Henry, Cadnum, Jennifer L., Donskey, Curtis J.

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