An inhibitor of RORγ for chronic pulmonary obstructive disease treatment von Desai, Harshada, Marathe, Megha, Potdar, Varada, Tiwari, Prabhakar, Joshi, Ashwini, Kadam, Sheetal R., Joshi, Arti Rajesh, Kulkarni, Abhay, Bhosale, Vikram, Hadambar, Avinash, Lodhiya, Bhavik, Udupa, Venkatesha, Behera, Dayanidhi, Chaudhari, Sachin S., Das, Sanjib, Bajpai, Malini, Gowda, Nagaraj, Iyer, Pravin S.

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Identification and Characterization of RHOA-Interacting Proteins in Bovine Spermatozoa von Fiedler, Sarah E, Bajpai, Malini, Carr, Daniel W

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Design, Synthesis, and Pharmacological Evaluation of 5,6-Disubstituted Pyridin-2(1H)‑one Derivatives as Phosphodiesterase 10A (PDE10A) Antagonists von Lingam, V. S. Prasadarao, Dahale, Dnyaneshwar H, Rathi, Vijay E, Shingote, Yogesh B, Thakur, Rajni R, Mindhe, Ajit S, Kummari, Srinivas, Khairatkar-Joshi, Neelima, Bajpai, Malini, Shah, Daisy M, Sapalya, Ratika S, Gullapalli, Srinivas, Gupta, Praveen K, Gudi, Girish S, Jadhav, Satyawan B, Pattem, Rambabu, Thomas, Abraham

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848 Novel small molecule HPK1 inhibitor PCC-1 induces strong anti-tumor activity von Das, Sanjib, Mandadi, Sravan, Saini, Jagmohan, Chaudhari, Sachin, Deshpande, Ameya, Chinnapattu, Murugan, Bajpai, Malini, Pangre, Priyanka, Potdar, Varada, Marathe, Megha, Sawant, Pooja, Akarte, Atul, Misra, Chandrasekhar, Das, Subhadip, Singh, Anuj, Das, Avratanu, Lambade, Pandurang, Tirumalasetty, Chaitanya, Patole, Raju, Biswas, Nilanjana, Karande, Vikas, Shah, Heta, Behera, Dayanidhi, Gowda, Nagaraj, Iyer, Pravin

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Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: Part I von Das, Sanjib, Harde, Rajendra L., Shelke, Dnyaneshwar E., Khairatkar-Joshi, Neelima, Bajpai, Malini, Sapalya, Ratika S., Surve, Harshada V., Gudi, Girish S., Pattem, Rambabu, Behera, Dayanidhi B., Jadhav, Satyawan B., Thomas, Abraham

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AKAP3 Selectively Binds PDE4A Isoforms in Bovine Spermatozoa von BAJPAI, Malini, FIEDLER, Sarah E, ZAOHUA HUANG, VIJAYARAGHAVAN, Srinivasan, OLSON, Gary E, LIVERA, Gabriel, CONTI, Marco, CARR, Daniel W

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Role of energy metabolism in the pregnancy interceptive action of Ferula assafoetida and Melia azedarach extracts in rat von Keshri, Govind, Bajpai, Malini, Lakshmi, Vijai, Setty, Bachu Sreenivasulu, Gupta, Gopal

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Abstract 1709: Novel small molecule HPK1 inhibitor induces immunogenic anti-tumor effects von Chaudhari, Sachin S., Bajpai, Malini, Mandadi, Sravan, Kattige, Vidya G., Thorat, Sandeep, Potdar, Varada, Pangre, Priyanka, Sawant, Pooja, Misra, Chandrasekhar, Das, Subhadip, Akarte, Atul, Singh, Anuj, Mahankali, Sandeep, Lambade, Pandurang, Das, Avratanu, Patole, Raju, Udupa, Venkatesha, Sancheti, Pavankumar, Pawar, Pramod K., Kakade, Somesh, R, Vinod K., Biswas, Nilanjana, Shah, Heta, Behera, Dayanidhi, Jain, Pankaj, Gowda, Nagaraj, Iyer, Pravin S.

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AKAP3 Selectively Binds PDE4A Isoforms in Bovine Spermatozoa1 von Bajpai, Malini, Fiedler, Sarah E, Huang, Zaohua, Vijayaraghavan, Srinivasan, Olson, Gary E, Livera, Gabriel, Conti, Marco, Carr, Daniel W

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MK2: a novel molecular target for anti-inflammatory therapy von Duraisamy, Senthil, Bajpai, Malini, Bughani, Usha, Dastidar, Sunanda G, Ray, Abhijit, Chopra, Puneet

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Imidazopyridazinones as novel PDE7 inhibitors: SAR and in vivo studies in Parkinson’s disease model von Banerjee, Abhisek, Patil, Sandip, Pawar, Mahesh Y., Gullapalli, Srinivas, Gupta, Praveen K., Gandhi, Maulik N., Bhateja, Deepak K., Bajpai, Malini, Sangana, Ramachandra Rao, Gudi, Girish S., Khairatkar-Joshi, Neelima, Gharat, Laxmikant A.

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Abstract 463: GRC 54276, a novel small molecule inhibitor of HPK1 has entered phase 1/2 clinical trial insolid malignancies and Hodgkin’s/non Hodgkin’s lymphoma von Mandadi, Sravan, Das, Sanjib, Bajpai, Malini, Saini, Jagmohan, Chinnapattu, Murugan, Patale, Sanjay, Patil, Sandip, Kadlag, Nanasaheb, Waghmare, Nayan, Gavhane, Balasaheb, Deshpande, Ameya, Dahale, Dnyaneshwar, Kattige, Vidya, Pangre, Priyanka, Singh, Namrata, Kashyap, Ekta, Marathe, Megha, Mani, Jiju, Akarte, Atul, Misra, Chandrasekhar, Das, Subhadip, Singh, Anuj, Lambade, Pandurang, Das, Avratanu, Tirumalasetty, Chaitanya, Patole, Raju, Biswas, Nilanjana, Karande, Vikas, Shah, Heta, Behera, Dayanidhi, Jain, Pankaj, Sancheti, Pavankumar, Pawar, Pramod, KR, Vinod, Udupa, Venkatesha, Chaudhari, Sachin S., Gowda, Nagaraj, Iyer, Pravin S.

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Discovery of benzo[d]imidazo[5,1-b]thiazole as a new class of phosphodiesterase 10A inhibitors von Banerjee, Abhisek, Narayana, Lakshminarayana, Raje, Firoj A., Pisal, Dnyandeo V., Kadam, Pradip A., Gullapalli, Srinivas, Kumar, Hemant, More, Sandeep V., Bajpai, Malini, Sangana, Ramachandra Rao, Jadhav, Satyawan, Gudi, Girish S., Khairatkar-Joshi, Neelima, Merugu, Ravi R.T., Voleti, Sreedhara R., Gharat, Laxmikant A.

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Abstract 1804: IND-ready clinical candidate for HPK1 developed with excellent efficacy and safety profile von Mandadi, Sravan, Das, Sanjib, Saini, Jagmohan, Chaudhari, Sachin S., Chinnapattu, Murugan, Deshpande, Ameya, Dahale, Dnyaneshwar, Bajpai, Malini, Pangre, Priyanka, Singh, Namrata, Kashyap, Ekta, Marathe, Megha, Mani, Jiju, Akarte, Atul, Misra, Chandrasekhar, Das, Subhadip, Singh, Anuj, Das, Avratanu, Lambade, Pandurang, Tirumalasetty, Chaitanya, Patole, Raju, Biswas, Nilanjana, Karande, Vikas, Shah, Heta, Behera, Dayanidhi, Jain, Pankaj, Sancheti, Pavankumar, Kakade, Somesh, Pawar, Pramod K., KR, Vinod, Udupa, Venkatesha, Gowda, Nagaraj, Iyer, Pravin S.

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Isothiazole and isoxazole fused pyrimidones as PDE7 inhibitors: SAR and pharmacokinetic evaluation von Banerjee, Abhisek, Yadav, Pravin S., Bajpai, Malini, Sangana, Ramachandra Rao, Gullapalli, Srinivas, Gudi, Girish S., Gharat, Laxmikant A.

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Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: part II von Das, Sanjib, Shelke, Dnyaneshwar E, Harde, Rajendra L, Avhad, Vijayshree B, Khairatkar-Joshi, Neelima, Gullapalli, Srinivas, Gupta, Praveen K, Gandhi, Maulik N, Bhateja, Deepak K, Bajpai, Malini, Joshi, Ashwini A, Marathe, Megha Y, Gudi, Girish S, Jadhav, Satyawan B, Mahat, Mahamad Yunnus A, Thomas, Abraham

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Identification and Characterization of RHOA-lnteracting Proteins in Bovine Spermatozoa von FIEDLER, Sarah E, BAJPAI, Malini, CARR, Daniel W

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Development of a cell death-based method for the screening of nuclear factor-kappaB inhibitors von Chopra, Puneet, Bajpai, Malini, Dastidar, Sunanda G, Ray, Abhijit

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An improved zinc cocktail-mediated fluorescence polarization-based kinase assay for high-throughput screening of kinase inhibitors von Chopra, Puneet, Nanda, Kamna, Chatterjee, Mou, Bajpai, Malini, Dastidar, Sunanda G., Ray, Abhijit

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Spleen tyrosine kinase: a novel target for therapeutic intervention of rheumatoid arthritis von Bajpai, Malini, Chopra, Puneet, Dastidar, Sunanda G, Ray, Abhijit

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