Molecular design and chemical synthesis of potent enediynes. 1. Dynemicin model systems equipped with N-tethered triggering devices von Nicolaou, K. C, Maligres, P, Suzuki, T, Wendeborn, S. V, Dai, W. M, Chadha, R. K

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Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides: Synthesis of the Merck HIV-1 protease inhibitor epoxide intermediate von Maligres, P.E., Upadhyay, V., Rossen, K., Cianciosi, S.J., Purick, R.M., Eng, K.K., Reamer, R.A., Askin, D., Volante, R.P., Reider, P.J.

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Synthesis of a β-Amino Acid Pharmacophore via a β-Lactam Intermediate von Angelaud, Rémy, Zhong, Yong-Li, Maligres, Peter, Lee, Jaemoon, Askin, David

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Cyclic imidate salts in acyclic stereochemistry: Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides von Maligres, P.E., Weissman, S.A., Upadhyay, V., Cianciosi, S.J., Reamer, R.A., Purick, R.M., Sager, J., Rossen, K., Eng, K.K., Askin, D., Volante, R.P., Reider, P.J.

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Synthesis of a Muscarinic Receptor Antagonist via a Diastereoselective Michael Reaction, Selective Deoxyfluorination and Aromatic Metal−Halogen Exchange Reaction von Mase, Toshiaki, Houpis, Ioannis N, Akao, Atsushi, Dorziotis, Ilias, Emerson, Khateeta, Hoang, Thoa, Iida, Takehiko, Itoh, Takahiro, Kamei, Keisuke, Kato, Shinji, Kato, Yoshiaki, Kawasaki, Masashi, Lang, Fengrui, Lee, Jaemoon, Lynch, Joseph, Maligres, Peter, Molina, Audrey, Nemoto, Takayuki, Okada, Shigemitsu, Reamer, Robert, Song, Jake Z, Tschaen, David, Wada, Toshihiro, Zewge, Daniel, Volante, R. P, Reider, Paul J, Tomimoto, Koji

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A highly catalytic robust palladium catalyzed cyanation of aryl bromides von Maligres, Peter E., Waters, Marjorie S., Fleitz, Fred, Askin, David

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Highly Regioselective DABCO-Catalyzed Nucleophilic Aromatic Substitution (SNAr) Reaction of Methyl 2,6-Dichloronicotinate with Phenols von Shi, Yao-Jun, Humphrey, Guy, Maligres, Peter E., Reamer, Robert A., Williams, J. Michael

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Enantioselective Hydrogenation of α-Aryloxy α,β-Unsaturated Acids. Asymmetric Synthesis of α-Aryloxycarboxylic Acids von Maligres, Peter E, Krska, Shane W, Humphrey, Guy R

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Nosylaziridines: Activated aziridine electrophiles von Maligres, Peter E., See, Marjorie M., Askin, David, Reider, Paul J.

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Selectivity and Mechanism of Action of Novel DNA-Cleaving Sulfones von Nicolaou, K. C., Wendeborn, S., Maligres, P., Isshiki, K., Zein, N., Ellestad, G.

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A New Class of DNA-Cleaving Molecules: pH-Dependent DNA Cleavage by Propargylic and Allenic Sulfones von Nicolaou, K. C., Skokotas, G., Maligres, P., Zuccarello, G., Schweiger, E. J., Toshima, K., Wendeborn, S.

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A new designed tumor selective daunomycin derivative von Maligres, P.E., Nicolaou, K.C., Wrasidlo, W.

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DNA-cleavage and antitumor activity of designed molecules with conjugated phosphine oxide-allene-ene-yne functionalities von Nicolaou, K. C, Maligres, P, Shin, J, De Leon, E, Rideout, Darryl

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Stereocontrolled Preparation of a Nonpeptidal (−)-Spirobicyclic NK-1 Receptor Antagonist von Maligres, Peter E, Waters, Marjorie M, Lee, Jaemoon, Reamer, Robert A, Askin, David, Ashwood, Michael S, Cameron, Mark

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Thiol addition to aryl propargyl alcohols under mild conditions: an accelerating neighboring group effect von See Waters, Marjorie, Cowen, Jennifer A, McWilliams, J.Christopher, Maligres, Peter E, Askin, David

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Synthesis of a Muscarinic Receptor Antagonist via a Diastereoselective Michael Reaction, Selective Deoxyfluorination and Aromatic Metal-Halogen Exchange Reaction von Mase, Toshiaki, Houpis, Ioannis N, Akao, Atsushi, Dorziotis, Ilias, Emerson, Khateeta, Hoang, Thoa, Iida, Takehiko, Itoh, Takahiro, Kamei, Keisuke, Kato, Shinji, Kawasaki, Masashi, Lang, Fengrui, Lee, Jaemoon, Lynch, Joseph, Maligres, Peter, Molina, Audrey, Nemoto, Takayuki, Okada, Shigemitsu, Reamer, Robert, Song, Zhiguo J, Tschaen, David, Wada, Toshihiro, Zewge, David, Volante, R. P, Reider, Paul J, Tomimoto, Koji

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Synthesis of the orally active spiroindoline-based growth hormone secretagogue, MK-677 von Maligres, Peter E., Houpis, Ioannis, Rossen, Kai, Molina, Audrey, Sager, Jess, Upadhyay, Veena, Wells, Kenneth M., Reamer, Robert A., Lynch, Joseph E., Askin, David, Volante, R.P., Reider, Paul J., Houghton, Peter

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Preparation of a clinically investigated ras farnesyl transferase inhibitor von Maligres, Peter E., Waters, Marjorie S., Weissman, Steven A., McWilliams, J. Christopher, Lewis, Stephanie, Cowen, Jennifer, Reamer, Robert A., Volante, R. P., Reider, Paul J., Askin, David

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Porcine liver esterase-catalyzed enantioselective hydrolysis of a prochiral diester into its optically pure ( S)-ester acid, a precursor to a growth hormone secretagogue von Chartrain, Michel, Maligres, Peter, Cohen, Deborah, Upadhyay, Veena, Pecore, Victor, Askin, David, Greasham, Randolph

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Preparation of (S)-3-Carbethoxy-3-benzylpiperidine and the Growth Hormone Secretagogue L-163,540 von Maligres, Peter E, Chartrain, Michel M, Upadhyay, Veena, Cohen, Deborah, Reamer, Robert A, Askin, David, Volante, R. P, Reider, Paul J

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