Dual hypocretin receptor antagonism is more effective for sleep promotion than antagonism of either receptor alone von Morairty, Stephen R, Revel, Florent G, Malherbe, Pari, Moreau, Jean-Luc, Valladao, Daniel, Wettstein, Joseph G, Kilduff, Thomas S, Borroni, Edilio

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Biochemical and Electrophysiological Characterization of Almorexant, a Dual Orexin 1 Receptor (OX1)/Orexin 2 Receptor (OX2) Antagonist: Comparison with Selective OX1 and OX2 Antago... von Malherbe, Pari, Borroni, Edilio, Pinard, Emmanuel, Wettstein, Joseph G, Knoflach, Frédéric

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Molecular cloning and functional characterization of human vesicular glutamate transporter 3 von Takamori, Shigeo, Malherbe, Pari, Broger, Clemens, Jahn, Reinhard

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Positive Allosteric Modulators of Metabotropic Glutamate 1 Receptor: Characterization, Mechanism of Action, and Binding Site von Knoflach, Frédéric, Mutel, Vincent, Jolidon, Synèse, James N. C. Kew, Malherbe, Pari, Vieira, Eric, Wichmann, Jürgen, Kemp, John A.

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Mutational Analysis and Molecular Modeling of the Binding Pocket of the Metabotropic Glutamate 5 Receptor Negative Modulator 2-Methyl-6-(phenylethynyl)-pyridine von Malherbe, Pari, Kratochwil, Nicole, Zenner, Marie-Thérèse, Piussi, Jenny, Diener, Catherine, Kratzeisen, Claudia, Fischer, Christophe, Porter, Richard H P

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Mutational Analysis and Molecular Modeling of the Allosteric Binding Site of a Novel, Selective, Noncompetitive Antagonist of the Metabotropic Glutamate 1 Receptor von Malherbe, Pari, Kratochwil, Nicole, Knoflach, Frédéric, Zenner, Marie-Thérèse, Kew, James N C, Kratzeisen, Claudia, Maerki, Hans P, Adam, Geo, Mutel, Vincent

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Comparison of the binding pockets of two chemically unrelated allosteric antagonists of the mGlu5 receptor and identification of crucial residues involved in the inverse agonism of... von Malherbe, Pari, Kratochwil, Nicole, Mühlemann, Andreas, Zenner, Marie‐Thérèse, Fischer, Christophe, Stahl, Martin, Gerber, Paul R., Jaeschke, Georg, Porter, Richard H. P.

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Me-Talnetant and Osanetant Interact within Overlapping but Not Identical Binding Pockets in the Human Tachykinin Neurokinin 3 Receptor Transmembrane Domains von Malherbe, Pari, Bissantz, Caterina, Marcuz, Anne, Kratzeisen, Claudia, Zenner, Marie-Thérèse, Wettstein, Joseph G, Ratni, Hasane, Riemer, Claus, Spooren, Will

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Determination of key amino acids implicated in the actions of allosteric modulation by 3,3′-difluorobenzaldazine on rat mGlu5 receptors von Mühlemann, Andreas, Ward, Natalie A., Kratochwil, Nicole, Diener, Catherine, Fischer, Christophe, Stucki, Andy, Jaeschke, Georg, Malherbe, Pari, Porter, Richard H.P.

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Identification of Essential Residues Involved in the Glutamate Binding Pocket of the Group II Metabotropic Glutamate Receptor von Malherbe, P, Knoflach, F, Broger, C, Ohresser, S, Kratzeisen, C, Adam, G, Stadler, H, Kemp, J A, Mutel, V

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The positive allosteric GABAB receptor modulator rac-BHFF enhances baclofen-mediated analgesia in neuropathic mice von Zemoura, Khaled, Ralvenius, William T., Malherbe, Pari, Benke, Dietmar

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The positive allosteric GABAB receptor modulator rac-BHFF enhances baclofen-mediated analgesia in neuropathic mice von Zemoura, Khaled, Ralvenius, William T, Malherbe, Pari, Benke, Dietmar

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Recombinant GABAA receptor function and ethanol von Sigel, Erwin, Baur, Roland, Malherbe, Pari

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Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: comparison with the selective OX1 antagonist SB-674042 and the selective OX2 anta... von Malherbe, Pari, Roche, Olivier, Marcuz, Anne, Kratzeisen, Claudia, Wettstein, Joseph G, Bissantz, Caterina

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Stoichiometry of a recombinant GABAA receptor deduced from mutation-induced rectification von Backus, Kurt H, Arigoni, Michele, Drescher, Uwe, Scheurer, Louis, Malherbe, Pari, Möhler, Hanns, Benson, Jack A

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Inhibition of alcohol self-administration by positive allosteric modulators of the GABAB receptor in rats: lack of tolerance and potentiation of baclofen von Maccioni, Paola, Vargiolu, Daniela, Thomas, Andrew W., Malherbe, Pari, Mugnaini, Claudia, Corelli, Federico, Leite-Morris, Kimberly A., Gessa, Gian Luigi, Colombo, Giancarlo

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Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: Biochemical and electrophysiological characterization von Malherbe, Pari, Knoflach, Frédéric, Marcuz, Anne, Bohnert, Claudia, Weber, Michael, Knust, Henner, Ratni, Hasane, Spooren, Will, Ballard, Theresa M., Bissantz, Caterina

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Reduction of alcohol intake by the positive allosteric modulator of the GABA(B) receptor, rac-BHFF, in alcohol-preferring rats von Loi, Barbara, Maccioni, Paola, Lobina, Carla, Carai, Mauro A M, Gessa, Gian Luigi, Thomas, Andrew W, Malherbe, Pari, Colombo, Giancarlo

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The positive allosteric modulator of the GABA(B) receptor, rac-BHFF, suppresses alcohol self-administration von Maccioni, Paola, Thomas, Andrew W, Carai, Mauro A M, Gessa, Gian Luigi, Malherbe, Pari, Colombo, Giancarlo

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Identification of a Crucial Amino Acid in the Helix Position 6.51 of Human Tachykinin Neurokinin 1 and 3 Receptors Contributing to the Insurmountable Mode of Antagonism by Dual NK... von Bissantz, Caterina, Bohnert, Claudia, Hoffmann, Torsten, Marcuz, Anne, Schnider, Patrick, Malherbe, Pari

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