Binding Mode and Structure-Activity Relationships around Direct Inhibitors of the Nrf2-Keap1 Complex von Jnoff, Eric, Albrecht, Claudia, Barker, John J., Barker, Oliver, Beaumont, Edward, Bromidge, Steven, Brookfield, Frederick, Brooks, Mark, Bubert, Christian, Ceska, Tom, Corden, Vincent, Dawson, Graham, Duclos, Stephanie, Fryatt, Tara, Genicot, Christophe, Jigorel, Emilie, Kwong, Jason, Maghames, Rosemary, Mushi, Innocent, Pike, Richard, Sands, Zara A., Smith, Myron A., Stimson, Christopher C., Courade, Jean-Philippe

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Discovery of an Orally Bioavailable Pan αv Integrin Inhibitor for Idiopathic Pulmonary Fibrosis von Anderson, Niall A, Campos, Sebastien, Butler, Sharon, Copley, Royston C. B, Duncan, Ian, Harrison, Stephen, Le, Joelle, Maghames, Rosemary, Pastor-Garcia, Aleix, Pritchard, John M, Rowedder, James E, Smith, Claire E, Thomas, Jack, Vitulli, Giovanni, Macdonald, Simon J. F

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Design, synthesis and structure-activity relationships of a novel class of sulfonylpyridine inhibitors of Interleukin-2 inducible T-cell kinase (ITK) von Trani, Giancarlo, Barker, John J, Bromidge, Steven M, Brookfield, Frederick A, Burch, Jason D, Chen, Yuan, Eigenbrot, Charles, Heifetz, Alexander, Ismaili, M Hicham A, Johnson, Adam, Krülle, Thomas M, MacKinnon, Colin H, Maghames, Rosemary, McEwan, Paul A, Montalbetti, Christian A G N, Ortwine, Daniel F, Pérez-Fuertes, Yolanda, Vaidya, Darshan G, Wang, Xiaolu, Zarrin, Ali A, Pei, Zhonghua

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Structure-based design and synthesis of potent benzothiazole inhibitors of interleukin-2 inducible T cell kinase (ITK) von MacKinnon, Colin H., Lau, Kevin, Burch, Jason D., Chen, Yuan, Dines, Jonathon, Ding, Xiao, Eigenbrot, Charles, Heifetz, Alexander, Jaochico, Allan, Johnson, Adam, Kraemer, Joachim, Kruger, Susanne, Krülle, Thomas M., Liimatta, Marya, Ly, Justin, Maghames, Rosemary, Montalbetti, Christian A.G.N., Ortwine, Daniel F., Pérez-Fuertes, Yolanda, Shia, Steven, Stein, Daniel B., Trani, Giancarlo, Vaidya, Darshan G., Wang, Xiaolu, Bromidge, Steven M., Wu, Lawren C., Pei, Zhonghua

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Inside Cover: Binding Mode and Structure-Activity Relationships around Direct Inhibitors of the Nrf2-Keap1 Complex (ChemMedChem 4/2014) von Jnoff, Eric, Albrecht, Claudia, Barker, John J., Barker, Oliver, Beaumont, Edward, Bromidge, Steven, Brookfield, Frederick, Brooks, Mark, Bubert, Christian, Ceska, Tom, Corden, Vincent, Dawson, Graham, Duclos, Stephanie, Fryatt, Tara, Genicot, Christophe, Jigorel, Emilie, Kwong, Jason, Maghames, Rosemary, Mushi, Innocent, Pike, Richard, Sands, Zara A., Smith, Myron A., Stimson, Christopher C., Courade, Jean-Philippe

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