Exploring Factors Influencing Stroke Risk: Insights From a Predictive Analysis von Murugesan, Venkatram, Natesan, Murugesan, Sulthana, Vahidha, Donapaty, Pranav R

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Biphenylsulfonamide Endothelin Receptor Antagonists. 4. Discovery of N-[[2‘-[[(4,5-Dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1‘-biphenyl]- 2-yl]methyl]-N,3,3-trimethyl... von Murugesan, Natesan, Gu, Zhengxiang, Spergel, Steven, Young, Marian, Chen, Ping, Mathur, Arvind, Leith, Leslie, Hermsmeier, Mark, Liu, Eddie C.-K, Zhang, Rongan, Bird, Eileen, Waldron, Tom, Marino, Anthony, Koplowitz, Barry, Humphreys, W. Griffith, Chong, Saeho, Morrison, Richard A, Webb, Maria L, Moreland, Suzanne, Trippodo, Nick, Barrish, Joel C

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Discovery of N-Isoxazolyl Biphenylsulfonamides as Potent Dual Angiotensin II and Endothelin A Receptor Antagonists von Murugesan, Natesan, Tellew, John E, Gu, Zhengxiang, Kunst, Bridgette L, Fadnis, Leena, Cornelius, Lyndon A, Baska, Rose Ann F, Yang, Yifan, Beyer, Sophie M, Monshizadegan, Hossain, Dickinson, Kenneth E, Panchal, Balkrushna, Valentine, Maria T, Chong, Saeho, Morrison, Richard A, Carlson, Kenneth E, Powell, James R, Moreland, Suzanne, Barrish, Joel C, Kowala, Mark C, Macor, John E

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The Discovery of Sulfonamide Endothelin Antagonists and the Development of the Orally Active ETA Antagonist 5-(Dimethylamino)-N-(3,4-dimethyl-5- isoxazolyl)-1-naphthalenesulfonamid... von Stein, Philip D, Hunt, John T, Floyd, David M, Moreland, Suzanne, Dickinson, Kenneth E. J, Mitchell, Caroline, Liu, Eddie C.-K, Webb, Maria L, Murugesan, Natesan

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Standardization and quantification of total tannins, condensed tannin and soluble phlorotannins extracted from thirty-two drifted coastal macroalgae using high performance liquid c... von Petchidurai, Ganeshan, Nagoth, Joseph Amruthraj, John, Maria Sindhura, Sahayaraj, Kitherian, Murugesan, Natesan, Pucciarelli, Sandra

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Discovery of 4′-[(Imidazol-1-yl)methyl]biphenyl-2-sulfonamides as dual endothelin/Angiotensin II receptor antagonists von Tellew, John E, Baska, Rose Ann F, Beyer, Sophie M, Carlson, Kenneth E, Cornelius, Lyndon A, Fadnis, Leena, Gu, Zhengxiang, Kunst, Bridgette L, Kowala, Mark C, Monshizadegan, Hossain, Murugesan, Natesan, Ryan, Carol S, Valentine, Maria T, Yang, Yifan, Macor, John E

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Optimization of Nicotinamides as Potent and Selective IRAK4 Inhibitors with Efficacy in a Murine Model of Psoriasis von Nair, Satheesh, Kumar, Sreekantha Ratna, Paidi, Venkatram Reddy, Sistla, Ramesh, Kantheti, Durgarao, Polimera, Subba Rao, Thangavel, Soodamani, Mukherjee, Amrita Jha, Das, Mitalee, Bhide, Rajeev S, Pitts, William J, Murugesan, Natesan, Dudhgoankar, Shailesh, Nagar, Jignesh, Subramani, Siva, Mazumder, Debarati, Carman, Julie A, Holloway, Deborah A, Li, Xin, Fereshteh, Mark P, Ruepp, Stefan, Palanisamy, Kamalavenkatesh, Mariappan, T. Thanga, Maddi, Srinivas, Saxena, Ajay, Elzinga, Paul, Chimalakonda, Anjaneya, Ruan, Qian, Ghosh, Kaushik, Bose, Sucharita, Sack, John, Yan, Chunhong, Kiefer, Susan E, Xie, Dianlin, Newitt, John A, Saravanakumar, S. Pon, Rampulla, Richard A, Barrish, Joel C, Carter, Percy H, Hynes, John

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Reductions in log P Improved Protein Binding and Clearance Predictions Enabling the Prospective Design of Cannabinoid Receptor (CB1) Antagonists with Desired Pharmacokinetic Proper... von Ellsworth, Bruce A, Sher, Philip M, Wu, Ximao, Wu, Gang, Sulsky, Richard B, Gu, Zhengxiang, Murugesan, Natesan, Zhu, Yeheng, Yu, Guixue, Sitkoff, Doree F, Carlson, Kenneth E, Kang, Liya, Yang, Yifan, Lee, Ning, Baska, Rose A, Keim, William J, Cullen, Mary Jane, Azzara, Anthony V, Zuvich, Eva, Thomas, Michael A, Rohrbach, Kenneth W, Devenny, James J, Godonis, Helen E, Harvey, Susan J, Murphy, Brian J, Everlof, Gerry G, Stetsko, Paul I, Gudmundsson, Olafur, Johnghar, Susan, Ranasinghe, Asoka, Behnia, Kamelia, Pelleymounter, Mary Ann, Ewing, William R

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Dual Angiotensin II and Endothelin A Receptor Antagonists:  Synthesis of 2‘-Substituted N-3-Isoxazolyl Biphenylsulfonamides with Improved Potency and Pharmacokinetics von Murugesan, Natesan, Gu, Zhengxiang, Fadnis, Leena, Tellew, John E, Baska, Rose Ann F, Yang, Yifan, Beyer, Sophie M, Monshizadegan, Hossain, Dickinson, Kenneth E, Valentine, Maria T, Humphreys, W. Griffith, Lan, Shih-Jung, Ewing, William R, Carlson, Kenneth E, Kowala, Mark C, Zahler, Robert, Macor, John E

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Discovery and Structure-Activity Relationships of Sulfonamide ETA-Selective Antagonists von Stein, Philip D, Floyd, David M, Bisaha, Sharon, Dickey, Joyce, Girotra, Ravindar N, Gougoutas, Jack Z, Kozlowski, Michael, Lee, Ving G, Liu, Eddie C.-K

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Chemistry of the alkali-labile lesion formed from iron(II) bleomycin and d(CGCTTTAAAGCG) von Sugiyama, Hiroshi, Xu, Cheng, Murugesan, Natesan, Hecht, Sidney M, Van der Marel, Gijs A, Van Boom, Jacques H

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The chemistry of vicinal tricarbonyls. A stable vinyl tricarbonyl hydrate as a di- and trielectrophile von Wasserman, Harry H, Fukuyama, James, Murugesan, Natesan, Van Duzer, John, Lombardo, Louis, Rotello, Vincent, McCarthy, Keith

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Characterization of a novel and selective CB1 antagonist as a radioligand for receptor occupancy studies von Yang, Yifan, Miller, Keith J., Zhu, Yeheng, Hong, Yang, Tian, Yuan, Murugesan, Natesan, Gu, Zhengxiang, O’Tanyi, Eva, Keim, William J., Rohrbach, Kenneth W., Johnghar, Susan, Behnia, Kamelia, Pelleymounter, Mary Ann, Carlson, Kenneth E., Ewing, William R.

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Synthesis and In Vivo Evaluation of Novel PET Radioligands for Imaging the Endothelin-A Receptor von Mathews, William B, Murugesan, Natesan, Xia, Jinsong, Scheffel, Ursula, Hilton, John, Ravert, Hayden T, Dannals, Robert F, Szabo, Zsolt

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Structure of the alkali-labile product formed during iron(II)-bleomycin-mediated DNA strand scission von Sugiyama, Hiroshi, Xu, Cheng, Murugesan, Natesan, Hecht, Sidney M

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Tryptamine and homotryptamine-based sulfonamides as potent and selective inhibitors of 15-lipoxygenase von Weinstein, David S., Liu, Wen, Gu, Zhengxiang, Langevine, Charles, Ngu, Khehyong, Fadnis, Leena, Combs, Donald W., Sitkoff, Doree, Ahmad, Saleem, Zhuang, Shaobin, Chen, Xing, Wang, Feng-Lai, Loughney, Deborah A., Atwal, Karnail S., Zahler, Robert, Macor, John E., Madsen, Cort S., Murugesan, Natesan

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Design and SAR of selective T-type calcium channel antagonists containing a biaryl sulfonamide core von Hangeland, Jon J., Cheney, Daniel L., Friends, Todd J., Swartz, Stephen, Levesque, Paul C., Rich, Adam J., Sun, Lucy, Bridal, Terry R., Adam, Leonard P., Normandin, Diane E., Murugesan, Natesan, Ewing, William R.

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Activation of oxygen and mediation of DNA degradation by manganese-bleomycin von Ehrenfeld, Guy M, Murugesan, Natesan, Hecht, Sidney M

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TRICYCLIC HETEROARYL COMPOUNDS USEFUL AS IRAK4 INHIBITORS von SARKUNAM, Kandhasamy, PAIDI, Venkatram Reddy, MURUGESAN, Natesan, NAIR, Satheesh Kesavan, SISTLA, Ramesh Kumar, HYNES, John

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von Jalagam, Prasada Rao, Panda, Manoranjan, Natesan, Murugesan, Devasthale, Pratik, Nara, Susheel Jethanand

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