A Survey of the Borrowing Hydrogen Approach to the Synthesis of some Pharmaceutically Relevant Intermediates von Leonard, John, Blacker, A. John, Marsden, Stephen P, Jones, Martin F, Mulholland, Keith R, Newton, Rebecca

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The Identification of Potent, Selective, and Orally Available Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase: The Discovery of AZD0156 (8-{6-[3-(Dimethylamino)propoxy]pyr... von Pike, Kurt G, Barlaam, Bernard, Cadogan, Elaine, Campbell, Andrew, Chen, Yingxue, Colclough, Nicola, Davies, Nichola L, de-Almeida, Camila, Degorce, Sebastien L, Didelot, Myriam, Dishington, Allan, Ducray, Richard, Durant, Stephen T, Hassall, Lorraine A, Holmes, Jane, Hughes, Gareth D, MacFaul, Philip A, Mulholland, Keith R, McGuire, Thomas M, Ouvry, Gilles, Pass, Martin, Robb, Graeme, Stratton, Natalie, Wang, Zhenhua, Wilson, Joanne, Zhai, Baochang, Zhao, Kang, Al-Huniti, Nidal

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An (R)-Imine Reductase Biocatalyst for the Asymmetric Reduction of Cyclic Imines von Hussain, Shahed, Leipold, Friedemann, Man, Henry, Wells, Elizabeth, France, Scott P., Mulholland, Keith R., Grogan, Gideon, Turner, Nicholas J.

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One-Pot Cascade Synthesis of Mono- and Disubstituted Piperidines and Pyrrolidines using Carboxylic Acid Reductase (CAR), ω‑Transaminase (ω-TA), and Imine Reductase (IRED) Biocataly... von France, Scott P, Hussain, Shahed, Hill, Andrew M, Hepworth, Lorna J, Howard, Roger M, Mulholland, Keith R, Flitsch, Sabine L, Turner, Nicholas J

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The Identification of Potent, Selective, and Orally Available Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase: The Discovery of AZD0156 (8-{6-[3-(Dimethylamino)propoxy]pyr... von Pike, Kurt G, Barlaam, Bernard, Cadogan, Elaine, Campbell, Andrew, Chen, Yingxue, Colclough, Nicola, Davies, Nichola L, de-Almeida, Camila, Degorce, Sebastien L, Didelot, Myriam, Dishington, Allan, Ducray, Richard, Durant, Stephen T, Hassall, Lorraine A, Holmes, Jane, Hughes, Gareth D, MacFaul, Philip A, Mulholland, Keith R, McGuire, Thomas M, Ouvry, Gilles, Pass, Martin, Robb, Graeme, Stratton, Natalie, Wang, Zhenhua, Wilson, Joanne, Zhai, Baochang, Zhao, Kang, Al-Huniti, Nidal

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Double Arylation of Allyl Alcohol via a One-Pot Heck Arylation–Isomerization–Acylation Cascade von Colbon, Paul, Ruan, Jiwu, Purdie, Mark, Mulholland, Keith, Xiao, Jianliang

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Bifunctional catalysis: direct reductive amination of aliphatic ketones with an iridium-phosphate catalyst von Villa-Marcos, Barbara, Li, Chaoqun, Mulholland, Keith R, Hogan, Philip J, Xiao, Jianliang

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Development of a Chemoenzymatic Route to (R)‑Allyl-(3-amino-2-(2-methylbenzyl)propyl)carbamate von Lindhagen, Marika, Klingstedt, Tomas, Andersen, Søren M, Mulholland, Keith R, Tinkler, Laura, McPheators, Gary, Chubb, Richard

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Efficient Synthesis of (S)‑1-(5-Fluoropyrimidin-2-yl)ethylamine Using an ω‑Transaminase Biocatalyst in a Two-Phase System von Meadows, Rebecca E, Mulholland, Keith R, Schürmann, Martin, Golden, Michael, Kierkels, Hans, Meulenbroeks, Elise, Mink, Daniel, May, Oliver, Squire, Christopher, Straatman, Harrie, Wells, Andrew S

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Glycosylated Foldamers To Probe the Carbohydrate−Carbohydrate Interaction von Simpson, Graham L, Gordon, Andrew H, Lindsay, David M, Promsawan, Netnepa, Crump, Matthew P, Mulholland, Keith, Hayter, Barry R, Gallagher, Timothy

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Pseudocyst formation in gastric ectopic pancreas von Mulholland, Keith C, Wallace, William D, Epanomeritakis, Emmanuel, Hall, Stephen R

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Thioester-mediated biocatalytic amide bond synthesis with in situ thiol recycling von Schnepel, Christian, Pérez, Laura Rodríguez, Yu, Yuqi, Angelastro, Antonio, Heath, Rachel S., Lubberink, Max, Falcioni, Francesco, Mulholland, Keith, Hayes, Martin A., Turner, Nicholas J., Flitsch, Sabine L.

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Biocatalytic N-Alkylation of Amines Using Either Primary Alcohols or Carboxylic Acids via Reductive Aminase Cascades von Ramsden, Jeremy I, Heath, Rachel S, Derrington, Sasha R, Montgomery, Sarah L, Mangas-Sanchez, Juan, Mulholland, Keith R, Turner, Nicholas J

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Evaluation of fluoropyruvate as nucleophile in reactions catalysed by N-acetyl neuraminic acid lyase variants: scope, limitations and stereoselectivity von Stockwell, Jennifer, Daniels, Adam D, Windle, Claire L, Harman, Thomas A, Woodhall, Thomas, Lebl, Tomas, Trinh, Chi H, Mulholland, Keith, Pearson, Arwen R, Berry, Alan, Nelson, Adam

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Evaluation of fluoropyruvate as nucleophile in reactions catalysed by N-acetyl neuraminic acid lyase variants: scope, limitations and stereoselectivityElectronic supplementary info... von Stockwell, Jennifer, Daniels, Adam D, Windle, Claire L, Harman, Thomas A, Woodhall, Thomas, Lebl, Tomas, Trinh, Chi H, Mulholland, Keith, Pearson, Arwen R, Berry, Alan, Nelson, Adam

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Evaluation of fluoropyruvate as nucleophile in reactions catalysed by N-acetyl neuraminic acid lyase variants: scope, limitations and stereoselectivity† †Electronic supplementary i... von Stockwell, Jennifer, Daniels, Adam D., Windle, Claire L., Harman, Thomas A., Woodhall, Thomas, Lebl, Tomas, Trinh, Chi H., Mulholland, Keith, Pearson, Arwen R., Berry, Alan, Nelson, Adam

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Feeding the Heck Reaction with Alcohol: One-Pot Synthesis of Stilbenes from Aryl Alcohols and Bromides von Colbon, Paul, Barnard, Jonathan H., Purdie, Mark, Mulholland, Keith, Kozhevnikov, Ivan, Xiao, Jianliang

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Studies into the asymmetric Meisenheimer rearrangement von Buston, Jonathan E.H, Coldham, Iain, Mulholland, Keith R

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Chirality Transfer from Nitrogen to Carbon in the [2,3]-Meisenheimer Rearrangement von Buston, Jonathan E.H., Coldham, Iain, Mulholland, Keith R.

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(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide von Gaster, Laramie M, Jennings, Andrew J, Joiner, Graham F, King, Frank D, Mulholland, Keith R, Rahman, Shirley K, Starr, Susannah, Wyman, Paul A, Wardle, Kay A

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