Applying label-free dynamic mass redistribution technology to frame signaling of G protein–coupled receptors noninvasively in living cells von Schröder, Ralf, Schmidt, Johannes, Blättermann, Stefanie, Peters, Lucas, Janssen, Nicole, Grundmann, Manuel, Seemann, Wiebke, Kaufel, Dorina, Merten, Nicole, Drewke, Christel, Gomeza, Jesus, Milligan, Graeme, Mohr, Klaus, Kostenis, Evi

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Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements von Schröder, Ralf, Janssen, Nicole, Schmidt, Johannes, Kebig, Anna, Merten, Nicole, Hennen, Stephanie, Müller, Anke, Blättermann, Stefanie, Mohr-Andrä, Marion, Zahn, Sabine, Wenzel, Jörg, Smith, Nicola J, Gomeza, Jesús, Drewke, Christel, Milligan, Graeme, Mohr, Klaus, Kostenis, Evi

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The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling von Bock, Andreas, Merten, Nicole, Schrage, Ramona, Dallanoce, Clelia, Bätz, Julia, Klöckner, Jessica, Schmitz, Jens, Matera, Carlo, Simon, Katharina, Kebig, Anna, Peters, Lucas, Müller, Anke, Schrobang-Ley, Jasmin, Tränkle, Christian, Hoffmann, Carsten, De Amici, Marco, Holzgrabe, Ulrike, Kostenis, Evi, Mohr, Klaus

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Rational design of dualsteric GPCR ligands: quests and promise von Mohr, Klaus, Tränkle, Christian, Kostenis, Evi, Barocelli, Elisabetta, De Amici, Marco, Holzgrabe, Ulrike

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Repurposing HAMI3379 to Block GPR17 and Promote Rodent and Human Oligodendrocyte Differentiation von Merten, Nicole, Fischer, Julia, Simon, Katharina, Zhang, Liguo, Schröder, Ralf, Peters, Lucas, Letombe, Anne-Gaelle, Hennen, Stephanie, Schrage, Ramona, Bödefeld, Theresa, Vermeiren, Celine, Gillard, Michel, Mohr, Klaus, Lu, Qing Richard, Brüstle, Oliver, Gomeza, Jesus, Kostenis, Evi

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Dynamic ligand binding dictates partial agonism at a G protein–coupled receptor von Bock, Andreas, Chirinda, Brian, Krebs, Fabian, Messerer, Regina, Bätz, Julia, Muth, Mathias, Dallanoce, Clelia, Klingenthal, Dominika, Tränkle, Christian, Hoffmann, Carsten, De Amici, Marco, Holzgrabe, Ulrike, Kostenis, Evi, Mohr, Klaus

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Rational Design of Partial Agonists for the Muscarinic M1 Acetylcholine Receptor von Chen, Xinyu, Klöckner, Jessika, Holze, Janine, Zimmermann, Cornelia, Seemann, Wiebke K, Schrage, Ramona, Bock, Andreas, Mohr, Klaus, Tränkle, Christian, Holzgrabe, Ulrike, Decker, Michael

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Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity von Antony, Johannes, Kellershohn, Kerstin, Mohr-Andrä, Marion, Kebig, Anna, Prilla, Stefanie, Muth, Mathias, Heller, Eberhard, Disingrini, Teresa, Dallanoce, Clelia, Bertoni, Simona, Schrobang, Jasmin, Tränkle, Christian, Kostenis, Evi, Christopoulos, Arthur, Höltje, Hans-Dieter, Barocelli, Elisabetta, De Amici, Marco, Holzgrabe, Ulrike, Mohr, Klaus

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Hybrid Molecules from Xanomeline and Tacrine: Enhanced Tacrine Actions on Cholinesterases and Muscarinic M1 Receptors von Fang, Lei, Jumpertz, Sabine, Zhang, Yihua, Appenroth, Dorothea, Fleck, Christian, Mohr, Klaus, Tränkle, Christian, Decker, Michael

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Ligand-Specific Allosteric Coupling Controls G‑Protein-Coupled Receptor Signaling von Holze, Janine, Bermudez, Marcel, Pfeil, Eva Marie, Kauk, Michael, Bödefeld, Theresa, Irmen, Matthias, Matera, Carlo, Dallanoce, Clelia, De Amici, Marco, Holzgrabe, Ulrike, König, Gabriele Maria, Tränkle, Christian, Wolber, Gerhard, Schrage, Ramona, Mohr, Klaus, Hoffmann, Carsten, Kostenis, Evi, Bock, Andreas

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Allosteric Small Molecules Unveil a Role of an Extracellular E2/Transmembrane Helix 7 Junction for G Protein-coupled Receptor Activation von Jäger, Dorothea, Schmalenbach, Caroline, Prilla, Stefanie, Schrobang, Jasmin, Kebig, Anna, Sennwitz, Matthias, Heller, Eberhard, Tränkle, Christian, Holzgrabe, Ulrike, Höltje, Hans-Dieter, Mohr, Klaus

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Allosteric Site on Muscarinic Acetylcholine Receptors: Identification of Two Amino Acids in the Muscarinic M2 Receptor That Account Entirely for the M2/M5 Subtype Selectivities of... von Voigtländer, Uta, Jöhren, Kirstin, Mohr, Marion, Raasch, Alexandra, Tränkle, Christian, Buller, Stefan, Ellis, John, Höltje, Hans-Dieter, Mohr, Klaus

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An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators von Kebig, Anna, Kostenis, Evi, Mohr, Klaus, Mohr-Andrä, Marion

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Interactions of Orthosteric and Allosteric Ligands with [3H]Dimethyl-W84 at the Common Allosteric Site of Muscarinic M2 Receptors von Tränkle, Christian, Weyand, Oliver, Voigtländer, Uta, Mynett, Anita, Lazareno, Sebastian, Birdsall, Nigel J. M, Mohr, Klaus

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Allosteric modulators targeting CNS muscarinic receptors von Bock, Andreas, Schrage, Ramona, Mohr, Klaus

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Allosteric Site on Muscarinic Acetylcholine Receptors: A Single Amino Acid in Transmembrane Region 7 Is Critical to the Subtype Selectivities of Caracurine V Derivatives and Alkane... von Buller, Stefan, Zlotos, Darius Paul, Mohr, Klaus, Ellis, John

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Divergent Modes of Action among Cationic Allosteric Modulators of Muscarinic M2 Receptors von Tränkle, Christian, Mohr, Klaus

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Structure−Activity Relationships in a Series of Bisquaternary Bisphthalimidine Derivatives Modulating the Muscarinic M2-Receptor Allosterically von Botero Cid, Hector M, Tränkle, Christian, Baumann, Knut, Pick, Rainer, Mies-Klomfass, Elisabeth, Kostenis, Evi, Mohr, Klaus, Holzgrabe, Ulrike

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Critical Amino Acid Residues of the Common Allosteric Site on the M2 Muscarinic Acetylcholine Receptor: More Similarities than Differences between the Structurally Divergent Agents... von Huang, Xi-Ping, Prilla, Stefanie, Mohr, Klaus, Ellis, John

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Allosteric Interactions with Muscarinic Acetylcholine Receptors: Complex Role of the Conserved Tryptophan M2422Trp in a Critical Cluster of Amino Acids for Baseline Affinity, Subty... von Prilla, Stefanie, Schrobang, Jasmin, Ellis, John, Höltje, Hans-Dieter, Mohr, Klaus

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