Exploitation of silicon medicinal chemistry in drug discovery von Mills, John S, Showell, Graham A

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Neutrophil Formylpeptide Receptor Single Nucleotide Polymorphism 348T>C in Aggressive Periodontitis von Maney, Pooja, Emecen, Pinar, Mills, John S., Walters, John D.

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Trimethylsilylpyrazoles as novel inhibitors of p38 MAP kinase: A new use of silicon bioisosteres in medicinal chemistry von Barnes, Matthew J., Conroy, Richard, Miller, David J., Mills, John S., Montana, John G., Pooni, Parminder K., Showell, Graham A., Walsh, Louise M., Warneck, Julie B.H.

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Donor‐Dependent and Other Nondefined Factors have Greater Influence on the Hepatic Phenotype than the Starting Cell Type in Induced Pluripotent Stem Cell Derived Hepatocyte‐Like Ce... von Heslop, James A., Kia, Richard, Pridgeon, Christopher S., Sison‐Young, Rowena L., Liloglou, Triantafillos, Elmasry, Mohamed, Fenwick, Stephen W., Mills, John S., Kitteringham, Neil R., Goldring, Chris E., Park, B. Kevin

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Chemistry challenges in lead optimization: silicon isosteres in drug discovery von Showell, Graham A, Mills, John S

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Stem cell‐derived hepatocytes as a predictive model for drug‐induced liver injury: are we there yet? von Kia, Richard, Sison, Rowena L. C., Heslop, James, Kitteringham, Neil R., Hanley, Neil, Mills, John S., Park, B. Kevin, Goldring, Chris E. P.

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Rational Design of Peptide-Based HIV Proteinase Inhibitors von Roberts, Noel A., Martin, Joseph A., Kinchington, Derek, Broadhurst, Anne V., Craig, J. Charles, Duncan, Ian B., Galpin, Sarah A., Handa, Balraj K., Kay, John, Kröhn, Antonin, Lambert, Robert W., Merrett, John H., Mills, John S., Kevin E. B. Parkes, Redshaw, Sally, Ritchie, Alison J., Taylor, Debra L., Thomas, Gareth J., Machin, Peter J.

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Functional Epitope on Human Neutrophil Flavocytochrome b558 von Burritt, James B, Foubert, Thomas R, Baniulis, Danas, Lord, Connie I, Taylor, Ross M, Mills, John S, Baughan, Travis D, Roos, Dirk, Parkos, Charles A, Jesaitis, Algirdas J

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Peptides derived from HIV-1, HIV-2, Ebola virus, SARS coronavirus and coronavirus 229E exhibit high affinity binding to the formyl peptide receptor von Mills, John S.

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Donor‐Dependent and Other Nondefined Factors Have Greater Influence on the Hepatic Phenotype Than the Starting Cell Type in Induced Pluripotent Stem Cell Derived Hepatocyte‐Like Ce... von Heslop, James A., Kia, Richard, Pridgeon, Christopher S., Sison‐Young, Rowena L., Liloglou, Triantafillos, Elmasry, Mohamed, Fenwick, Stephen W., Mills, John S., Kitteringham, Neil R., Goldring, Chris E., Park, B. Kevin

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Differential activation of polymorphisms of the formyl peptide receptor by formyl peptides von Mills, John S.

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Sila-venlafaxine, a Sila-Analogue of the Serotonin/Noradrenaline Reuptake Inhibitor Venlafaxine:  Synthesis, Crystal Structure Analysis, and Pharmacological Characterization von Daiss, Jürgen O, Burschka, Christian, Mills, John S, Montana, John G, Showell, Graham A, Warneck, Julie B. H, Tacke, Reinhold

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Synthesis, Crystal Structure Analysis, and Pharmacological Characterization of Disila-bexarotene, a Disila-Analogue of the RXR-Selective Retinoid Agonist Bexarotene von Daiss, Jürgen O, Burschka, Christian, Mills, John S, Montana, John G, Showell, Graham A, Fleming, Ian, Gaudon, Claudine, Ivanova, Diana, Gronemeyer, Hinrich, Tacke, Reinhold

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( R)-Sila-venlafaxine: A selective noradrenaline reuptake inhibitor for the treatment of emesis von Showell, Graham A., Barnes, Matthew J., Daiss, Jürgen O., Mills, John S., Montana, John G., Tacke, Reinhold, Warneck, Julie B.H.

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Silicon Analogues of the Nonpeptidic GnRH Antagonist AG-045572: Syntheses, Crystal Structure Analyses, and Pharmacological Characterization von Barnes, Matthew J., Burschka, Christian, Büttner, Matthias W., Conroy, Richard, Daiss, Jürgen O., Gray, Ian C., Hendrick, Alan G., Tam, L. H., Kuehn, Diana, Miller, David J., Mills, John S., Mitchell, Philip, Montana, John G., Muniandy, Parameswary A., Rapley, Helen, Showell, Graham A., Tebbe, David, Tacke, Reinhold, Warneck, Julie B. H., Zhu, Bin

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Action of ( R)-sila-venlafaxine and reboxetine to antagonize cisplatin-induced acute and delayed emesis in the ferret von Warneck, Julie B., Cheng, Frankie H.M., Barnes, Matthew J., Mills, John S., Montana, John G., Naylor, Robert J., Ngan, Man-P., Wai, Man-K., Daiss, Jürgen O., Tacke, Reinhold, Rudd, John A.

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Variable responses of formyl peptide receptor haplotypes toward bacterial peptides von Gripentrog, Jeannie M, Mills, John S, Saari, George J, Miettinen, Heini M

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Characterization of the Binding Site on the Formyl Peptide Receptor Using Three Receptor Mutants and Analogs of Met-Leu-Phe and Met-Met-Trp-Leu-Leu von Mills, John S., Miettinen, Heini M., Cummings, David, Jesaitis, Algirdas J.

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Mutations of F110 and C126 of the Formyl Peptide Receptor Interfere with G‐Protein Coupling and Chemotaxis von Jones, Barbara E., Miettinen, Heini M., Jesaitis, Algirdas J., Mills, John S.

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Identification of a Ligand Binding Site in the Human Neutrophil Formyl Peptide Receptor Using a Site-specific Fluorescent Photoaffinity Label and Mass Spectrometry von Mills, John S., Miettinen, Heini M., Barnidge, David, Vlases, Michael J., Wimer-Mackin, Susan, Dratz, Edward A., Sunner, Jan, Jesaitis, Algirdas J.

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