Leucettinibs, a Class of DYRK/CLK Kinase Inhibitors Inspired by the Marine Sponge Natural Product Leucettamine B von Deau, Emmanuel, Lindberg, Mattias F., Miege, Frédéric, Roche, Didier, George, Nicolas, George, Pascal, Krämer, Andreas, Knapp, Stefan, Meijer, Laurent

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Chemical, Biochemical, Cellular, and Physiological Characterization of Leucettinib-21, a Down Syndrome and Alzheimer’s Disease Drug Candidate von Lindberg, Mattias F., Deau, Emmanuel, Miege, Frédéric, Greverie, Marie, Roche, Didier, George, Nicolas, George, Pascal, Merlet, Laura, Gavard, Julie, Brugman, Sander J. T., Aret, Edwin, Tinnemans, Paul, de Gelder, René, Sadownik, Jan, Verhofstad, Eva, Sleegers, Dennis, Santangelo, Sara, Dairou, Julien, Fernandez-Blanco, Álvaro, Dierssen, Mara, Krämer, Andreas, Knapp, Stefan, Meijer, Laurent

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Structure–Activity Relationship in the Leucettine Family of Kinase Inhibitors von Tahtouh, Tania, Durieu, Emilie, Villiers, Benoît, Bruyère, Céline, Nguyen, Thu Lan, Fant, Xavier, Ahn, Kwang H, Khurana, Leepakshi, Deau, Emmanuel, Lindberg, Mattias F, Sévère, Elodie, Miege, Frédéric, Roche, Didier, Limanton, Emmanuelle, L’Helgoual’ch, Jean-Martial, Burgy, Guillaume, Guiheneuf, Solène, Herault, Yann, Kendall, Debra A, Carreaux, François, Bazureau, Jean-Pierre, Meijer, Laurent

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Intramolecular Cyclopropanation and C–H Insertion Reactions with Metal Carbenoids Generated from Cyclopropenes von Archambeau, Alexis, Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Synthesis of 3-Oxa- and 3-Azabicyclo[4.1.0]heptanes by Gold-Catalyzed Cycloisomerization of Cyclopropenes von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Rhodium-Catalyzed Cycloisomerization Involving Cyclopropenes: Efficient Stereoselective Synthesis of Medium-Sized Heterocyclic Scaffolds von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Development of ProPhenol Ligands for the Diastereo- and Enantioselective Synthesis of β‑Hydroxy-α-amino Esters von Trost, Barry M, Miege, Frédéric

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Gold(I)-Catalysed Cycloisomerisation of 1,6-Cyclopropene-enes von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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When cyclopropenes meet gold catalysts von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Highly Efficient Stereoselective Catalytic C(sp3)H Insertions with Donor Rhodium Carbenoids Generated from Cyclopropenes von Archambeau, Alexis, Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Ring-Rearrangement Metathesis of Cyclopropenes: Synthesis of Heterocycles von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Rational design, synthesis and pharmacological characterization of novel aminopeptidase A inhibitors von Balavoine, Fabrice, Compere, Delphine, Miege, Frédéric, De Mota, Nadia, Keck, Mathilde, Fer, Mickael, Christen, Aude, Martin, Emmeline, Roche, Didier, Llorens-Cortes, Catherine, Rodeschini, Vincent

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Gold-Catalyzed Rearrangement of (Silylcyclopropenyl)methyl Ethers into (Silylmethylene)cyclopropanes von Hiault, Florence, Archambeau, Alexis, Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Rhodium-Catalyzed Cycloisomerization Involving Cyclopropenes: Efficient Stereoselective Synthesis of Medium-Sized Heterocyclic Scaffolds von Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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Highly Efficient Stereoselective Catalytic C(sp3)H Insertions with Donor Rhodium Carbenoids Generated from Cyclopropenes von Archambeau, Alexis, Miege, Frédéric, Meyer, Christophe, Cossy, Janine

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[1,2,4]-TRIAZOLO[4,3-B]PYRIDAZINE DERIVATIVES USEFUL AS A MEDICAMENT von MIEGE, Frédéric, GEORGE, Pascal, ELIE, Jonathan, MEIJER, Laurent

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IMIDAZOLONE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES IN PARTICULAR DYRK1A, CLK1 AND/OR CLK4 von MIEGE, Frédéric, GEORGE, Pascal, DEAU, Emmanuel, MEIJER, Laurent

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IMIDAZOLONE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES IN PARTICULAR DYRK1A, CLK1 AND/OR CLK4 von MIEGE, Frédéric, GEORGE, Pascal, DEAU, Emmanuel, MEIJER, Laurent

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IMIDAZOLONE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES IN PARTICULAR DYRK1A, CLK1 AND/OR CLK4 von ARCHAMBAUD, Sylvie, MIEGE, Frédéric, GEORGE, Pascal, DEAU, Emmanuel, MEIJER, Laurent

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NOVEL PIPERAZINE-BASED SULFONAMIDES AND THEIR USE AS NEUROPROTECTIVE AND/OR NEURORESTORATIVE AGENTS von MIEGE, Frédéric, CHARVIN, Delphine, MIGNANI, Serge, RIBEILL, Yves, RODESCHINI, Vincent

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