Synthesis and Biological Activities of New Checkpoint Kinase 1 Inhibitors Structurally Related to Granulatimide von Conchon, Elisabeth, Anizon, Fabrice, Aboab, Bettina, Prudhomme, Michelle

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Synthesis, Kinase Inhibitory Potencies, and in Vitro Antiproliferative Evaluation of New Pim Kinase Inhibitors von Akué-Gédu, Rufine, Rossignol, Emilie, Azzaro, Stéphane, Knapp, Stefan, Filippakopoulos, Panagis, Bullock, Alex N, Bain, Jenny, Cohen, Philip, Prudhomme, Michelle, Anizon, Fabrice, Moreau, Pascale

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Pim-selective inhibitor DHPCC-9 reveals Pim kinases as potent stimulators of cancer cell migration and invasion von Santio, Niina M, Vahakoski, Riitta L, Rainio, Eeva-Marja, Sandholm, Jouko A, Virtanen, Sanna S, Prudhomme, Michelle, Anizon, Fabrice, Moreau, Pascale, Koskinen, Päivi J

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Inhibition of Chk1 kills tetraploid tumor cells through a p53-dependent pathway von Vitale, Ilio, Galluzzi, Lorenzo, Vivet, Sonia, Nanty, Lisa, Dessen, Philippe, Senovilla, Laura, Olaussen, Ken A, Lazar, Vladimir, Prudhomme, Michelle, Golsteyn, Roy M, Castedo, Maria, Kroemer, Guido

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Synthesis of aminopyrimidylindoles structurally related to meridianins von Rossignol, Emilie, Youssef, Ali, Moreau, Pascale, Prudhomme, Michelle, Anizon, Fabrice

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Rebeccamycin analogues as anti-cancer agents von Prudhomme, Michelle

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Synthesis, in vitro antiproliferative activities, and Chk1 inhibitory properties of pyrrolo[3,4- a]carbazole-1,3-diones, pyrrolo[3,4- c]carbazole-1,3-diones, and 2-aminopyridazino[... von Conchon, Elisabeth, Anizon, Fabrice, Aboab, Bettina, Golsteyn, Roy M., Léonce, Stéphane, Pfeiffer, Bruno, Prudhomme, Michelle

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Synthesis and antiproliferative activities of indolin-2-one derivatives bearing amino acid moieties von Sassatelli, Mathieu, Debiton, Éric, Aboab, Bettina, Prudhomme, Michelle, Moreau, Pascale

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In-vitro antiproliferative activities and kinase inhibitory potencies of glycosyl-isoindigo derivatives von Sassatelli, Mathieu, Bouchikhi, Fadoua, Aboab, Bettina, Anizon, Fabrice, Fabbro, Doriano, Prudhomme, Michelle, Moreau, Pascale

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Synthesis of dipyrrolo[3,4- a:3,4- c]carbazole-1,3,4,6-tetraones bearing a sugar moiety von Hénon, Hélène, Anizon, Fabrice, Pfeiffer, Bruno, Prudhomme, Michelle

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Rebeccamycin Derivatives as Dual DNA-Damaging Agents and Potent Checkpoint Kinase 1 Inhibitors von Marminon, Christelle, Anizon, Fabrice, Moreau, Pascale, Pfeiffer, Bruno, Pierré, Alain, Golsteyn, Roy M, Peixoto, Paul, Hildebrand, Marie-Paule, David-Cordonnier, Marie-Hélène, Lozach, Olivier, Meijer, Laurent, Prudhomme, Michelle

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Synthesis and biological evaluation of oxindoles and benzimidazolinones derivatives von Messaoudi, Samir, Sancelme, Martine, Polard-Housset, Valérie, Aboab, Bettina, Moreau, Pascale, Prudhomme, Michelle

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Synthesis of pyridino[3′,2′:4,5]pyrrolo[3,2- g]pyrrolo[3,4- e]indolizin-1,3-dione and pyrrolo[3,2- c]pyrazole skeletons von Anizon, Fabrice, Pfeiffer, Bruno, Prudhomme, Michelle

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DNA Cleavage by Topoisomerase I in the Presence of Indolocarbazole Derivatives of Rebeccamycin von Bailly, Christian, Riou, Jean-François, Colson, Pierre, Houssier, Claude, Rodrigues-Pereira, Elisabète, Prudhomme, Michelle

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Structure−Activity Relationships in a Series of Substituted Indolocarbazoles:  Topoisomerase I and Protein Kinase C Inhibition and Antitumoral and Antimicrobial Properties von Rodrigues Pereira, Elisabète, Belin, Laure, Sancelme, Martine, Prudhomme, Michelle, Ollier, Monique, Rapp, Maryse, Sevère, Danièle, Riou, Jean-François, Fabbro, Doriano, Meyer, Thomas

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Enhanced Binding to DNA and Topoisomerase I Inhibition by an Analog of the Antitumor Antibiotic Rebeccamycin Containing an Amino Sugar Residue von Bailly, C, Qu, X, Anizon, F, Prudhomme, M, Riou, J F, Chaires, J B

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Synthesis and biological activities of aminopyrimidyl-indoles structurally related to meridianins von AKUE-GEDU, Rufine, DEBITON, Eric, FERANDIN, Yoan, MEIJER, Laurent, PRUDHOMME, Michelle, ANIZON, Fabrice, MOREAU, Pascale

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Induction of Radiosensitization by Indolocarbazole Derivatives: The Role of DNA Topoisomerase I von Chen, Allan Y, Shih, Shyh-Jen, Hsiao, Michael, Rothenberg, Mace L, Prudhomme, Michelle

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Synthesis of dipyrrolo[3,4-a:3,4-c]carbazoles: new kinase inhibitors von Pereira, Elisabeth, Youssef, Ali, El-Ghozzi, Malika, Avignant, Daniel, Bain, Jennifer, Prudhomme, Michelle, Anizon, Fabrice, Moreau, Pascale

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Recognition of Specific Sequences in DNA by a Topoisomerase I Inhibitor Derived from the Antitumor Drug Rebeccamycin von Bailly, C, Colson, P, Houssier, C, Rodrigues-Pereira, E, Prudhomme, M, Waring, M J

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