Development of a Phase Transfer Catalyzed Asymmetric Synthesis for an Estrogen Receptor Beta Selective Agonist von Scott, Jeremy P, Ashwood, Michael S, Brands, Karel M. J, Brewer, Sarah E, Cowden, Cameron J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Goodyear, Adrian, Oliver, Steven F, Stewart, Gavin W, Wallace, Debra J

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Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction von Zhao, Matthew M, McNamara, James M, Ho, Guo-Jie, Emerson, Khateeta M, Song, Zhiguo J, Tschaen, David M, Brands, Karel M. J, Dolling, Ulf-H, Grabowski, Edward J. J, Reider, Paul J, Cottrell, Ian F, Ashwood, Michael S, Bishop, Brian C

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Stereoselective double ring closing metathesis reactions in the synthesis of spirocyclic compounds von Wallace, Debra J, Cowden, Cameron J, Kennedy, Derek J, Ashwood, Michael S, Cottrell, Ian F, Dolling, Ulf-H

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Efficient One-Pot Synthesis of the 2-Aminocarbonylpyrrolidin-4-ylthio-Containing Side Chain of the New Broad-Spectrum Carbapenem Antibiotic Ertapenem von Brands, Karel M. J, Jobson, Ronald B, Conrad, Karen M, Williams, J. Michael, Pipik, Brenda, Cameron, Mark, Davies, Antony J, Houghton, Peter G, Ashwood, Michael S, Cottrell, Ian F, Reamer, Robert A, Kennedy, Derek J, Dolling, Ulf-H, Reider, Paul J

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Process Development for the Manufacture of a Topical Pan-Trk Inhibitor Incorporating Decarboxylative sp2–sp3 Cross-Coupling von Ashwood, Michael S., Balmond, Edward I., Fengas, David, McGuffog, Jane, Moore, Jonathan, Robas, Nicola M., Stevenson, Neil G., Wise, Lisa

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Process Development for the Manufacture of a Topical Pan-Trk Inhibitor Incorporating Decarboxylative sp 2 –sp 3 Cross-Coupling von Ashwood, Michael S., Balmond, Edward I., Fengas, David, McGuffog, Jane, Moore, Jonathan, Robas, Nicola M., Stevenson, Neil G., Wise, Lisa

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A Double Ring Closing Metathesis Reaction in the Rapid, Enantioselective Synthesis of NK-1 Receptor Antagonists von Wallace, Debra J, Goodman, Jonathan M, Kennedy, Derek J, Davies, Antony J, Cowden, Cameron J, Ashwood, Michael S, Cottrell, Ian F, Dolling, Ulf-H, Reider, Paul J

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Stereocontrolled Preparation of a Nonpeptidal (−)-Spirobicyclic NK-1 Receptor Antagonist von Maligres, Peter E, Waters, Marjorie M, Lee, Jaemoon, Reamer, Robert A, Askin, David, Ashwood, Michael S, Cameron, Mark

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Development of a Scaleable Synthesis of a Partial Nicotinic Acid Receptor Agonist von Wilson, Robert D, Cleator, Ed, Ashwood, Michael S, Bio, Matthew M, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, McKeown, Arlene E, Oliver, Steven F, Reamer, Robert A, Sheen, Faye J, Stewart, Gavin W, Zhou, George X

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Development of a Scaleable Synthesis of a 3-Aminopyrazinone Acetamide Thrombin Inhibitor von Ashwood, Michael S, Alabaster, Ramon J, Cottrell, Ian F, Cowden, Cameron J, Davies, Antony J, Dolling, Ulf H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, Wallace, Debra J, Wilson, Robert D

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Synthesis of the selective muscarinic agonist (3R)-3-(6-chloropyrazin-2-yl)-1-azabicyclo [2.2.2] octane von Ashwood, Michael S., Gibson, Andrew W., Houghton, Peter G., Humphrey, Guy R., Roberts, D. Craig, Wright, Stanley H. B.

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Copper-mediated reaction of 2-halopyridines with ethyl bromodifluoroacetate von Ashwood, Michael S., Cottrell, Ian F., Cowden, Cameron J., Wallace, Debra J., Davies, Antony J., Kennedy, Derek J., Dolling, Ulf H.

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Stereoselective Double Ring Closing Metathesis Reactions in the Synthesis of Spirocyclic Compounds von Wallace, Debra J., Bulger, Paul G., Kennedy, Derek J., Ashwood, Michael S., Cottrell, Ian F., Dolling, Ulf-H.

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A Facile Synthesis of Substituted Phenylglycines von Davies, Antony J., Ashwood, Michael S., Cottrell, Ian F.

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Synthesis of 5,6-dihydro-4H-imidazo[1,5-a][4,1]benzoxazepin-6-ones and their transformation into 5,6-dihydro-4H-imidazo[1,5-a][1,4]benzodiazepin-6-ones von ASHWOOD, M. S, GOURLAY, J. A, HOUGHTON, P. G, NAGEL, M. A, WRIGHT, S. H. B

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Selective Deprotection of Triethylsilyl Group in the Presence of t-Butyldimethylsilyl Group with MCM-41/MeOH Heterogeneous System von Itoh, Akichika, Kodama, Tomohiro, Masaki, Yukio

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Stereoselective synthesis of 2-( S)-(3,5-bis(trifluoromethyl)benzyloxy)-3-( S)-phenyl-1,4-oxazine von Ashwood, Michael S., Cottrell, Ian F., Davies, Antony J.

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Synthesis of 1,1-Diaryl-2,2-dimethoxyethanes von Ashwood, Michael S., Bell, Lawrence A., Houghton, Peter G., Wright, Stanley H. B.

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ChemInform Abstract: A Facile Synthesis of Substituted Phenylglycines von Davies, Antony J., Ashwood, Michael S., Cottrell, Ian F.

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A Practical Synthesis of Lithium 3-Fluoropyridine-2-carboxylate von Emerson, Khateeta M., Wilson, Robert D., Ashwood, Michael S., Kennedy, Derek J., Hands, David, Brands, Karel M. J., Cottrell, Ian F., Dolling, Ulf-H.

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