CYP450 phenotyping and accurate mass identification of metabolites of the 8-aminoquinoline, anti-malarial drug primaquine von Pybus, Brandon S, Sousa, Jason C, Jin, Xiannu, Ferguson, James A, Christian, Robert E, Barnhart, Rebecca, Vuong, Chau, Sciotti, Richard J, Reichard, Gregory A, Kozar, Michael P, Walker, Larry A, Ohrt, Colin, Melendez, Victor

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Nanoparticle formulations of decoquinate increase antimalarial efficacy against liver stage Plasmodium infections in mice von Wang, Hongxing, MD, Li, Qigui, PhD, Reyes, Sean, BSc, Zhang, Jing, BSc, Zeng, Qiang, MSc, Zhang, Ping, BSc, Xie, Lisa, PhD, Lee, Patricia J., BSc, Roncal, Norma, MSc, Melendez, Victor, PhD, Hickman, Mark, PhD, Kozar, Michael P., PhD

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Formulation and Particle Size Reduction Improve Bioavailability of Poorly Water-Soluble Compounds with Antimalarial Activity von Wang, Hongxing, Li, Qigui, Reyes, Sean, Zhang, Jing, Xie, Lisa, Melendez, Victor, Hickman, Mark, Kozar, Michael P.

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In Vitro Metabolism of Phenoxypropoxybiguanide Analogues in Human Liver Microsomes to Potent Antimalarial Dihydrotriazines von Shearer, Todd. W, Kozar, Michael. P, O'Neil, Michael T, Smith, Philip L, Schiehser, Guy A, Jacobus, David. P, Diaz, Damaris S, Yang, Young-Sun, Milhous, Wilbur. K, Skillman, Donald. R

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Antimalarial Activity of Novel 5-Aryl-8-Aminoquinoline Derivatives von Shiraki, Hiroaki, Kozar, Michael P, Melendez, Victor, Hudson, Thomas H, Ohrt, Colin, Magill, Alan J, Lin, Ai J

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Synthesis and Antimalarial Activity of 2-Guanidino-4-oxoimidazoline Derivatives von Liu, Xianjun, Wang, Xihong, Li, Qigui, Kozar, Michael P, Melendez, Victor, O’Neil, Michael T, Lin, Ai J

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Causal Prophylactic Efficacy of Primaquine, Tafenoquine, and Atovaquone-Proguanil Against Plasmodium cynomolgi in a Rhesus Monkey Model von DiTusa, Charles, Kozar, Michael P, Pybus, Brandon, Sousa, Jason, Berman, Jonathan, Gettayacamin, Montip, Im-erbsin, Rawiwan, Tungtaeng, Anchalee, Ohrt, Colin

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Pharmacokinetics, Safety, and Hydrolysis of Oral Pyrroloquinazolinediamines Administered in Single and Multiple Doses in Rats von QIGUI LI, KOZAR, Michael P, SKILLMAN, Donald R, SHEARER, Todd W, XIE, Lisa H, LIN, Ai J, SMITH, Kirsten S, YUANZHENG SI, ANOVA, Lalaine, JING ZHANG, MILHOUS, Wilbur K

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New imidazolidinedione derivatives as antimalarial agents von Zhang, Liang, Sathunuru, Ramadas, Luong, ThuLan, Melendez, Victor, Kozar, Michael P., Lin, Ai J.

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Antimalarial Activities of New Guanidylimidazole and Guanidylimidazoline Derivatives von Zhang, Liang, Sathunuru, Ramadas, Caridha, Diana, Pybus, Brandon, O’Neil, Michael T, Kozar, Michael P, Lin, Ai J

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Muramic Acid Is Not Generally Present in the Human Spleen as Determined by Gas Chromatography-Tandem Mass Spectrometry von KOZAR, Michael P, LAMAN, Jon D, FOX, Alvin

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The use of a prodrug approach to minimize potential CNS exposure of next generation quinoline methanols while maintaining efficacy in in vivo animal models von Sousa, Jason C., Milner, Erin, Carroll, Dustin, McCalmont, William, Gardner, Sean, Moon, Jay, Johnson, Jacob D., Lee, Patricia, Auschwitz, Jennifer, Roncal, Norma, Caridha, Diana, Tungteung, Anchalee, Zeng, Qiang, Reyes, Sean, Smith, Bryan, Li, Qigui, Kozar, Michael P., Melendez, Victor, Dow, Geoffrey

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Malaria Causal Prophylactic Activity of Imidazolidinedione Derivatives von Guan, Jian, Wang, Xihong, Smith, Kirsten, Ager, Arba, Gettayacamin, Montip, Kyle, Dennis E, Milhous, Wilbur K, Kozar, Michael P, Magill, Alan J, Lin, Ai J

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In vitro Biotransformation, in vivo Efficacy and Pharmacokinetics of Antimalarial Chalcones von Gutteridge, Clare E., Thota, Darshan S., Curtis, Sean M., Kozar, Michael P., Li, Qigui, Xie, Lisa, Zhang, Jing, Melendez, Victor, Asher, Constance O., Luong, Thulan T., Gerena, Lucia, Nichols, Daniel A., Montip, Gettayacamin

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Ketotifen is an antimalarial prodrug of norketotifen with blood schizonticidal and liver-stage efficacy von Milner, Erin, Sousa, Jason, Pybus, Brandon, Auschwitz, Jennifer, Caridha, Diana, Gardner, Sean, Grauer, Kristina, Harris, Erin, Hickman, Mark, Kozar, Michael P., Lee, Patricia, Leed, Susan, Li, Qigui, Melendez, Victor, Moon, Jay, Ngundam, Franklyn, O’Neil, Michael, Parriott, Sandi, Potter, Brittney, Sciotti, Rick, Tangteung, Anchalee, Dow, Geoffrey S.

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Analysis of a stable halogenated derivative of muramic acid by gas chromatography–negative ion chemical ionization tandem mass spectrometry von Kozar, Michael P, Fox, Alvin

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Failure To Detect Muramic Acid in Normal Rat Tissues but Detection in Cerebrospinal Fluids from Patients with Pneumococcal Meningitis von KOZAR, M. P, KRAHMER, M. T, FOX, A, GRAY, B. M

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Trace analysis of muramic acid in indoor air using an automated derivatization instrument and GC-MS(2) or GC-MS(3) von Harley, William M, Kozar, Michael P, Fox, Alvin

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Trace analysis of muramic acid in indoor air using an automated derivatization instrument and GC-MS2 or GC-MS3 von HARLEY, William M, KOZAR, Michael P, FOX, Alvin

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Lunar dust: a negative control for biomarker analyses of extraterrestrial samples? von Kozar, Michael P, Krahmer, Mark T, Fox, Alvin, Larsson, Lennart, Allton, Judith

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