Evaluation of Kilogram-Scale Sonagashira, Suzuki, and Heck Coupling Routes to Oncology Candidate CP-724,714 von Ripin, David H. Brown, Bourassa, Dennis E, Brandt, Thomas, Castaldi, Michael J, Frost, Heather N, Hawkins, Joel, Johnson, Phillip J, Massett, Stephen S, Neumann, Karin, Phillips, James, Raggon, Jeffery W, Rose, Peter R, Rutherford, Jennifer L, Sitter, Barbara, Stewart, A. Morgan, Vetelino, Michael G, Wei, Lulin

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An Efficient and Cost-Effective Synthesis of 2-Phenyl-3-aminopyridine von Caron, Stéphane, Massett, Steve S., Bogle, David E., Castaldi, Michael J., Braish, Tamim F.

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Case Study of a γ-Butyrolactone Alkylation with 1,3-Dimethyl-2-imidazolidinone as a Promoter von Li, Bryan, Buzon, Richard A, Castaldi, Michael J

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Safety vs Efficiency in the Development of a High-Energy Compound von Ruggeri, Sally Gut, Bill, David R, Bourassa, Dennis E, Castaldi, Michael J, Houck, Tim L, Ripin, David H. Brown, Wei, Lulin, Weston, Neil

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Synthesis and Purification of 6-Ethoxy-4-oxo-1,4-dihydro-[1,5]naphthyridine-3-carboxylic Acid Benzylamide von Beaudin, Justin, Bourassa, Dennis E, Bowles, Paul, Castaldi, Michael J, Clay, Ronald, Couturier, Michel A, Karrick, Gregory, Makowski, Teresa W, McDermott, Ruth E, Meltz, Clifford N, Meltz, Morgan, Phillips, James E, Ragan, John A, Ripin, David H. Brown, Singer, Robert A, Tucker, John L, Wei, Lulin

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Investigation of Methods for Seven-Membered Ring Synthesis:  A Practical Synthesis of 4-Oxo-5,6,7,8-tetrahydro-4H-cyclohepta[b]furan-3-carboxylic Acid von Ragan, John A, Murry, Jerry A, Castaldi, Michael J, Conrad, Alyson K, Jones, Brian P, Li, Bryan, Makowski, Teresa W, McDermott, Ruth, Sitter, Barb J, White, Timothy D, Young, Gregory R

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3-Quinolinecarboxamides. A series of novel orally-active antiherpetic agents von Wentland, Mark P, Perni, Robert B, Dorff, Peter H, Brundage, R. Pauline, Castaldi, Michael J, Bailey, Thomas R, Carabateas, Philip M, Bacon, Edward R, Young, Dorothy C

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Synthesis of (1α,5α,6α)-6-Amino-3-azabicyclo[3.1.0]hexane, a Novel Achiral Diamine von Brighty, Katherine E., Castaldi, Michael J.

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Synthesis and antidepressant properties of novel 2-substituted 4,5-dihydro-1H-imidazole derivatives von Wentland, Mark P, Bailey, Denis M, Alexander, E. John, Castaldi, Michael J, Ferrari, Richard A, Haubrich, Dean R, Luttinger, Daniel A, Perrone, Mark H

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2,5-Dimethylpyrrole Protection Facilitates Copper(I)-Mediated Methoxylations of Aryl Iodides in the Presence of Anilines von Ragan, John A., Makowski, Teresa W., Castaldi, Michael J., Hill, Paul D.

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In vitro activity of CP-99,219, a novel 7-(3-azabicyclo[3.1.0]hexyl) naphthyridone antimicrobial von D. Gootz, Thomas, Brighty, Katherine E., Anderson, Marge R., Schmieder, Brenda J., Haskell, Suzanne L., Sutcliffe, Joyce A., Castaldi, Michael J., McGuirk, Paul R.

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ULLMAN METHOXYLATION IN THE PRESENCE OF A 2,5-DIMETHYLPYRROLE-BLOCKED ANILINE: PREPARATION OF 2-FLUORO-4-METHOXYANILINE

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Crystalline anhydrous and monohydrate benzoate salts of (2'S,3S)-3-hydroxy-N-{2-[N-methyl-N-4-(N-propylamino-carbonyl)phenyl]amino-2-phenyl}-ethylpyrrolidine von CASTALDI MICHAEL J, QUALLICH GEORGE

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Crystalline anhydrous and monohydrate benzoate salts of (2'S,3S)-3-hydroxy-N-(2-[N-methyl-N-4-(N-propylamino-carbonyl)phenyl]amino-2-phenyl)-ethylpyrrolidine von QUALLICH GEORGE J, CASTALDI MICHAEL J

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Crystalline anhydrous and monohydrate benzoate salts of (2′S,3S)-3-hydroxy-N-(2-[N-methyl-N-4-(N-propylamino-carbonyl)phenyl]amino-2-phenyl)-ethylpyrrolidine von Quallich, George J, Castaldi, Michael J

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Scalable Process for 4-(2-Hydroxy-2-methyl)-ethyl-benzylamine von Tucker, John L., Couturier, Michel, Castaldi, Michael J., Chiu, Charles K. F., Gestmann, Detlef

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Process for preparing 2-phenyl-3-aminopyridine, substituted phenyl derivatives thereof, and salts thereof von BRAISH, TAMIM F, CASTALDI, MICHAEL J, CARON, STEPHANE

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Polymorphs of a crystalline azabicyclo[2,2.2]octan-3-amine citrate and their pharmaceutical compositions von CASTALDI, MICHAEL J, QUALLICH, GEORGE JOSEPH, WINT, LEWIN THEOPHILUS

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Processes for the Preparation of Benzoimidazole Derivatives von RIPIN DAVID B, TOM NORMA J, CASTALDI MICHAEL J

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Processes for the preparation of benzoimidazole derivatives von Tom, Norma J, Castaldi, Michael J, Ripin, David B

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