Discovery of Novel Chemotypes to a G-Protein-Coupled Receptor through Ligand-Steered Homology Modeling and Structure-Based Virtual Screening von Cavasotto, Claudio N, Orry, Andrew J. W, Murgolo, Nicholas J, Czarniecki, Michael F, Kocsi, Sue Ann, Hawes, Brian E, O’Neill, Kim A, Hine, Heather, Burton, Marybeth S, Voigt, Johannes H, Abagyan, Ruben A, Bayne, Marvin L, Monsma, Frederick J

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Structure based design of iminohydantoin BACE1 inhibitors: Identification of an orally available, centrally active BACE1 inhibitor von Cumming, Jared N., Smith, Elizabeth M., Wang, Lingyan, Misiaszek, Jeffrey, Durkin, James, Pan, Jianping, Iserloh, Ulrich, Wu, Yusheng, Zhu, Zhaoning, Strickland, Corey, Voigt, Johannes, Chen, Xia, Kennedy, Matthew E., Kuvelkar, Reshma, Hyde, Lynn A., Cox, Kathleen, Favreau, Leonard, Czarniecki, Michael F., Greenlee, William J., McKittrick, Brian A., Parker, Eric M., Stamford, Andrew W.

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Synthesis and structure–activity relationships of new disubstituted phenyl-containing 3,4-diamino-3-cyclobutene-1,2-diones as CXCR2 receptor antagonists von Lai, Gaifa, Merritt, J. Robert, He, Zhenmin, Feng, Daming, Chao, Jianhua, Czarniecki, Michael F., Rokosz, Laura L., Stauffer, Tara M., Rindgen, Diane, Taveras, Arthur G.

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Carbon-13 nuclear magnetic resonance spin-lattice relaxation in the N-acylneuraminic acids. Probes for internal dynamics and conformational analysis von Czarniecki, Michael F, Thornton, Edward R

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Very Fast acylation of .beta.-cyclodextrin by bound p-nitrophenyl ferrocinnamate von Czarniecki, Michael F, Breslow, Ronald

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Photochemical probes for model membrane structures von Czarniecki, Michael F, Breslow, Ronald

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Carbon-13 nuclear magnetic resonance of ganglioside sugars. Spin-lattice relaxation probes for structure and microdynamics of cell surface carbohydrates von Czarniecki, Michael F, Thornton, Edward R

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Improved acylation rates within cyclodextrin complexes from flexible capping of the cyclodextrin and from adjustment of the substrate geometry von Breslow, Ronald, Czarniecki, Michael F, Emert, Jack, Hamaguchi, Hiroshi

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Carbon-13 spin lattice relaxation in the neuraminic acids. Evidence for an unusual intramolecular hydrogen bonding network von Czarniecki, Michael F, Thornton, Edward R

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5476847 Derivatives of phosphinic acid useful as endothelin converting enzyme inhibitors : McKittrick Brian A; Czarniecki Michael F; Chackalamannil Samuel; Chung Shin; DeFrees Shaw; Stamford Andrew W Bloomfield, NJ, United States assigned to Schering Corporation

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13C NMR chemical shift titration of metal ion-carbohydrate complexes. An unexpected dichotomy for Ca +2 binding between anomeric derivatives of N-Acetylneuraminic acid (1) von Czarniecki, Michael F., Thornton, Edward R.

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TRIAZOLOPYRAZINONES AS P2X7 RECEPTOR ANTAGONISTS von CZARNIECKI, MICHAEL, F, POKER, CORY SETH, LABROLI, MARC

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TRIAZOLOPYRAZINONES AS P2X7 RECEPTOR ANTAGONISTS von POKER CORY SETH, LABROLI MARC, CZARNIECKI MICHAEL F

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DERIVATIVES OF 7,8-DIHYDRO-1H-IMIDAZO[2,1-b] PURIN-4(5H)-ONE and METHODS OF USE THEREOF von MATASI JULIUS, TULSHIAN DEEN, CZARNIECKI MICHAEL F, BRUMFIELD STEPHANIE N

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TRIAZOLOPYRAZINONES AS P2X7 RECEPTOR ANTAGONISTS von CZARNIECKI, MICHAEL, F, POKER, CORY SETH, LABROLI, MARC

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TRIAZOLOPYRAZINONES AS P2X7 RECEPTOR ANTAGONISTS von CZARNIECKI, MICHAEL, F, POKER, CORY SETH, LABROLI, MARC

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TRIAZOLOPYRAZINONES AS P2X7 RECEPTOR ANTAGONISTS von CZARNIECKI, MICHAEL, F, POKER, CORY SETH, LABROLI, MARC

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DERIVATIVES OF 7,8-DIHYDRO-1H-IMIDAZO[2,1-b]PURIN-4(5H)-ONE AND METHODS OF USE THEREOF von TULSHIAN, DEEN, MATASI, JULIUS, J, BRUMFIELD, STEPHANIE NICOLE, CZARNIECKI, MICHAEL, F

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DERIVATIVES OF 7,8-DIHYDRO-1H-IMIDAZO[2,1-b]PURIN-4(5H)-ONE AND METHODS OF USE THEREOF von TULSHIAN, DEEN, MATASI, JULIUS, J, BRUMFIELD, STEPHANIE NICOLE, CZARNIECKI, MICHAEL, F

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DERIVADOS DE GUANINA POLICÍCLICA E MÉTODOS DE USO DOS MESMOS von WILLAIM B. GEISS, MICHAEL F. CZARNIECKI, JULIUS J. MATASI, VAN-DUC LE, JAMES C. HABER, STEPHANIE NICOLE COOKE, DEEN TULSHIAN, GREGORY S. MARTIN

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