Small-Molecule Inhibition of the Interaction between the Translation Initiation Factors eIF4E and eIF4G von Moerke, Nathan J., Aktas, Huseyin, Chen, Han, Cantel, Sonia, Reibarkh, Mikhail Y., Fahmy, Amr, Gross, John D., Degterev, Alexei, Yuan, Junying, Chorev, Michael, Halperin, Jose A., Wagner, Gerhard

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The partial retro-inverso modification: A road traveled together von Chorev, Michael

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Plasma Glycated CD59, a Novel Biomarker for Detection of Pregnancy-Induced Glucose Intolerance von Ghosh, Pamela, Luque-Fernandez, Miguel A, Vaidya, Anand, Ma, Dongdong, Sahoo, Rupam, Chorev, Michael, Zera, Chloe, McElrath, Thomas F, Williams, Michelle A, Seely, Ellen W, Halperin, Jose A

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Structure of the eukaryotic translation initiation factor eIF4E in complex with 4EGI-1 reveals an allosteric mechanism for dissociating eIF4G von Papadopoulos, Evangelos, Jenni, Simon, Kabha, Eihab, Takrouri, Khuloud J, Yi, Tingfang, Salvi, Nicola, Luna, Rafael E, Gavathiotis, Evripidis, Mahalingam, Poornachandran, Arthanari, Haribabu, Rodriguez-Mias, Ricard, Yefidoff-Freedman, Revital, Aktas, Bertal H, Chorev, Michael, Halperin, Jose A, Wagner, Gerhard

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Glycation of the Complement Regulatory Protein CD59 Is a Novel Biomarker for Glucose Handling in Humans von Ghosh, Pamela, Vaidya, Anand, Sahoo, Rupam, Goldfine, Allison, Herring, Neil, Bry, Lynn, Chorev, Michael, Halperin, Jose A

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Design, synthesis, conformational analysis, and biological activity of Cα1-to-Cα6 1,4- and 4,1-disubstituted 1H-[1,2,3]triazol-1-yl-bridged oxytocin analogues von Nuti, Francesca, Larregola, Maud, Staśkiewicz, Agnieszka, Retzl, Bernhard, Tomašević, Nataša, Macchia, Lorenzo, Street, Maria E, Jewgiński, Michał, Lequin, Olivier, Latajka, Rafal, Rovero, Paolo, Gruber, Christian W, Chorev, Michael, Papini, Anna Maria

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Synthesis and Conformational Analysis of a Cyclic Peptide Obtained via i to i+4 Intramolecular Side-Chain to Side-Chain Azide−Alkyne 1,3-Dipolar Cycloaddition von Cantel, Sonia, Le Chevalier Isaad, Alexandra, Scrima, Mario, Levy, Jay J, DiMarchi, Richard D, Rovero, Paolo, Halperin, Jose A, D’Ursi, Anna Maria, Papini, Anna Maria, Chorev, Michael

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Human CD59 Inhibitor Sensitizes Rituximab-Resistant Lymphoma Cells to Complement-Mediated Cytolysis von WEIGUO HU, XIAOWEN GE, BROWN, Jennifer R, XUEBIN QIN, TAO YOU, TING XU, JINYAN ZHANG, GONGXIONG WU, ZHIHAI PENG, CHOREV, Michael, AKTAS, Bertal H, HALPERIN, Jose A

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Inhibition of the interactions between eukaryotic initiation factors 4E and 4G impairs long-term associative memory consolidation but not reconsolidation von Hoeffer, Charles A, Cowansage, Kiriana K, Arnold, Elizabeth C, Banko, Jessica L, Moerke, Nathan J, Rodriguez, Ricard, Schmidt, Enrico K, Klosi, Edvin, Chorev, Michael, Lloyd, Richard E, Pierre, Philippe, Wagner, Gerhard, LeDoux, Joseph E, Klann, Eric

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Explorations of Substituted Urea Functionality for the Discovery of New Activators of the Heme-Regulated Inhibitor Kinase von Chen, Ting, Takrouri, Khuloud, Hee-Hwang, Sung, Rana, Sandeep, Yefidoff-Freedman, Revital, Halperin, Jose, Natarajan, Amarnath, Morisseau, Christophe, Hammock, Bruce, Chorev, Michael, Aktas, Bertal H

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Activity of the Di-Substituted Urea-Derived Compound I-17 in Leishmania In Vitro Infections von Dos Santos, José Vitorino, Medina, Jorge Mansur, Dias Teixeira, Karina Luiza, Agostinho, Daniel Marcos Julio, Chorev, Michael, Diotallevi, Aurora, Galluzzi, Luca, Aktas, Bertal Huseyin, Gazos Lopes, Ulisses

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Parathyroid hormone 1–34 enhances titanium implant anchorage in low-density trabecular bone: A correlative micro-computed tomographic and biomechanical analysis von Gabet, Yankel, Müller, Ralph, Levy, Jay, Dimarchi, Richard, Chorev, Michael, Bab, Itai, Kohavi, David

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A specific and sensitive assay for blood levels of glycated CD59: A novel biomarker for diabetes von Ghosh, Pamela, Sahoo, Rupam, Vaidya, Anand, Cantel, Sonia, Kavishwar, Amol, Goldfine, Allison, Herring, Neil, Bry, Lynn, Chorev, Michael, Halperin, Jose A.

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Structure–activity relationship study of 4EGI-1, small molecule eIF4E/eIF4G protein–protein interaction inhibitors von Takrouri, Khuloud, Chen, Ting, Papadopoulos, Evangelos, Sahoo, Rupam, Kabha, Eihab, Chen, Han, Cantel, Sonia, Wagner, Gerhard, Halperin, Jose A., Aktas, Bertal H., Chorev, Michael

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Novel Dual Inhibitors of AChE and MAO Derived from Hydroxy Aminoindan and Phenethylamine as Potential Treatment for Alzheimer's Disease von Sterling, Jeffrey, Herzig, Yaacov, Goren, Tamar, Finkelstein, Nina, Lerner, David, Goldenberg, Willy, Miskolczi, Istvan, Molnar, Sandor, Rantal, Ferenc, Tamas, Tivadar, Toth, Gyorgy, Zagyva, Adela, Zekany, Andras, Lavian, Gila, Gross, Aviva, Friedman, Rachel, Razin, Michal, Huang, Wei, Krais, Boris, Chorev, Michael, Youdim, Moussa B, Weinstock, Marta

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Dual Activators of Protein Kinase R (PKR) and Protein Kinase R-Like Kinase (PERK) Identify Common and Divergent Catalytic Targets von Bai, Huijun, Chen, Ting, Ming, Jie, Sun, Hong, Cao, Peng, Fusco, Dahlene N., Chung, Raymond T., Chorev, Michael, Jin, Qi, Aktas, Bertal H.

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Osteogenic growth peptide modulates fracture callus structural and mechanical properties von Gabet, Yankel, Müller, Ralph, Regev, Eran, Sela, Jona, Shteyer, Arie, Salisbury, Kristy, Chorev, Michael, Bab, Itai

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Role of Complement and Complement Regulatory Proteins in the Complications of Diabetes von Ghosh, Pamela, Sahoo, Rupam, Vaidya, Anand, Chorev, Michael, Halperin, Jose A

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Selective Ligand-induced Stabilization of Active and Desensitized Parathyroid Hormone Type 1 Receptor Conformations von Bisello, Alessandro, Chorev, Michael, Rosenblatt, Michael, Monticelli, Luca, Mierke, Dale F., Ferrari, Serge L.

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The Mid-Region of Parathyroid Hormone (1−34) Serves as a Functional Docking Domain in Receptor Activation von Wittelsberger, Angela, Corich, Martina, Thomas, Beena E, Lee, Byung-Kwon, Barazza, Alessandra, Czodrowski, Paul, Mierke, Dale F, Chorev, Michael, Rosenblatt, Michael

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