Carbohydrates as Scaffolds in Drug Discovery von Meutermans, Wim, Le, Giang Thanh, Becker, Bernd

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Fragment-based drug discovery for disorders of the central nervous system: designing better drugs piece by piece von Chan, Bill W G L, Lynch, Nicholas B, Tran, Wendy, Joyce, Jack M, Savage, G Paul, Meutermans, Wim, Montgomery, Andrew P, Kassiou, Michael

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Difficult Macrocyclizations:  New Strategies for Synthesizing Highly Strained Cyclic Tetrapeptides von Meutermans, Wim D. F, Bourne, Gregory T, Golding, Simon W, Horton, Douglas A, Campitelli, Marc R, Craik, David, Scanlon, Martin, Smythe, Mark L

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Synthesis of Difficult Cyclic Peptides by Inclusion of a Novel Photolabile Auxiliary in a Ring Contraction Strategy von Meutermans, Wim D. F, Golding, Simon W, Bourne, Greg T, Miranda, Les P, Dooley, Michael J, Alewood, Paul F, Smythe, Mark L

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An Activated O → N Acyl Transfer Auxiliary:  Efficient Amide-Backbone Substitution of Hindered “Difficult” Peptides von Miranda, Les P, Meutermans, Wim D. F, Smythe, Mark L, Alewood, Paul F

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A Backbone Linker for BOC-Based Peptide Synthesis and On-Resin Cyclization:  Synthesis of Stylostatin 1 von Bourne, Gregory T, Meutermans, Wim D. F, Alewood, Paul F, McGeary, Ross P, Scanlon, Martin, Watson, Andrew A, Smythe, Mark L

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In vitro profiling of opioid ligands using the cAMP formation inhibition assay and the β-arrestin2 recruitment assay: No two ligands have the same profile von Kuo, Andy, Magiera, Julia, Rethwan, Nursyazwani, Andersson, Åsa, Leen Lam, Ai, Wyse, Bruce, Meutermans, Wim, Lewis, Richard, Smith, Maree

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Topological side-chain classification of beta-turns: ideal motifs for peptidomimetic development von Tran, Tran Trung, McKie, Jim, Meutermans, Wim D F, Bourne, Gregory T, Andrews, Peter R, Smythe, Mark L

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Targeting the forgotten transglycosylases von Halliday, Judy, McKeveney, Declan, Muldoon, Craig, Rajaratnam, Premraj, Meutermans, Wim

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Fighting Obesity with a Sugar-Based Library: Discovery of Novel MCH-1R Antagonists by a New Computational–VAST Approach for Exploration of GPCR Binding Sites von Heifetz, Alexander, Barker, Oliver, Verquin, Geraldine, Wimmer, Norbert, Meutermans, Wim, Pal, Sandeep, Law, Richard J, Whittaker, Mark

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Carbohydrate scaffolds as glycosyltransferase inhibitors with in vivo antibacterial activity von Zuegg, Johannes, Muldoon, Craig, Adamson, George, McKeveney, Declan, Le Thanh, Giang, Premraj, Rajaratnam, Becker, Bernd, Cheng, Mu, Elliott, Alysha G., Huang, Johnny X., Butler, Mark S., Bajaj, Megha, Seifert, Joachim, Singh, Latika, Galley, Nicola F., Roper, David I., Lloyd, Adrian J., Dowson, Christopher G., Cheng, Ting-Jen, Cheng, Wei-Chieh, Demon, Dieter, Meyer, Evelyne, Meutermans, Wim, Cooper, Matthew A.

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Targeting Bacterial Cell Wall Peptidoglycan Synthesis by Inhibition of Glycosyltransferase Activity von Mesleh, Michael F., Rajaratnam, Premraj, Conrad, Mary, Chandrasekaran, Vasu, Liu, Christopher M., Pandya, Bhaumik A., Hwang, You Seok, Rye, Peter T., Muldoon, Craig, Becker, Bernd, Zuegg, Johannes, Meutermans, Wim, Moy, Terence I.

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Solid-Phase Oligosaccharide Chemistry and Its Application to Library Synthesis von Grathwohl, Matthias, Drinnan, Nicholas, Broadhurst, Max, West, Michael L, Meutermans, Wim

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p-Cresol As a Reversible Acylium Ion Scavenger in Solid-Phase Peptide Synthesis von Miranda, Les P, Jones, Alun, Meutermans, Wim D. F, Alewood, Paul F

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Crystal Structures of the PBP2 Glycosyltransferase Domain: New Opportunities for Antibacterial Drug Design von Zuegg, Johannes, Meutermans, Wim

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The Development and Application of a Novel Safety-Catch Linker for BOC-Based Assembly of Libraries of Cyclic Peptides ‖ ,1 von Bourne, Gregory T, Golding, Simon W, McGeary, Ross P, Meutermans, Wim D. F, Jones, Alun, Marshall, Garland R, Alewood, Paul F, Smythe, Mark L

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Toward Larger Chemical Libraries:  Encoding with Fluorescent Colloids in Combinatorial Chemistry von Battersby, Bronwyn J, Bryant, Darryn, Meutermans, Wim, Matthews, Daniel, Smythe, Mark L, Trau, Matt

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A simple and effective procedure for the synthesis of the ‘difficult’ phosphotyrosine-containing peptide stat 91 (695–708) von Meutermans, Wim D.F, Alewood, Paul F

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Molecular diversity through sugar scaffolds von Thanh Le, Giang, Abbenante, Giovanni, Becker, Bernd, Grathwohl, Matthias, Halliday, Judy, Tometzki, Gerry, Zuegg, Johannes, Meutermans, Wim

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Biological Diversity from a Structurally Diverse Library: Systematically Scanning Conformational Space Using a Pyranose Scaffold von Abbenante, Giovanni, Becker, Bernd, Blanc, Sébastien, Clark, Chris, Condie, Glenn, Fraser, Graeme, Grathwohl, Matthias, Halliday, Judy, Henderson, Senka, Lam, Ann, Liu, Ligong, Mann, Maretta, Muldoon, Craig, Pearson, Andrew, Premraj, Rajaratnam, Ramsdale, Tracie, Rossetti, Tony, Schafer, Karl, Le Thanh, Giang, Tometzki, Gerald, Vari, Frank, Verquin, Géraldine, Waanders, Jennifer, West, Michael, Wimmer, Norbert, Yau, Annika, Zuegg, Johannes, Meutermans, Wim

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