Discovery of AZD-2098 and AZD-1678, Two Potent and Bioavailable CCR4 Receptor Antagonists von Kindon, Nicholas, Andrews, Glen, Baxter, Andrew, Cheshire, David, Hemsley, Paul, Johnson, Timothy, Liu, Yu-Zhen, McGinnity, Dermot, McHale, Mark, Mete, Antonio, Reuberson, James, Roberts, Bryan, Steele, John, Teobald, Barry, Unitt, John, Vaughan, Deborah, Walters, Iain, Stocks, Michael J

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discovery of AZD9164, a novel muscarinic M₃ antagonist von Mete, Antonio, Bowers, Keith, Chevalier, Eric, Donald, David K, Edwards, Helen, Escott, Katherine J, Ford, Rhonan, Grime, Ken, Millichip, Ian, Teobald, Barry, Russell, Vince

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Design and Synthesis of a Novel and Potent Series of Inhibitors of Cytosolic Phospholipase A2 Based on a 1,3-Disubstituted Propan-2-one Skeleton von Connolly, Stephen, Bennion, Colin, Botterell, Sarah, Croshaw, Pamela J, Hallam, Catherine, Hardy, Kim, Hartopp, Paul, Jackson, Clive G, King, Sarah J, Lawrence, Louise, Mete, Antonio, Murray, David, Robinson, David H, Smith, Gillian M, Stein, Linda, Walters, Iain, Wells, Edward, Withnall, W. John

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The relative rate of kill of the MMV Malaria Box compounds provides links to the mode of antimalarial action and highlights scaffolds of medicinal chemistry interest von Ullah, Imran, Sharma, Raman, Mete, Antonio, Biagini, Giancarlo A, Wetzel, Dawn M, Horrocks, Paul D

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Addressing the Intracellular Vestibule of the Plasmodial Lactate Transporter PfFNT by p‑Substituted Inhibitors Amplifies In Vitro Activity von Nerlich, Cornelius, Tiedjens, Finn, Hertel, Robin, Henke, Björn, Häuer, Susan, Panitzsch, Lea S., Hansen, Kerrin, Franck, Ole, Mete, Antonio, Leroy, Didier, Schade, Dennis, Peifer, Christian, Hannus, Stefan, Becker, Frank, Wittlin, Sergio, Spielmann, Tobias, Beitz, Eric

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Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase von Garcin, Elsa D, Getzoff, Elizabeth D, Arvai, Andrew S, Rosenfeld, Robin J, Kroeger, Matt D, Crane, Brian R, Andersson, Gunilla, Andrews, Glen, Hamley, Peter J, Mallinder, Philip R, Nicholls, David J, St-Gallay, Stephen A, Tinker, Alan C, Gensmantel, Nigel P, Mete, Antonio, Cheshire, David R, Connolly, Stephen, Stuehr, Dennis J, Åberg, Anders, Wallace, Alan V, Tainer, John A

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Cathepsin C Inhibitors: Property Optimization and Identification of a Clinical Candidate von Furber, Mark, Tiden, Anna-Karin, Gardiner, Philip, Mete, Antonio, Ford, Rhonan, Millichip, Ian, Stein, Linda, Mather, Andrew, Kinchin, Elizabeth, Luckhurst, Christopher, Barber, Simon, Cage, Peter, Sanganee, Hitesh, Austin, Rupert, Chohan, Kamaldeep, Beri, Raj, Thong, Bob, Wallace, Alan, Oreffo, Victor, Hutchinson, Ray, Harper, Steve, Debreczeni, Judit, Breed, Jason, Wissler, Lisa, Edman, Karl

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The discovery of AZD9164, a novel muscarinic M 3 antagonist von Mete, Antonio, Bowers, Keith, Chevalier, Eric, Donald, David K., Edwards, Helen, Escott, Katherine J., Ford, Rhonan, Grime, Ken, Millichip, Ian, Teobald, Barry, Russell, Vince

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Potassium channel inhibitors von Sørensen, Ulrik, Mete, Antonio

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The design of a novel series of muscarinic receptor antagonists leading to AZD8683, a potential inhaled treatment for COPD von Mete, Antonio, Bowers, Keith, Bull, Richard J., Coope, Helen, Donald, David K., Escott, Katherine J., Ford, Rhonan, Grime, Ken, Mather, Andrew, Ray, Nicholas C., Russell, Vince

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Potassium channel inhibitors von Sørensen, Ulrik, Mete, Antonio

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NOVEL POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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NOVEL POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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NOVEL POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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IMIDAZOLE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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IMIDAZOLE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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Asymmetric synthesis of azidotetrahydropyranols via Sharpless epoxidation von Ong, Quyen, Handa, Sheetal, Mete, Antonio, Hill, Alison M., Jones, Keith

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NOVEL POTASSIUM CHANNEL INHIBITORS von METE, ANTONIO, SORENSEN, ULRIK

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NOVEL POTASSIUM CHANNEL INHIBITORS von METE, Antonio, SØRENSEN, Ulrik

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The discovery of novel, potent and highly selective inhibitors of inducible nitric oxide synthase (iNOS) von Cheshire, David R., Åberg, Anders, Andersson, Gunilla M.K., Andrews, Glen, Beaton, Haydn G., Birkinshaw, Timothy N., Boughton-Smith, Nigel, Connolly, Stephen, Cook, Tony R., Cooper, Anne, Cooper, Sally L., Cox, David, Dixon, John, Gensmantel, Nigel, Hamley, Peter J., Harrison, Richard, Hartopp, Paul, Käck, Helena, Leeson, Paul D., Luker, Timothy, Mete, Antonio, Millichip, Ian, Nicholls, David J., Pimm, Austen D., St-Gallay, Steve A., Wallace, Alan V.

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