Small molecule chemokine mimetics suggest a molecular basis for the observation that CXCL10 and CXCL11 are allosteric ligands of CXCR3 von Nedjai, Belinda, Li, Hubert, Stroke, Ilana L, Wise, Emma L, Webb, Maria L, Merritt, J Robert, Henderson, Ian, Klon, Anthony E, Cole, Andrew G, Horuk, Richard, Vaidehi, Nagarajan, Pease, James E

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Discovery of 2-Hydroxy-N,N-dimethyl-3-{2-[[(R)-1-(5- methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobut-1-enylamino}benzamide (SCH 527123):  A Potent, Orally Bioavailable CXCR2/CXCR1... von Dwyer, Michael P, Yu, Younong, Chao, Jianping, Aki, Cynthia, Chao, Jianhua, Biju, Purakkattle, Girijavallabhan, Viyyoor, Rindgen, Diane, Bond, Richard, Mayer-Ezel, Rosemary, Jakway, James, Hipkin, R. William, Fossetta, James, Gonsiorek, Waldemar, Bian, Hong, Fan, Xuedong, Terminelli, Carol, Fine, Jay, Lundell, Daniel, Merritt, J. Robert, Rokosz, Laura L, Kaiser, Bernd, Li, Ge, Wang, Wei, Stauffer, Tara, Ozgur, Lynne, Baldwin, John, Taveras, Arthur G

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Identification of CXCR3 receptor agonists in combinatorial small-molecule libraries von Stroke, Ilana L., Cole, Andrew G., Simhadri, Srilatha, Brescia, Marc-Raleigh, Desai, Madhuri, Zhang, Joan J., Merritt, J. Robert, Appell, Kenneth C., Henderson, Ian, Webb, Maria L.

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3,4-Diamino-2,5-thiadiazole-1-oxides as potent CXCR2/CXCR1 antagonists von Biju, Purakkattle, Taveras, Arthur, Yu, Younong, Zheng, Junying, Chao, Jianhua, Rindgen, Diane, Jakway, James, Hipkin, R. William, Fossetta, James, Fan, Xuedong, Fine, Jay, Qiu, Hongchen, Merritt, J. Robert, Baldwin, John J.

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Synthesis and structure–activity relationships of new disubstituted phenyl-containing 3,4-diamino-3-cyclobutene-1,2-diones as CXCR2 receptor antagonists von Lai, Gaifa, Merritt, J. Robert, He, Zhenmin, Feng, Daming, Chao, Jianhua, Czarniecki, Michael F., Rokosz, Laura L., Stauffer, Tara M., Rindgen, Diane, Taveras, Arthur G.

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C(4)-alkyl substituted furanyl cyclobutenediones as potent, orally bioavailable CXCR2 and CXCR1 receptor antagonists von Chao, Jianhua, Taveras, Arthur G., Chao, Jianping, Aki, Cynthia, Dwyer, Michael, Yu, Younong, Purakkattle, Biju, Rindgen, Diane, Jakway, James, Hipkin, William, Fosetta, James, Fan, Xuedong, Lundell, Daniel, Fine, Jay, Minnicozzi, Michael, Phillips, Jonathan, Merritt, J. Robert

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Novel Pyrrolidine Ureas as C−C Chemokine Receptor 1 (CCR1) Antagonists von Merritt, J. Robert, Liu, Jinqi, Quadros, Elizabeth, Morris, Michelle L, Liu, Ruiyan, Zhang, Rui, Jacob, Biji, Postelnek, Jennifer, Hicks, Catherine M, Chen, Weiqing, Kimble, Earl F, Rogers, W. Lynn, O’Brien, Linda, White, Nicole, Desai, Hema, Bansal, Shalini, King, George, Ohlmeyer, Michael J, Appell, Kenneth C, Webb, Maria L

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Synthesis and structure–activity relationships of 3,4-diaminocyclobut-3-ene-1,2-dione CXCR2 antagonists von Merritt, J. Robert, Rokosz, Laura L., Nelson, Kingsley H., Kaiser, Bernd, Wang, Wei, Stauffer, Tara M., Ozgur, Lynne E., Schilling, Adriane, Li, Ge, Baldwin, John J., Taveras, Arthur G., Dwyer, Michael P., Chao, Jianping

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Novel pyrrolidine heterocycles as CCR1 antagonists von Merritt, J. Robert, James, Ray, Paradkar, Vidyadhar M., Zhang, Chongwu, Liu, Ruiyan, Liu, Jinqi, Jacob, Biji, Chiriac, Camelia, Ohlmeyer, Michael J., Quadros, Elizabeth, Wines, Pamela, Postelnek, Jennifer, Hicks, Catherine M., Chen, Weiqing, Kimble, Earl F., O’Brien, Linda, White, Nicole, Desai, Hema, Appell, Kenneth C., Webb, Maria L.

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Synthesis and structure–activity relationships of heteroaryl substituted-3,4-diamino-3-cyclobut-3-ene-1,2-dione CXCR2/CXCR1 receptor antagonists von Yu, Younong, Dwyer, Michael P., Chao, Jianping, Aki, Cynthia, Chao, Jianhua, Purakkattle, Biju, Rindgen, Diane, Bond, Richard, Mayer-Ezel, Rosemary, Jakway, James, Qiu, Hongchen, Hipkin, R. William, Fossetta, James, Gonsiorek, Waldemar, Bian, Hong, Fan, Xuedong, Terminelli, Carol, Fine, Jay, Lundell, Daniel, Merritt, J. Robert, He, Zhenmin, Lai, Gaifa, Wu, Minglang, Taveras, Arthur

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Diaminocyclobutenediones as potent and orally bioavailable CXCR2 receptor antagonists: SAR in the phenolic amide region von Aki, Cynthia, Chao, Jianping, Ferreira, Johan A., Dwyer, Michael P., Yu, Younong, Chao, Jianhua, Merritt, Robert J., Lai, Gaifa, Wu, Minglang, Hipkin, R. William, Fan, Xuedong, Gonsiorek, Waldemar, Fosseta, James, Rindgen, Diane, Fine, Jay, Lundell, Daniel, Taveras, Arthur G., Biju, Purakkattle

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n-Pentenyl Mannoside Precursors for Synthesis of the Nonamannan Component of High Mannose Glycoproteins von Merritt, J. Robert, Naisang, Elizabeth, Fraser-Reid, Bert

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n-Pentenyl Glycosides in Organic Chemistry: A Contemporary Example of Serendipity von Fraser-Reid, Bert, Udodong, Uko E., Wu, Zufan, Ottosson, Hakan, Merritt, J. Robert, Rao, C. Srinivas, Roberts, Carmichael, Madsen, Robert

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Rake prong von MERRITT ROBERT J

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n-Pentenyl glycoside methodology for rapid assembly of homoglycans exemplified with the nonasaccharide component of a high-mannose glycoprotein von Merritt, J. Robert, Fraser-Reid, Bert

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The chemistry of N-pentenyl glycosides: Synthetic, theoretical, and mechanistic ramifications von Fraser-Reid, B., Merritt, J. R., Handlon, A. L., Andrews, C. Webster

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Thiadiazoledioxides and thiadiazoleoxides as CXC- and CC-chemokine receptor ligands von TAVERAS ARTHUR G.,CHAO JIANHUA,BIJU PURAKKATTLE J.,YU YOUNONG,FINE JAY S.,HIPKIN WILLIAM,AKI CYNTHIA J.,MERRITT J. ROBERT,LI GE,BALDWIN JOHN J.,LAI GAIFA,WU MINGLANG,HECKER EVAN A

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Methods for Debrominating 4,5-Dibromopentanyl Glycosides von Merritt, J. Robert, Debenham, John S., Fraser-Reid, Bert

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Synthesis and Structure-Activity Relationships of 3,4-Diaminocyclobut-3-ene-1,2-dione CXCR2 Antagonists von Merritt, J. Robert, ., et al

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Covered stove von JR. ROBERT J. MERRITT

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